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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5,5-Dimethyl-2-(3-propan-2-yloxypropylcarbamoylamino)-4,7-dihydrothieno[2,3-c]pyran-3-carboxamide —— C17H27N3O4S
5,5-Dimethyl-2-(3-propan-2-yloxypropylcarbamoylamino)-4,7-dihydrothieno[2,3-c]pyran-3-carboxamide
—— 5-propyl-7-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C20H25N5O
5-propyl-7-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-[[(3R)-3-[(2-fluorophenoxy)methyl]piperidin-1-yl]methyl]-2-methoxyphenol —— C20H24FNO3
5-[[(3R)-3-[(2-fluorophenoxy)methyl]piperidin-1-yl]methyl]-2-methoxyphenol
—— (5S)-9-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22N4O4
(5S)-9-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-ethyl-N-methyl-N-[(3S)-1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide —— C21H30N4O
5-ethyl-N-methyl-N-[(3S)-1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
—— [(5S)-5-(cyclohexylcarbamoyl)-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazol-5-yl]acetic acid —— C18H21N3O6
[(5S)-5-(cyclohexylcarbamoyl)-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazol-5-yl]acetic acid
—— 5-chloro-2-methylsulfanyl-N-quinolin-8-ylpyrimidine-4-carboxamide —— C15H11ClN4OS
5-chloro-2-methylsulfanyl-N-quinolin-8-ylpyrimidine-4-carboxamide
—— 5-ethyl-1-(pyridin-4-ylmethyl)-1H-indole-2,3-dione —— C16H14N2O2
5-ethyl-1-(pyridin-4-ylmethyl)-1H-indole-2,3-dione
—— 5-ethyl-N-methyl-N-[(3R)-1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide —— C21H30N4O
5-ethyl-N-methyl-N-[(3R)-1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
—— (5S)-3-methyl-7-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H24N2O4
(5S)-3-methyl-7-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-5-(2,3-difluorophenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C19H13F2N3O2
(5R)-5-(2,3-difluorophenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— 5-[[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]quinoxaline —— C22H23N5
5-[[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]quinoxaline
—— (5R)-9-[2-(1-methylindol-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O3
(5R)-9-[2-(1-methylindol-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-(3,4-dimethylphenyl)-1-(4-fluorophenyl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one —— C19H15FN4O
5-(3,4-dimethylphenyl)-1-(4-fluorophenyl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one
—— (5S)-7-(2-benzyl-1,3-thiazole-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H19N3O3S
(5S)-7-(2-benzyl-1,3-thiazole-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(3R)-1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C15H20ClN3O2S
5-[(3R)-1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-[[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]-N,N-dimethyl-1,3-thiazol-2-amine —— C19H25N5S
5-[[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]-N,N-dimethyl-1,3-thiazol-2-amine
—— (5R)-9-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22N4O4
(5R)-9-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-cyclohexyl-1-(4-fluorophenyl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one —— C17H17FN4O
5-cyclohexyl-1-(4-fluorophenyl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one
—— (5R)-9-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H21N5O3
(5R)-9-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]quinoxaline —— C22H23N5
5-[[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]quinoxaline
—— 5-{[5-(3-ethoxy-4-methoxyphenyl)-2H-tetrazol-2-yl]methyl}-1H-tetrazole —— C12H14N8O2
5-{[5-(3-ethoxy-4-methoxyphenyl)-2H-tetrazol-2-yl]methyl}-1H-tetrazole
—— (5S)-9-[2-(1-methylindol-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O3
(5S)-9-[2-(1-methylindol-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3S)-1-(2-methyl-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C19H21N7O
5-[(3S)-1-(2-methyl-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5Z)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C20H24N2O5S
(5Z)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5S)-5-[2-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one —— C20H24N6O2
(5S)-5-[2-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one
—— 5-[(3S)-1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C15H20ClN3O2S
5-[(3S)-1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-[(3R)-1-(2-methyl-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C19H21N7O
5-[(3R)-1-(2-methyl-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5R)-7-(2-benzyl-1,3-thiazole-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H19N3O3S
(5R)-7-(2-benzyl-1,3-thiazole-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5,6-dimethyl-3-[(3R)-3-(4-propan-2-ylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H29N3O2
5,6-dimethyl-3-[(3R)-3-(4-propan-2-ylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5,5-dimethyl-2-[[(2R)-oxolan-2-yl]methylcarbamoylamino]-4,7-dihydrothieno[2,3-c]pyran-3-carboxamide —— C16H23N3O4S
5,5-dimethyl-2-[[(2R)-oxolan-2-yl]methylcarbamoylamino]-4,7-dihydrothieno[2,3-c]pyran-3-carboxamide
—— 5-[(3S)-2-oxospiro[1H-indole-3,3'-piperidine]-1'-carbonyl]pyridine-2-carbonitrile —— C19H16N4O2
5-[(3S)-2-oxospiro[1H-indole-3,3'-piperidine]-1'-carbonyl]pyridine-2-carbonitrile
—— 5,6-dimethyl-7-phenyl-3-(1,3-thiazol-2-yl)-3,7-dihydro-4H-pyrrolo[2,3-d]pyrimidin-4-imine —— C17H15N5S
5,6-dimethyl-7-phenyl-3-(1,3-thiazol-2-yl)-3,7-dihydro-4H-pyrrolo[2,3-d]pyrimidin-4-imine
—— 5-(3-Ethoxy-4-methoxyphenyl)-2-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-ylmethyl)tetrazole —— C12H13N8O2-
5-(3-Ethoxy-4-methoxyphenyl)-2-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-ylmethyl)tetrazole
—— (5S)-5-(4-nitrophenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C19H14N4O4
(5S)-5-(4-nitrophenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— 5-fluoro-3-methyl-2-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-indole —— C19H20FN3
5-fluoro-3-methyl-2-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-indole
—— [5-[[(6R)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]methyl]-2-ethoxyphenyl]methanol —— C18H28N2O4
[5-[[(6R)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]methyl]-2-ethoxyphenyl]methanol
—— (5S)-3-methyl-7-(2-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H22N4O3
(5S)-3-methyl-7-(2-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(2,2-dimethylpropyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,9-diazaspiro[4.5]decane —— C18H32N4O2S
(5S)-9-(2,2-dimethylpropyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,9-diazaspiro[4.5]decane
—— 5,6-dimethyl-N-(2-methylpropyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine —— C17H21N5
5,6-dimethyl-N-(2-methylpropyl)-7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
—— 5,6-Dimethyl-3-(2-methylpropyl)-7-(pyridin-3-ylmethyl)pyrrolo[2,3-d]pyrimidin-3-ium-4-amine —— C18H24N5+
5,6-Dimethyl-3-(2-methylpropyl)-7-(pyridin-3-ylmethyl)pyrrolo[2,3-d]pyrimidin-3-ium-4-amine
—— 5-ethyl-2-methyl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]pyrimidine —— C22H31N5
5-ethyl-2-methyl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]pyrimidine
—— 5-[(2S)-1-[(3-fluoropyridin-2-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C18H17FN4O
5-[(2S)-1-[(3-fluoropyridin-2-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— (5R)-5-(chloromethyl)-4,5-dihydro-1,3-oxazol-2-amine —— C4H7ClN2O
(5R)-5-(chloromethyl)-4,5-dihydro-1,3-oxazol-2-amine
—— (5S)-3-methyl-7-[3-(2-methylimidazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H22N4O2
(5S)-3-methyl-7-[3-(2-methylimidazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methyl-6-[4-(propan-2-yl)benzyl]-2-propyl[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one —— C19H24N4O
5-methyl-6-[4-(propan-2-yl)benzyl]-2-propyl[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one
—— 5,6-dimethyl-7-(2-methylpropyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine —— C12H18N4
5,6-dimethyl-7-(2-methylpropyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
—— (5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C20H24N2O5S
(5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5Z)-5-[(8-ethoxyquinolin-2-yl)methylidene]-3-phenyl-2-thioxoimidazolidin-4-one —— C21H17N3O2S
(5Z)-5-[(8-ethoxyquinolin-2-yl)methylidene]-3-phenyl-2-thioxoimidazolidin-4-one
—— 5,6-dimethyl-3-[(3S)-3-(4-propan-2-ylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H29N3O2
5,6-dimethyl-3-[(3S)-3-(4-propan-2-ylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one