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—— 5-ethyl-N-[6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyridin-2-yl]-1,3,4-thiadiazol-2-amine —— C20H24N6S
5-ethyl-N-[6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyridin-2-yl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[6-(1-pyrazin-2-ylpiperidin-4-yl)pyridin-2-yl]-1,3,4-thiadiazol-2-amine —— C18H21N7S
5-ethyl-N-[6-(1-pyrazin-2-ylpiperidin-4-yl)pyridin-2-yl]-1,3,4-thiadiazol-2-amine
—— 5-[[(6S)-4-ethyl-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C13H20N4O2
5-[[(6S)-4-ethyl-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— (5-methyl-1H-indazol-3-yl)-[(3R)-3-[6-[(5-methyl-1H-pyrazol-3-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone —— C23H25N7O
(5-methyl-1H-indazol-3-yl)-[(3R)-3-[6-[(5-methyl-1H-pyrazol-3-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone
—— 5-[[(6S)-4-(cyclopentanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C17H24N4O3
5-[[(6S)-4-(cyclopentanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— (5-methyl-1H-indazol-3-yl)-[(3S)-3-[6-[(5-methyl-1H-pyrazol-3-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone —— C23H25N7O
(5-methyl-1H-indazol-3-yl)-[(3S)-3-[6-[(5-methyl-1H-pyrazol-3-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone
—— 5-ethyl-N-[6-(1-pyrimidin-4-ylpiperidin-4-yl)pyridin-2-yl]-1,3,4-thiadiazol-2-amine —— C18H21N7S
5-ethyl-N-[6-(1-pyrimidin-4-ylpiperidin-4-yl)pyridin-2-yl]-1,3,4-thiadiazol-2-amine
—— [5-[[(3S)-1-methylpiperidin-3-yl]methyl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C16H24N4O
[5-[[(3S)-1-methylpiperidin-3-yl]methyl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— 5-[[(6R)-4-[(2-fluorophenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C18H21FN4O2
5-[[(6R)-4-[(2-fluorophenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6S)-4-[(2-fluorophenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C18H21FN4O2
5-[[(6S)-4-[(2-fluorophenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— [5-[[(3R)-1-methylpiperidin-3-yl]methyl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C16H24N4O
[5-[[(3R)-1-methylpiperidin-3-yl]methyl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— 5-[[(6R)-4-(2-methylpyrazole-3-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H20N6O3
5-[[(6R)-4-(2-methylpyrazole-3-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6R)-4-[(3-methylimidazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6R)-4-[(3-methylimidazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6R)-4-(1,3-thiazole-4-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C15H17N5O3S
5-[[(6R)-4-(1,3-thiazole-4-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6S)-4-(1,3-thiazole-4-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C15H17N5O3S
5-[[(6S)-4-(1,3-thiazole-4-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-methyl-N-[2-methyl-6-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H22N8S
5-methyl-N-[2-methyl-6-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-[[(6R)-4-(cyclohexanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C18H26N4O3
5-[[(6R)-4-(cyclohexanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6R)-4-(pyridin-3-ylmethyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C17H21N5O2
5-[[(6R)-4-(pyridin-3-ylmethyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6S)-4-(cyclohexanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C18H26N4O3
5-[[(6S)-4-(cyclohexanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6S)-4-(pyridin-3-ylmethyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C17H21N5O2
5-[[(6S)-4-(pyridin-3-ylmethyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6R)-4-[(2-methylpyrazol-3-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6R)-4-[(2-methylpyrazol-3-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6R)-4-[(1-methylpyrazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6R)-4-[(1-methylpyrazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6S)-4-[(3-methylimidazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6S)-4-[(3-methylimidazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-[[(6S)-4-(2-methylpyrazole-3-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H20N6O3
5-[[(6S)-4-(2-methylpyrazole-3-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-ethyl-N-[6-methyl-2-[(3S)-1-pyrimidin-4-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H20N8S
5-ethyl-N-[6-methyl-2-[(3S)-1-pyrimidin-4-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-[[(6R)-4-(cyclopentanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C17H24N4O3
5-[[(6R)-4-(cyclopentanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-ethyl-N-[6-methyl-2-[(3R)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C18H26N6OS
5-ethyl-N-[6-methyl-2-[(3R)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-methyl-N-[2-methyl-6-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C15H21N5S
5-methyl-N-[2-methyl-6-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 5-methyl-N-[2-methyl-6-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C16H24N6S
5-methyl-N-[2-methyl-6-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-methyl-N-[2-methyl-6-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C16H24N6S
5-methyl-N-[2-methyl-6-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[6-methyl-2-[(3S)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H20N8S
5-ethyl-N-[6-methyl-2-[(3S)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-[[(6S)-4-[(2-methylpyrazol-3-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6S)-4-[(2-methylpyrazol-3-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-oxolane-2-carboxylate —— C12H12N2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-oxolane-2-carboxylate
—— [5-[[Benzyl-[(3,4-dimethoxyphenyl)methyl]amino]methyl]furan-2-yl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone —— C32H34FN3O4
[5-[[Benzyl-[(3,4-dimethoxyphenyl)methyl]amino]methyl]furan-2-yl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone
—— 5-ethyl-N-[6-methyl-2-[(3R)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H20N8S
5-ethyl-N-[6-methyl-2-[(3R)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H22N8S
5-ethyl-N-[2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-[[(6S)-4-[(1-methylpyrazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6S)-4-[(1-methylpyrazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 5-methyl-N-[2-methyl-6-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C15H21N5S
5-methyl-N-[2-methyl-6-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 5-ethyl-N-[6-methyl-2-[(3R)-1-pyrimidin-4-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H20N8S
5-ethyl-N-[6-methyl-2-[(3R)-1-pyrimidin-4-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[6-methyl-2-[(3S)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C18H26N6OS
5-ethyl-N-[6-methyl-2-[(3S)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-methyl-N-[6-methyl-2-[(3S)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,2-oxazol-3-amine —— C17H19N7O
5-methyl-N-[6-methyl-2-[(3S)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,2-oxazol-3-amine
—— 5-methyl-N-[6-methyl-2-[(3R)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,2-oxazol-3-amine —— C17H19N7O
5-methyl-N-[6-methyl-2-[(3R)-1-pyrimidin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,2-oxazol-3-amine
—— 5-methyl-N-[6-methyl-2-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,2-oxazol-3-amine —— C16H23N5O
5-methyl-N-[6-methyl-2-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,2-oxazol-3-amine
—— 5-ethyl-N-[6-methyl-2-[(3S)-1-pyrazin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H20N8S
5-ethyl-N-[6-methyl-2-[(3S)-1-pyrazin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[6-methyl-2-[(3R)-1-pyrazin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H20N8S
5-ethyl-N-[6-methyl-2-[(3R)-1-pyrazin-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[6-methyl-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C19H23N7S
5-ethyl-N-[6-methyl-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H22N8S
5-ethyl-N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-[6-[(3R)-1-methylpiperidin-3-yl]pyrazin-2-yl]pyridin-2-amine —— C15H19N5
5-[6-[(3R)-1-methylpiperidin-3-yl]pyrazin-2-yl]pyridin-2-amine
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2,4,6-trimethylbenzoate —— C19H17N3O5
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2,4,6-trimethylbenzoate
—— 5-ethyl-N-[6-methyl-2-[(3R)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C19H23N7S
5-ethyl-N-[6-methyl-2-[(3R)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine