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—— (5S)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H24N4O3
(5S)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-Cyclopropylimino-3,3-dimethylcyclohexan-1-one —— C11H17NO
5-Cyclopropylimino-3,3-dimethylcyclohexan-1-one
—— (5-ethyl-4-methyl-1H-pyrazol-3-yl)-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone —— C17H28N4O2
(5-ethyl-4-methyl-1H-pyrazol-3-yl)-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone
—— [5-(diethylaminomethyl)-2-methylfuran-3-yl]-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C17H28N2O4
[5-(diethylaminomethyl)-2-methylfuran-3-yl]-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— (5S)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H23N3O3
(5S)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C15H17FN4O2
5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5R)-7-(2-chloro-4-pyrazol-1-ylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H17ClN4O3
(5R)-7-(2-chloro-4-pyrazol-1-ylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(5-acetyl-6-methyl-2-oxo-1H-pyridine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H23N3O5
(5S)-9-(5-acetyl-6-methyl-2-oxo-1H-pyridine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[1-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H17N5O3
5-[1-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[2-[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one —— C20H24N4O4
5-[2-[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one
—— 5-[(3R)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]-5-oxopentanamide —— C21H32N4O2
5-[(3R)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]-5-oxopentanamide
—— (5S)-9-[(3,4,5-trifluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H18F3NO2
(5S)-9-[(3,4,5-trifluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H24N4O3
(5R)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(1S)-cyclohex-3-en-1-yl]methyl]-2-[(4,4-difluoropiperidin-1-yl)methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine —— C20H30F2N4
5-[[(1S)-cyclohex-3-en-1-yl]methyl]-2-[(4,4-difluoropiperidin-1-yl)methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine
—— (5S)-3-methyl-9-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H24N4O2S
(5S)-3-methyl-9-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(2,1,3-benzoxadiazol-5-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H18N4O3
(5R)-9-(2,1,3-benzoxadiazol-5-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H23N3O3
(5R)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[3-(6-oxo-1H-pyridazin-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H18N4O4
(5R)-9-[3-(6-oxo-1H-pyridazin-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C16H18ClNO5
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— 5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C15H17FN4O2
5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5S)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O3S
(5S)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C16H18ClNO5
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— 5-[(3S)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]-5-oxopentanamide —— C21H32N4O2
5-[(3S)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]-5-oxopentanamide
—— (5S)-9-(1-benzylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O3
(5S)-9-(1-benzylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[(3,4,5-trifluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H18F3NO2
(5R)-9-[(3,4,5-trifluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C17H20F2N4O2
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5S)-9-[5-(methylsulfanylmethyl)furan-2-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H20N2O4S
(5S)-9-[5-(methylsulfanylmethyl)furan-2-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— [5-(diethylaminomethyl)-2-methylfuran-3-yl]-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C17H28N2O4
[5-(diethylaminomethyl)-2-methylfuran-3-yl]-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— (5aS,10aR)-2-[(1S,5R,6R)-6-(2,4-dihydroxybenzoyl)-5-(2,4-dihydroxyphenyl)-3-methylcyclohex-2-en-1-yl]-1,3,5a,8-tetrahydroxy-10a-(3-methylbut-2-enyl)-[1]benzofuro[3,2-b]chromen-11-one —— C40H36O12
(5aS,10aR)-2-[(1S,5R,6R)-6-(2,4-dihydroxybenzoyl)-5-(2,4-dihydroxyphenyl)-3-methylcyclohex-2-en-1-yl]-1,3,5a,8-tetrahydroxy-10a-(3-methylbut-2-enyl)-[1]benzofuro[3,2-b]chromen-11-one
—— 5-[1-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H17N5O3
5-[1-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(3,3,3-trifluoropropyl)pyridazin-3-one —— C13H19F3N4O2
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(3,3,3-trifluoropropyl)pyridazin-3-one
—— (5S)-3-methyl-9-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H25N3O3
(5S)-3-methyl-9-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O3S
(5R)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(1,3-benzothiazol-2-yl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H22FN3OS
(5R)-2-(1,3-benzothiazol-2-yl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-(3,3,3-trifluoropropyl)pyridazin-3-one —— C13H19F3N4O2
5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-(3,3,3-trifluoropropyl)pyridazin-3-one
—— 5-[[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine —— C18H21N5O
5-[[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine
—— (5R)-2-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H27N5O3
(5R)-2-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[[4-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H20F3NO2
(5R)-9-[[4-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[[4-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H20F3NO2
(5S)-9-[[4-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19FN6O
5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S)-2-(1,3-benzothiazol-2-yl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H22FN3OS
(5S)-2-(1,3-benzothiazol-2-yl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(3-oxo-4H-quinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O3
(5S)-9-[(3-oxo-4H-quinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20N4O3
(5S)-9-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3S)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine —— C21H27N5
5-[[(3S)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine
—— 5-[[4-[(3-fluorophenyl)methyl]piperazin-1-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C21H28FN5O
5-[[4-[(3-fluorophenyl)methyl]piperazin-1-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— 5-(2-fluorophenyl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H17FN6
5-(2-fluorophenyl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(2-fluorophenyl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H17FN6
5-(2-fluorophenyl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-9-[(3-oxo-4H-quinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O3
(5R)-9-[(3-oxo-4H-quinoxalin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C20H20FN3O
5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— 5-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine —— C18H21N5O
5-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine