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—— (5S)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3S
(5S)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H28N2O4
(5S)-2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-methoxy-3-methyl-2-[[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1H-indole —— C22H27N3O2
5-methoxy-3-methyl-2-[[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1H-indole
—— (5E)-5-(2-morpholin-4-yl-2-sulfanylideneethylidene)pyrrolidin-2-one —— C10H14N2O2S
(5E)-5-(2-morpholin-4-yl-2-sulfanylideneethylidene)pyrrolidin-2-one
—— 5-(3-amino-4-cyano-1H-pyrazol-5-yl)pentyl-[(3,4-dichlorophenyl)methyl]azanium —— C16H20Cl2N5+
5-(3-amino-4-cyano-1H-pyrazol-5-yl)pentyl-[(3,4-dichlorophenyl)methyl]azanium
—— 5-[[2-[(dimethylamino)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C19H29N7O
5-[[2-[(dimethylamino)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (5R)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3S
(5R)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(3-methyl-4-oxoquinazoline-7-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H20N4O4
(5R)-9-(3-methyl-4-oxoquinazoline-7-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C13H16ClN3O4
(5R)-7-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[3-(4-oxoquinazolin-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O4
(5S)-9-[3-(4-oxoquinazolin-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H25ClN4O2
(5S)-9-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[3-[2-[(4R)-2,2-dimethyloxan-4-yl]imidazol-1-yl]propyl]-2H-tetrazole —— C14H22N6O
5-[3-[2-[(4R)-2,2-dimethyloxan-4-yl]imidazol-1-yl]propyl]-2H-tetrazole
—— (5R)-9-(4-methoxy-2-methylbenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H22N2O4
(5R)-9-(4-methoxy-2-methylbenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H21N3O3S
(5S)-9-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-2-[3-(1H-indol-3-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N3O2
(5R)-2-[3-(1H-indol-3-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C15H23N5O2
5-[[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R)-9-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H28N4O2
(5R)-9-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-7-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H21N3O3
(5S)-3-methyl-7-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl]-N-[(3R)-pyrrolidin-3-yl]pyridin-2-amine —— C19H21N5O2
5-[3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl]-N-[(3R)-pyrrolidin-3-yl]pyridin-2-amine
—— (5S)-9-[(1-ethylimidazol-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H23N3O2
(5S)-9-[(1-ethylimidazol-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C20H25FN4O
(5R)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-[[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C15H23N5O2
5-[[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C20H25FN4O
(5S)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— (5S)-2,2,6,6-tetramethyl-4,5-diphenyl-1,3-diazabicyclo[3.1.0]hex-3-ene —— C20H22N2
(5S)-2,2,6,6-tetramethyl-4,5-diphenyl-1,3-diazabicyclo[3.1.0]hex-3-ene
—— (5S)-9-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H28N4O2
(5S)-9-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H17N5O3
(5R)-9-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H17N5O3
(5S)-9-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N2O6
(5S)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-phenyl-2-[(1S)-1-pyrrolidin-1-ylethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C18H19N3OS
5-phenyl-2-[(1S)-1-pyrrolidin-1-ylethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5R)-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H21N3O3
(5R)-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-3-methyl-7-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H20N4O4
(5S)-3-methyl-7-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-(imidazo[1,2-a]pyridin-2-ylmethylsulfanyl)-N-(3-methoxyphenyl)-1,3,4-thiadiazol-2-amine —— C17H15N5OS2
5-(imidazo[1,2-a]pyridin-2-ylmethylsulfanyl)-N-(3-methoxyphenyl)-1,3,4-thiadiazol-2-amine
—— (5R)-3-methyl-7-(1H-pyrrole-2-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H15N3O3
(5R)-3-methyl-7-(1H-pyrrole-2-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-7-[3-(5-phenyltetrazol-2-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H20N6O3
(5S)-3-methyl-7-[3-(5-phenyltetrazol-2-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-phenyl-2-[(1S)-1-pyrrolidin-1-ium-1-ylethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C18H20N3OS+
5-phenyl-2-[(1S)-1-pyrrolidin-1-ium-1-ylethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-(Cycloheptyliminomethyl)-1,3-diethyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C16H25N3O2S
5-(Cycloheptyliminomethyl)-1,3-diethyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-cyano-4-(3-fluorophenyl)-2-methyl-N-(2-methylphenyl)-6-prop-2-enylsulfanylpyridine-3-carboxamide —— C24H20FN3OS
5-cyano-4-(3-fluorophenyl)-2-methyl-N-(2-methylphenyl)-6-prop-2-enylsulfanylpyridine-3-carboxamide
—— (5R)-9-(3-pyridin-4-yl-1H-pyrazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H19N5O3
(5R)-9-(3-pyridin-4-yl-1H-pyrazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-phenyl-2-[(1S)-1-(2-phenylethylamino)ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C22H21N3OS
5-phenyl-2-[(1S)-1-(2-phenylethylamino)ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-[2-[(3R)-3-(4-methoxyanilino)piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C19H24N4O3
5-[2-[(3R)-3-(4-methoxyanilino)piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— (5R)-3-methyl-7-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H20N4O4
(5R)-3-methyl-7-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-phenyl-2-[(1R)-1-(2-phenylethylamino)ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C22H21N3OS
5-phenyl-2-[(1R)-1-(2-phenylethylamino)ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-[2-[(3S)-3-(4-methoxyanilino)piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C19H24N4O3
5-[2-[(3S)-3-(4-methoxyanilino)piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[(3S)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyridazin-3-one —— C15H21N5O2
5-[(3S)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyridazin-3-one
—— 5-bromo-N-[(Z)-(1-butyl-2-oxoindol-3-ylidene)amino]-2-hydroxybenzamide —— C19H18BrN3O3
5-bromo-N-[(Z)-(1-butyl-2-oxoindol-3-ylidene)amino]-2-hydroxybenzamide
—— (5E)-3-butyl-5-[(4-phenylmethoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C21H22N2O2S
(5E)-3-butyl-5-[(4-phenylmethoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5E)-3-butyl-5-[(3-phenylmethoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C21H22N2O2S
(5E)-3-butyl-5-[(3-phenylmethoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— 5-piperidin-1-ylsulfonyl-2-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]pyridin-1-ium —— C18H24N3O2S2+
5-piperidin-1-ylsulfonyl-2-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]pyridin-1-ium
—— 5-methoxy-3-methyl-N-[3-[(E)-2-pyridin-2-ylethenyl]phenyl]-1-benzofuran-2-carboxamide —— C24H20N2O3
5-methoxy-3-methyl-N-[3-[(E)-2-pyridin-2-ylethenyl]phenyl]-1-benzofuran-2-carboxamide
—— 5-piperidin-1-ylsulfonyl-2-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]pyridine —— C18H23N3O2S2
5-piperidin-1-ylsulfonyl-2-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]pyridine