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—— (5-Methylpyrazin-2-yl)-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)methanone —— C20H24N4O4S
(5-Methylpyrazin-2-yl)-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)methanone
—— 5-chloro-2-[(3S)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C20H23ClN2O4S
5-chloro-2-[(3S)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— [5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-methoxyphenyl]methanol —— C20H25ClN2O4S
[5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-methoxyphenyl]methanol
—— 5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-1,3-dimethylbenzimidazol-2-one —— C21H25ClN4O3S
5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-1,3-dimethylbenzimidazol-2-one
—— 5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-ethylsulfanylpyrimidine —— C18H23ClN4O2S2
5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-ethylsulfanylpyrimidine
—— 5-chloro-2-[(3S)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C21H27ClN2O4S
5-chloro-2-[(3S)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— [5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-methoxyphenyl]methanol —— C20H25ClN2O4S
[5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-methoxyphenyl]methanol
—— 5-chloro-2-[(3S)-1-[(7-chloro-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C19H20Cl2N2O4S
5-chloro-2-[(3S)-1-[(7-chloro-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-propylsulfanylpyrimidine —— C19H25ClN4O2S2
5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-propylsulfanylpyrimidine
—— 5-chloro-2-[(3R)-1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C20H25ClN2O4S
5-chloro-2-[(3R)-1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-ethylsulfanylpyrimidine —— C18H23ClN4O2S2
5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-ethylsulfanylpyrimidine
—— 5-bromo-N-(4-phenyl-1,3-thiazol-2-yl)thiophene-2-sulfonamide —— C13H9BrN2O2S3
5-bromo-N-(4-phenyl-1,3-thiazol-2-yl)thiophene-2-sulfonamide
—— 5-chloro-2-[(3R)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C20H23ClN2O4S
5-chloro-2-[(3R)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3S)-1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C21H27ClN2O4S
5-chloro-2-[(3S)-1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3S)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine —— C18H21ClN2O4S2
5-chloro-2-[(3S)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3R)-1-[(2,4-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C20H25ClN2O4S
5-chloro-2-[(3R)-1-[(2,4-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-1,3-dimethylbenzimidazol-2-one —— C21H25ClN4O3S
5-[[(3R)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-1,3-dimethylbenzimidazol-2-one
—— 5-chloro-2-[(3S)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C21H27ClN2O4S
5-chloro-2-[(3S)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3S)-1-(4-chlorophenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine —— C17H18Cl2N2O4S2
5-chloro-2-[(3S)-1-(4-chlorophenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C21H27ClN2O4S
5-chloro-2-[(3R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3S)-1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C20H25ClN2O4S
5-chloro-2-[(3S)-1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3R)-1-[(7-chloro-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C19H20Cl2N2O4S
5-chloro-2-[(3R)-1-[(7-chloro-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine —— C18H21ClN2O5S2
5-chloro-2-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine
—— 5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-(2-methoxyethyl)pyrimidine —— C19H25ClN4O3S
5-[[(3S)-3-(5-chloro-3-methylsulfonylpyridin-2-yl)piperidin-1-yl]methyl]-2-(2-methoxyethyl)pyrimidine
—— 5-[[4-(Difluoromethylsulfanyl)phenyl]sulfamoyl]-2-fluorobenzoate —— C14H9F3NO4S2-
5-[[4-(Difluoromethylsulfanyl)phenyl]sulfamoyl]-2-fluorobenzoate
—— 5-[(4-Bromo-2-methylphenyl)sulfamoyl]-2-fluorobenzoate —— C14H10BrFNO4S-
5-[(4-Bromo-2-methylphenyl)sulfamoyl]-2-fluorobenzoate
—— 5-chloro-2-[(3R)-1-[(6-chloro-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine —— C19H20Cl2N2O4S
5-chloro-2-[(3R)-1-[(6-chloro-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-2-[(3R)-1-(4-chlorophenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine —— C17H18Cl2N2O4S2
5-chloro-2-[(3R)-1-(4-chlorophenyl)sulfonylpiperidin-3-yl]-3-methylsulfonylpyridine
—— 5-chloro-N-(4-phenyl-1,3-thiazol-2-yl)thiophene-2-sulfonamide —— C13H9ClN2O2S3
5-chloro-N-(4-phenyl-1,3-thiazol-2-yl)thiophene-2-sulfonamide
—— 5-[(2-Bromophenyl)sulfamoyl]-2-fluorobenzoic acid —— C13H9BrFNO4S
5-[(2-Bromophenyl)sulfamoyl]-2-fluorobenzoic acid
—— 5-[(2,5-Dimethylphenyl)sulfamoyl]-2-fluorobenzoic acid —— C15H14FNO4S
5-[(2,5-Dimethylphenyl)sulfamoyl]-2-fluorobenzoic acid
—— 5-chloro-N-(2-methoxy-5-nitrophenyl)thiophene-2-sulfonamide —— C11H9ClN2O5S2
5-chloro-N-(2-methoxy-5-nitrophenyl)thiophene-2-sulfonamide
—— 5-(2,3-Dihydro-1,4-benzodioxin-6-ylsulfamoyl)-2-fluorobenzoic acid —— C15H12FNO6S
5-(2,3-Dihydro-1,4-benzodioxin-6-ylsulfamoyl)-2-fluorobenzoic acid
—— 5-[[4-(Difluoromethylsulfanyl)phenyl]sulfamoyl]-2-fluorobenzoic acid —— C14H10F3NO4S2
5-[[4-(Difluoromethylsulfanyl)phenyl]sulfamoyl]-2-fluorobenzoic acid
—— 5-(1,3-Benzodioxol-5-ylsulfamoyl)-2-fluorobenzoate —— C14H9FNO6S-
5-(1,3-Benzodioxol-5-ylsulfamoyl)-2-fluorobenzoate
—— 5-bromo-N-(4-pyrrolidin-1-ylphenyl)thiophene-2-sulfonamide —— C14H15BrN2O2S2
5-bromo-N-(4-pyrrolidin-1-ylphenyl)thiophene-2-sulfonamide
—— (5-methylthiophen-2-yl)-[(3S)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone —— C16H17N5OS
(5-methylthiophen-2-yl)-[(3S)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone
—— 5-bromo-N-[4-(tetrazol-1-yl)phenyl]thiophene-2-sulfonamide —— C11H8BrN5O2S2
5-bromo-N-[4-(tetrazol-1-yl)phenyl]thiophene-2-sulfonamide
—— 5-(1,3-Benzodioxol-5-ylsulfamoyl)-2-fluorobenzoic acid —— C14H10FNO6S
5-(1,3-Benzodioxol-5-ylsulfamoyl)-2-fluorobenzoic acid
—— (5-methylthiophen-2-yl)-[(3R)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone —— C16H17N5OS
(5-methylthiophen-2-yl)-[(3R)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone
—— 5-bromo-2-methoxy-N-(4-pyrrolidin-1-ylphenyl)benzenesulfonamide —— C17H19BrN2O3S
5-bromo-2-methoxy-N-(4-pyrrolidin-1-ylphenyl)benzenesulfonamide
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 3,4,5-trichloropyridine-2-carboxylate —— C15H10Cl3N3O4
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 3,4,5-trichloropyridine-2-carboxylate
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3R)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone —— C20H18ClN5O3
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3R)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone
—— 5-[(3,4-Diethoxyphenyl)sulfamoyl]-2-fluorobenzoate —— C17H17FNO6S-
5-[(3,4-Diethoxyphenyl)sulfamoyl]-2-fluorobenzoate
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3S)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone —— C20H18ClN5O3
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3S)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone
—— 5-[(3-Fluorophenyl)sulfonylamino]-2-methoxybenzenesulfonamide —— C13H13FN2O5S2
5-[(3-Fluorophenyl)sulfonylamino]-2-methoxybenzenesulfonamide
—— 5-[[(E)-2-(4-chlorophenyl)ethenyl]sulfonylamino]-2-methoxybenzenesulfonamide —— C15H15ClN2O5S2
5-[[(E)-2-(4-chlorophenyl)ethenyl]sulfonylamino]-2-methoxybenzenesulfonamide
—— [(5R)-3-phenyl-4,5-dihydro-1,2-oxazol-5-yl]-[(3S)-3-[7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C21H19F3N6O2
[(5R)-3-phenyl-4,5-dihydro-1,2-oxazol-5-yl]-[(3S)-3-[7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-[7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C19H22F3N7O
(5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-[7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— [(5S)-3-phenyl-4,5-dihydro-1,2-oxazol-5-yl]-[(3R)-3-[7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C21H19F3N6O2
[(5S)-3-phenyl-4,5-dihydro-1,2-oxazol-5-yl]-[(3R)-3-[7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone