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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(4S)-4-(dimethylamino)azepan-1-yl]methyl]-2-hydroxybenzoic acid —— C16H24N2O3
5-[[(4S)-4-(dimethylamino)azepan-1-yl]methyl]-2-hydroxybenzoic acid
—— (5E)-5-benzylidene-3-[(2S)-1-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H24N2O3S2
(5E)-5-benzylidene-3-[(2S)-1-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[(3-chlorophenyl)methylidene]-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C19H21ClN2O4S
(5Z)-5-[(3-chlorophenyl)methylidene]-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— (5S)-9-(1,3-benzothiazol-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H21N3O2S
(5S)-9-(1,3-benzothiazol-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H25N3O3
(5R)-9-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H20N4O3
(5S)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one —— C18H22N2O3S3
(5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one
—— 5-(2-fluorophenyl)-N-[(2R)-2-methoxybutyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H19FN4O
5-(2-fluorophenyl)-N-[(2R)-2-methoxybutyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5E)-5-benzylidene-3-[(2S)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H24N2O3S2
(5E)-5-benzylidene-3-[(2S)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-benzylidene-3-[4-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-4-oxobutyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H26N2O3S2
(5Z)-5-benzylidene-3-[4-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-4-oxobutyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— [(5S)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-5-(cyclohexylcarbamoyl)-4,5-dihydro-1,2-oxazol-5-yl]acetic acid —— C21H25N3O6
[(5S)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-5-(cyclohexylcarbamoyl)-4,5-dihydro-1,2-oxazol-5-yl]acetic acid
—— (5R)-9-(quinolin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H22N2O2
(5R)-9-(quinolin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-4-amino-5-(2-chlorophenyl)-3-[2-(diethylamino)ethyl]-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C23H26ClN4O2+
(5R)-4-amino-5-(2-chlorophenyl)-3-[2-(diethylamino)ethyl]-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— 5-[(5E)-5-(2H-chromen-3-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]-2-hydroxybenzoic acid —— C20H13NO5S2
5-[(5E)-5-(2H-chromen-3-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]-2-hydroxybenzoic acid
—— (5R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-prop-2-enoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H20N2O5
(5R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-prop-2-enoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5Z)-5-(furan-2-ylmethylidene)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C17H20N2O5S
(5Z)-5-(furan-2-ylmethylidene)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— (5R)-9-[(5-methoxy-4-oxopyran-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H20N2O5
(5R)-9-[(5-methoxy-4-oxopyran-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(1,3-benzothiazol-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H21N3O2S
(5R)-9-(1,3-benzothiazol-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-4-amino-3-(3-imidazol-1-ylpropyl)-5-(4-methylphenyl)-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C24H24N5O2+
(5S)-4-amino-3-(3-imidazol-1-ylpropyl)-5-(4-methylphenyl)-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— (5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-(thiophen-2-ylmethylidene)-1,3-thiazolidine-2,4-dione —— C17H20N2O4S2
(5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-(thiophen-2-ylmethylidene)-1,3-thiazolidine-2,4-dione
—— (5R)-3-(2,4-dichlorophenyl)-N-(2,5-dimethoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H16Cl2N2O4
(5R)-3-(2,4-dichlorophenyl)-N-(2,5-dimethoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(4-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C21H26N2O5S
(5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(4-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5S)-3-(2,4-dichlorophenyl)-N-(2,5-dimethoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H16Cl2N2O4
(5S)-3-(2,4-dichlorophenyl)-N-(2,5-dimethoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-4-amino-3-[2-(dimethylamino)ethyl]-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C21H23N4O2+
(5S)-4-amino-3-[2-(dimethylamino)ethyl]-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— (5R)-9-[4-(4-fluorophenyl)oxane-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H25FN2O4
(5R)-9-[4-(4-fluorophenyl)oxane-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[2-(2-methylphenoxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H20N2O4
(5R)-9-[2-(2-methylphenoxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(E)-3-phenylprop-2-enylidene]-1,3-thiazolidine-2,4-dione —— C21H24N2O4S
(5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(E)-3-phenylprop-2-enylidene]-1,3-thiazolidine-2,4-dione
—— (5S)-9-[(5-methoxy-4-oxopyran-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H20N2O5
(5S)-9-[(5-methoxy-4-oxopyran-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-4-amino-3-[2-(dimethylamino)ethyl]-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C21H23N4O2+
(5R)-4-amino-3-[2-(dimethylamino)ethyl]-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— (5E)-5-benzylidene-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-1,3-thiazolidine-2,4-dione —— C20H24N2O4S
(5E)-5-benzylidene-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-1,3-thiazolidine-2,4-dione
—— (5E)-5-benzylidene-3-[(2R)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H24N2O3S2
(5E)-5-benzylidene-3-[(2R)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(4-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C21H26N2O5S
(5Z)-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(4-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— 5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one —— C18H25N5O3
5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one
—— (5R)-4-amino-3-(3-imidazol-1-ylpropyl)-5-(4-methylphenyl)-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C24H24N5O2+
(5R)-4-amino-3-(3-imidazol-1-ylpropyl)-5-(4-methylphenyl)-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— (5R)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H20N4O3
(5R)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5Z)-5-[(4-fluorophenyl)methylidene]-3-[(2R)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H23FN2O3S2
(5Z)-5-[(4-fluorophenyl)methylidene]-3-[(2R)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[(4-fluorophenyl)methylidene]-3-[(2R)-1-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H23FN2O3S2
(5Z)-5-[(4-fluorophenyl)methylidene]-3-[(2R)-1-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(2-fluorophenyl)-N-[(2S)-2-methoxybutyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H19FN4O
5-(2-fluorophenyl)-N-[(2S)-2-methoxybutyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H25N3O3
(5S)-9-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5Z)-5-[(6-methoxyquinolin-2-yl)methylidene]-3-phenyl-2-thioxoimidazolidin-4-one —— C20H15N3O2S
(5Z)-5-[(6-methoxyquinolin-2-yl)methylidene]-3-phenyl-2-thioxoimidazolidin-4-one
—— (5Z)-5-[(4-fluorophenyl)methylidene]-3-[(2S)-1-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H23FN2O3S2
(5Z)-5-[(4-fluorophenyl)methylidene]-3-[(2S)-1-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(3R)-3-(4-methoxyanilino)piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H22N4O3
5-[(3R)-3-(4-methoxyanilino)piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[3-(5-tert-butyl-1H-pyrazol-3-yl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-2-chlorobenzoate —— C16H15ClN5O2S-
5-[3-(5-tert-butyl-1H-pyrazol-3-yl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-2-chlorobenzoate
—— 5-[2-(4-fluorophenoxy)ethyl]-2-methyl[1,2,4]triazino[2,3-a]benzimidazol-3(5H)-one —— C18H15FN4O2
5-[2-(4-fluorophenoxy)ethyl]-2-methyl[1,2,4]triazino[2,3-a]benzimidazol-3(5H)-one
—— (5R)-9-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H21N3O4
(5R)-9-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C21H26N2O5S
(5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5S)-3-methyl-9-(3-methyl-1-propylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H24N4O3
(5S)-3-methyl-9-(3-methyl-1-propylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5Z)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(4-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H24N2O4S2
(5Z)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(4-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C21H26N2O5S
(5Z)-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one —— C18H25N5O3
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one