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—— 5-methyl-3-phenyl-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)-1,2-oxazole-4-carboxamide —— C19H14N4O2S
5-methyl-3-phenyl-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)-1,2-oxazole-4-carboxamide
—— (5-Tert-butyl-2-methylpyrazol-3-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C22H27F3N6O
(5-Tert-butyl-2-methylpyrazol-3-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-[(3R)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C18H19F3N4O
5-[(3R)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-[(3R)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C23H27F3N4O2
5-[(3R)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— (5-Tert-butyl-3-methylfuran-2-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C23H27F3N4O2
(5-Tert-butyl-3-methylfuran-2-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— (5S,7R)-3-chloro-N'-(3-hydroxybenzoyl)adamantane-1-carbohydrazide —— C18H21ClN2O3
(5S,7R)-3-chloro-N'-(3-hydroxybenzoyl)adamantane-1-carbohydrazide
—— 5-chloro-2-hydroxy-N'-(3-hydroxybenzoyl)benzohydrazide —— C14H11ClN2O4
5-chloro-2-hydroxy-N'-(3-hydroxybenzoyl)benzohydrazide
—— 5-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C22H23F3N4O3
5-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— [5-(furan-2-yl)-1,2-oxazol-3-yl]-[(3R)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C21H18F3N5O3
[5-(furan-2-yl)-1,2-oxazol-3-yl]-[(3R)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-[(3S)-1-[(2-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C21H23F3N4O
5-[(3S)-1-[(2-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C18H19F3N4O
5-[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C21H23F3N4O
5-[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-propan-2-yl-N-(pyridin-2-ylmethyl)pyrimidin-2-amine —— C17H19N5O
5-(3-methyl-1,2-oxazol-5-yl)-4-propan-2-yl-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
—— 5-[1-[(6-Methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C22H23F3N4O3
5-[1-[(6-Methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-[(3S)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C23H27F3N4O2
5-[(3S)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-[[4-(Furan-2-ylmethyl)piperazin-1-yl]methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole —— C23H24N6O2
5-[[4-(Furan-2-ylmethyl)piperazin-1-yl]methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole
—— 5-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C21H23F3N4O
5-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-[(3R)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C22H23F3N4O3
5-[(3R)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-[(3R)-1-(3-fluorophenyl)sulfonylpiperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C19H18F4N4O2S
5-[(3R)-1-(3-fluorophenyl)sulfonylpiperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-(3,4-dimethyl-1,2-oxazol-5-yl)-N-(3-ethenoxypropyl)-4-(furan-2-yl)pyrimidin-2-amine —— C18H20N4O3
5-(3,4-dimethyl-1,2-oxazol-5-yl)-N-(3-ethenoxypropyl)-4-(furan-2-yl)pyrimidin-2-amine
—— 5-methyl-N-[2-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-oxoethyl]furan-2-carboxamide —— C21H22F3N5O3
5-methyl-N-[2-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-oxoethyl]furan-2-carboxamide
—— [5-(furan-2-yl)-1H-pyrazol-3-yl]-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C21H19F3N6O2
[5-(furan-2-yl)-1H-pyrazol-3-yl]-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— (5-Cyclopropyl-2-methylfuran-3-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C22H23F3N4O2
(5-Cyclopropyl-2-methylfuran-3-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-(1-methylimidazol-2-yl)-N-(2-pyrazin-2-ylethyl)-4-thiophen-2-ylpyrimidin-2-amine —— C18H17N7S
5-(1-methylimidazol-2-yl)-N-(2-pyrazin-2-ylethyl)-4-thiophen-2-ylpyrimidin-2-amine
—— [5-(furan-2-yl)-1,2-oxazol-3-yl]-[(3S)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C21H18F3N5O3
[5-(furan-2-yl)-1,2-oxazol-3-yl]-[(3S)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-[[4-[2-fluoro-6-[(S)-hydroxy-(1-methylimidazol-2-yl)methyl]phenyl]piperazin-1-yl]methyl]-2-methoxyphenol —— C23H27FN4O3
5-[[4-[2-fluoro-6-[(S)-hydroxy-(1-methylimidazol-2-yl)methyl]phenyl]piperazin-1-yl]methyl]-2-methoxyphenol
—— 5-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C21H23F3N4O
5-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C21H18F3N5O3
[5-(Furan-2-yl)-1,2-oxazol-3-yl]-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-[1-[(7-Methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C22H23F3N4O3
5-[1-[(7-Methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— 5-methyl-N-[2-(5-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-2-yl)ethyl]-1H-pyrazole-4-carboxamide —— C18H17N7O
5-methyl-N-[2-(5-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5-Ethoxyfuran-2-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C20H21F3N4O3
(5-Ethoxyfuran-2-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— (5-Methyl-1-propylpyrazol-4-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C21H25F3N6O
(5-Methyl-1-propylpyrazol-4-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-chloro-2-hydroxy-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)benzamide —— C15H10ClN3O2S
5-chloro-2-hydroxy-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)benzamide
—— 5-bromo-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)pyridine-3-carboxamide —— C14H9BrN4OS
5-bromo-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)pyridine-3-carboxamide
—— (5S,7R)-3-acetamido-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)adamantane-1-carboxamide —— C21H24N4O2S
(5S,7R)-3-acetamido-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)adamantane-1-carboxamide
—— 5-bromo-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)pyridine-3-carboxamide —— C14H9BrN4OS
5-bromo-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 5-[[4-[2-fluoro-6-[(R)-hydroxy-(1-methylimidazol-2-yl)methyl]phenyl]piperazin-1-yl]methyl]-2-methoxyphenol —— C23H27FN4O3
5-[[4-[2-fluoro-6-[(R)-hydroxy-(1-methylimidazol-2-yl)methyl]phenyl]piperazin-1-yl]methyl]-2-methoxyphenol
—— 5-(1-Methylimidazol-2-yl)-2-(4-methylpiperidin-1-yl)-4-thiophen-2-ylpyrimidine —— C18H21N5S
5-(1-Methylimidazol-2-yl)-2-(4-methylpiperidin-1-yl)-4-thiophen-2-ylpyrimidine
—— 5-(1,3-benzodioxol-5-yl)-N-(2-methoxyethyl)-4-thiophen-2-ylpyrimidin-2-amine —— C18H17N3O3S
5-(1,3-benzodioxol-5-yl)-N-(2-methoxyethyl)-4-thiophen-2-ylpyrimidin-2-amine
—— 5-(1,3-benzodioxol-5-yl)-N-(3-ethoxypropyl)-4-thiophen-2-ylpyrimidin-2-amine —— C20H21N3O3S
5-(1,3-benzodioxol-5-yl)-N-(3-ethoxypropyl)-4-thiophen-2-ylpyrimidin-2-amine
—— (5-Chloro-2-hydroxyphenyl)-[4-(2,5-dimethylphenyl)sulfonylpiperazin-1-yl]methanone —— C19H21ClN2O4S
(5-Chloro-2-hydroxyphenyl)-[4-(2,5-dimethylphenyl)sulfonylpiperazin-1-yl]methanone
—— 5-chloro-1,3-dimethyl-N-[2-(5-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-2-yl)ethyl]pyrazole-4-sulfonamide —— C18H18ClN7O2S
5-chloro-1,3-dimethyl-N-[2-(5-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-2-yl)ethyl]pyrazole-4-sulfonamide
—— (5S,7R)-3-phenyl-N-(thiophen-2-ylmethyl)adamantane-1-carboxamide —— C22H25NOS
(5S,7R)-3-phenyl-N-(thiophen-2-ylmethyl)adamantane-1-carboxamide
—— 5-[4-(4-methylphenyl)sulfonylpiperazine-1-carbonyl]-1H-pyridin-2-one —— C17H19N3O4S
5-[4-(4-methylphenyl)sulfonylpiperazine-1-carbonyl]-1H-pyridin-2-one
—— (5S,7R)-3-chloro-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)adamantane-1-carboxamide —— C19H20ClN3OS
(5S,7R)-3-chloro-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)adamantane-1-carboxamide
—— 5-[(4-Ethylpiperazin-1-yl)methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole —— C20H24N6O
5-[(4-Ethylpiperazin-1-yl)methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole
—— (5-ethyl-4-methyl-1H-pyrazol-3-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C20H23F3N6O
(5-ethyl-4-methyl-1H-pyrazol-3-yl)-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-(1-methylimidazol-2-yl)-N-propan-2-yl-4-thiophen-2-ylpyrimidin-2-amine —— C15H17N5S
5-(1-methylimidazol-2-yl)-N-propan-2-yl-4-thiophen-2-ylpyrimidin-2-amine
—— 5-[4-Cyclopropyl-2-(4-methylsulfonylpiperazin-1-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole —— C16H21N5O3S
5-[4-Cyclopropyl-2-(4-methylsulfonylpiperazin-1-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole
—— 5-chloro-2-methoxy-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)benzamide —— C16H12ClN3O2S
5-chloro-2-methoxy-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)benzamide