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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-3-methyl-9-[2-(N-methylanilino)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H25N3O3
(5R)-3-methyl-9-[2-(N-methylanilino)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-[[3-(2-methylpropyl)imidazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H26N4O2
(5R)-3-methyl-9-[[3-(2-methylpropyl)imidazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[4-(1H-pyrazol-4-yl)butanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H20N4O3
(5R)-9-[4-(1H-pyrazol-4-yl)butanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O5
(5R)-7-[3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[2-(2-methylphenoxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H20N2O4
(5S)-9-[2-(2-methylphenoxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(1-ethyl-4,6-dimethyl-2-oxopyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H25N3O4
(5S)-9-(1-ethyl-4,6-dimethyl-2-oxopyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]quinoxaline —— C22H23N5
5-[[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]quinoxaline
—— 5-[(3S)-3-(4-methoxyanilino)piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H22N4O3
5-[(3S)-3-(4-methoxyanilino)piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole —— C19H26N4OS
5-[[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole
—— (5R)-9-(1-ethyl-4,6-dimethyl-2-oxopyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H25N3O4
(5R)-9-(1-ethyl-4,6-dimethyl-2-oxopyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-5-(3,4-dimethoxyphenyl)-3,5-dihydrotetrazolo[1,5-c]quinazoline —— C16H15N5O2
(5R)-5-(3,4-dimethoxyphenyl)-3,5-dihydrotetrazolo[1,5-c]quinazoline
—— 5-[[(3S)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]quinoxaline —— C22H23N5
5-[[(3S)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]quinoxaline
—— (5S)-2,4,8-triamino-5-(3-bromophenyl)-5H-chromeno[2,3-b]pyridine-3-carbonitrile —— C19H14BrN5O
(5S)-2,4,8-triamino-5-(3-bromophenyl)-5H-chromeno[2,3-b]pyridine-3-carbonitrile
—— (5R)-5-(1H-imidazol-5-ylmethyl)-3-(oxan-4-yl)-7-(1H-pyrrolo[2,3-b]pyridin-6-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C21H24N8O
(5R)-5-(1H-imidazol-5-ylmethyl)-3-(oxan-4-yl)-7-(1H-pyrrolo[2,3-b]pyridin-6-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— (5R)-2-(1,3-benzoxazol-2-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C24H27N3O4
(5R)-2-(1,3-benzoxazol-2-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H26N4O4
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(methoxymethyl)-3-[[(3R)-3-[2-[3-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C19H24F3N3O2
5-(methoxymethyl)-3-[[(3R)-3-[2-[3-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-tert-butyl-4-[[(5R)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]methyl]furan-2-carboxamide —— C18H27N3O4
5-tert-butyl-4-[[(5R)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]methyl]furan-2-carboxamide
—— (5R)-9-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H18ClN3O4
(5R)-9-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(3S)-3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C19H21N3O5
5-[(3S)-3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5R)-3-methyl-9-[2-(4-propoxyphenoxy)ethyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H28N2O4
(5R)-3-methyl-9-[2-(4-propoxyphenoxy)ethyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[3-[(3R)-3-anilinopiperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C20H26N4O2
5-[3-[(3R)-3-anilinopiperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— 5-[(4-Ethoxyphenyl)sulfonylamino]-2-methyl-1-benzofuran-3-carboxylate —— C18H16NO6S-
5-[(4-Ethoxyphenyl)sulfonylamino]-2-methyl-1-benzofuran-3-carboxylate
—— (5R)-9-[3-(1H-indol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O3
(5R)-9-[3-(1H-indol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-[2-(4-propoxyphenoxy)ethyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H28N2O4
(5S)-3-methyl-9-[2-(4-propoxyphenoxy)ethyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-[4-(trifluoromethyl)phenyl]sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H19F3N2O4S
(5S)-3-methyl-9-[4-(trifluoromethyl)phenyl]sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-2-ethylsulfonyl-9-[(3-methylphenyl)methyl]-2,9-diazaspiro[4.5]decane —— C18H28N2O2S
(5R)-2-ethylsulfonyl-9-[(3-methylphenyl)methyl]-2,9-diazaspiro[4.5]decane
—— 5-{[(2,5-Dichlorophenyl)sulfonyl]amino}-2-methyl-1-benzofuran-3-carboxylic acid —— C16H11Cl2NO5S
5-{[(2,5-Dichlorophenyl)sulfonyl]amino}-2-methyl-1-benzofuran-3-carboxylic acid
—— (5R)-9-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H21N3O3S
(5R)-9-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-tert-butyl-4-[[(5S)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]methyl]furan-2-carboxamide —— C18H27N3O4
5-tert-butyl-4-[[(5S)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]methyl]furan-2-carboxamide
—— 5-[2-(4-chlorophenoxy)ethyl]-2-methyl[1,2,4]triazino[2,3-a]benzimidazol-3(5H)-one —— C18H15ClN4O2
5-[2-(4-chlorophenoxy)ethyl]-2-methyl[1,2,4]triazino[2,3-a]benzimidazol-3(5H)-one
—— 5-[[(3R)-3-[2-[3-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H21F3N4O2
5-[[(3R)-3-[2-[3-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-[(3S)-3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C20H23N3O4
5-[(3S)-3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— 5-[(3R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C20H23N3O4
5-[(3R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H26N4O4
(5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-3-methyl-7-(2-morpholin-4-ylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H21N5O4
(5S)-3-methyl-7-(2-morpholin-4-ylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[3-(3-oxo-4H-quinoxalin-2-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O4
(5R)-9-[3-(3-oxo-4H-quinoxalin-2-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(3-hydroxy-2-methylbenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H20N2O4
(5R)-9-(3-hydroxy-2-methylbenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C14H20N2O3
(5R)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-(1H-imidazol-5-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C13H20N4O2
(5S)-9-(1H-imidazol-5-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3R)-3-[[(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one —— C17H22N8O
5-[(3R)-3-[[(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one
—— (5R)-3-methyl-7-(2-morpholin-4-ylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H21N5O4
(5R)-3-methyl-7-(2-morpholin-4-ylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-(1H-imidazol-5-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C13H20N4O2
(5R)-9-(1H-imidazol-5-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C14H20N2O3
(5S)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(3S)-3-[[(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one —— C17H22N8O
5-[(3S)-3-[[(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one
—— (5S)-9-(1,6-dimethyl-4-oxoquinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H21N3O4
(5S)-9-(1,6-dimethyl-4-oxoquinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[3-(3-oxo-4H-quinoxalin-2-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O4
(5S)-9-[3-(3-oxo-4H-quinoxalin-2-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-7-(3-methyltriazolo[4,5-b]pyridine-6-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H16N6O3
(5S)-3-methyl-7-(3-methyltriazolo[4,5-b]pyridine-6-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyrazin-2-one —— C19H22N4O2
5-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyrazin-2-one
—— (5S)-3-methyl-7-[(2-methyl-7-oxo-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H18N6O3
(5S)-3-methyl-7-[(2-methyl-7-oxo-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one