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—— (5S)-2-(3-chloroanilino)-4,7-dioxo-N-[3-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H15ClF3N5O4
(5S)-2-(3-chloroanilino)-4,7-dioxo-N-[3-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-9-(4-amino-5-methylpyrimidin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C13H19N5O2
(5S)-9-(4-amino-5-methylpyrimidin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-2-(3,5-dichloroanilino)-N-(2,4-dimethoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H19Cl2N5O5
(5S)-2-(3,5-dichloroanilino)-N-(2,4-dimethoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 3-chloro-4,5-dimethoxybenzoate —— C18H17ClN2O6
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 3-chloro-4,5-dimethoxybenzoate
—— (5S)-N-(2,4-dimethoxyphenyl)-2-(4-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C23H23N5O6
(5S)-N-(2,4-dimethoxyphenyl)-2-(4-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-(3-chloroanilino)-4,7-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H15ClF3N5O4
(5S)-2-(3-chloroanilino)-4,7-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C23H18F3N5O5
(5S)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-2-(2,4-dichloroanilino)-N-(3-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H17Cl2N5O4
(5R)-2-(2,4-dichloroanilino)-N-(3-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(1,3-benzodioxol-5-yl)-2-(2,4-dichloroanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H15Cl2N5O5
(5S)-N-(1,3-benzodioxol-5-yl)-2-(2,4-dichloroanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-2-(3-chloroanilino)-4,7-dioxo-N-(3,4,5-trimethoxyphenyl)-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C23H22ClN5O6
(5R)-2-(3-chloroanilino)-4,7-dioxo-N-(3,4,5-trimethoxyphenyl)-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-(3-chloroanilino)-4,7-dioxo-N-[3-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H15ClF3N5O3
(5S)-2-(3-chloroanilino)-4,7-dioxo-N-[3-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-2-(3,5-dichloroanilino)-4,7-dioxo-N-[3-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H14Cl2F3N5O3
(5R)-2-(3,5-dichloroanilino)-4,7-dioxo-N-[3-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(2-methoxyphenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H18F3N5O4
(5S)-N-(2-methoxyphenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 4H-thieno[3,2-c]chromene-2-carboxylate —— C21H16N2O5S
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 4H-thieno[3,2-c]chromene-2-carboxylate
—— [5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enoate —— C21H16ClNO5
[5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enoate
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-ethoxy-3-methoxyphenyl)prop-2-enoate —— C21H22N2O6
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-ethoxy-3-methoxyphenyl)prop-2-enoate
—— (5S)-2-(3,5-dichloroanilino)-N-(4-fluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C20H14Cl2FN5O3
(5S)-2-(3,5-dichloroanilino)-N-(4-fluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-(4-nitrophenoxy)acetate —— C18H13ClN2O6
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-(4-nitrophenoxy)acetate
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 4,5-dihydrobenzo[g][1]benzothiole-2-carboxylate —— C22H18N2O4S
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 4,5-dihydrobenzo[g][1]benzothiole-2-carboxylate
—— (5R)-3-methyl-7-[(2-naphthalen-1-ylpyrimidin-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C22H22N4O2
(5R)-3-methyl-7-[(2-naphthalen-1-ylpyrimidin-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-nitrophenoxy)acetate —— C17H15N3O7
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-nitrophenoxy)acetate
—— (5S)-3-methyl-7-[(2-naphthalen-1-ylpyrimidin-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C22H22N4O2
(5S)-3-methyl-7-[(2-naphthalen-1-ylpyrimidin-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-2-(4,6-dimethoxypyrimidin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O4
(5R)-2-(4,6-dimethoxypyrimidin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-Carboxylatopropylsulfamoyl)-2-methoxybenzoate —— C12H13NO7S-2
5-(3-Carboxylatopropylsulfamoyl)-2-methoxybenzoate
—— (5S)-2-(4,6-dimethoxypyrimidin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O4
(5S)-2-(4,6-dimethoxypyrimidin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-thieno[2,3-d]pyrimidin-4-ylsulfanylacetate —— C17H14N4O4S2
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-thieno[2,3-d]pyrimidin-4-ylsulfanylacetate
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-chloro-4,5-dimethoxyphenyl)prop-2-enoate —— C20H19ClN2O6
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-chloro-4,5-dimethoxyphenyl)prop-2-enoate
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-(3-chlorophenoxy)acetate —— C18H13Cl2NO4
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-(3-chlorophenoxy)acetate
—— (5R)-9-[4-(dimethylamino)pyrimidin-2-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H21N5O2
(5R)-9-[4-(dimethylamino)pyrimidin-2-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H19FN4O2
(5R)-7-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H19FN4O2
(5S)-7-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-ethyl-N-[(2R)-2-pyridin-3-yloxypropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H19N5O
5-ethyl-N-[(2R)-2-pyridin-3-yloxypropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone —— C21H25N5O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone
—— (5R)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane —— C20H25FN4O
(5R)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone —— C21H25N5O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone
—— 5-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methylsulfanyl]-2-indol-3-ylidene-3H-1,3,4-oxadiazole —— C20H16ClN3O3S
5-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methylsulfanyl]-2-indol-3-ylidene-3H-1,3,4-oxadiazole
—— 5-ethyl-N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine —— C16H23N7
5-ethyl-N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-chloro-2-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine —— C18H25ClN6
5-chloro-2-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine
—— 5-[[1-(2,5-Dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole —— C20H20N6OS
5-[[1-(2,5-Dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole
—— 5-chloro-2-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine —— C18H25ClN6
5-chloro-2-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine
—— 5-ethyl-2-methyl-4-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine —— C20H31N7
5-ethyl-2-methyl-4-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine
—— 5-ethyl-2-methyl-4-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine —— C20H31N7
5-ethyl-2-methyl-4-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine
—— 5-[[(2S)-oxolan-2-yl]methylsulfanyl]-4-prop-2-enyl-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one —— C19H24N2O2S2
5-[[(2S)-oxolan-2-yl]methylsulfanyl]-4-prop-2-enyl-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
—— (5S)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane —— C20H25FN4O
(5S)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-[[(2R)-oxolan-2-yl]methylsulfanyl]-4-prop-2-enyl-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one —— C19H24N2O2S2
5-[[(2R)-oxolan-2-yl]methylsulfanyl]-4-prop-2-enyl-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
—— 5-[(4,6-Diamino-1,3,5-triazin-2-yl)methylsulfanyl]-4-prop-2-enyl-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one —— C18H21N7OS2
5-[(4,6-Diamino-1,3,5-triazin-2-yl)methylsulfanyl]-4-prop-2-enyl-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
—— 5,5-diethyl-3-[[(2S)-oxolan-2-yl]methyl]imidazolidine-2,4-dione —— C12H20N2O3
5,5-diethyl-3-[[(2S)-oxolan-2-yl]methyl]imidazolidine-2,4-dione
—— 5-[(2R)-2-pyridin-2-ylpyrrolidine-1-carbonyl]-1H-pyrazin-2-one —— C14H14N4O2
5-[(2R)-2-pyridin-2-ylpyrrolidine-1-carbonyl]-1H-pyrazin-2-one
—— (5S)-2-(7-chloroquinolin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H20ClN3O
(5S)-2-(7-chloroquinolin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C19H24N6O2
5-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one