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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19FN6O
5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-phenyl-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H18N6
5-phenyl-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C20H20FN3O
5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— (5S)-9-[2-(2-ethylphenoxy)ethyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H26N2O3
(5S)-9-[2-(2-ethylphenoxy)ethyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-9-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H24N4O2S
(5R)-3-methyl-9-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20N4O3
(5R)-9-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H25N3O3
(5R)-3-methyl-9-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-2-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H27N5O3
(5S)-2-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-3-ethyl-4-[[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-1-methylpyrazole —— C17H21ClFN3
5-chloro-3-ethyl-4-[[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-1-methylpyrazole
—— 5-phenyl-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H18N6
5-phenyl-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-9-[2-(2-ethylphenoxy)ethyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H26N2O3
(5R)-9-[2-(2-ethylphenoxy)ethyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-chloro-3-ethyl-4-[[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-1-methylpyrazole —— C17H21ClFN3
5-chloro-3-ethyl-4-[[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-1-methylpyrazole
—— (5R)-9-(2,4-difluoro-3-methoxybenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20F2N2O4
(5R)-9-(2,4-difluoro-3-methoxybenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pentyl-[(3R)-thiolan-3-yl]azanium —— C18H26N3O2S+
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pentyl-[(3R)-thiolan-3-yl]azanium
—— 5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide —— C19H23FN2O2
5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide
—— 5-methoxy-2-[[(3S)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]methyl]pyran-4-one —— C21H27NO3
5-methoxy-2-[[(3S)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]methyl]pyran-4-one
—— 5-propan-2-yl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]pyrimidine —— C22H31N5
5-propan-2-yl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]pyrimidine
—— (5-Methylthiophen-2-yl)methyl-(2-thiophen-2-ylethyl)azanium —— C12H16NS2+
(5-Methylthiophen-2-yl)methyl-(2-thiophen-2-ylethyl)azanium
—— 5-propyl-4-[(3S)-3-(1-pyrimidin-2-ylpiperidin-4-yl)pyrrolidin-1-yl]pyrimidine —— C20H28N6
5-propyl-4-[(3S)-3-(1-pyrimidin-2-ylpiperidin-4-yl)pyrrolidin-1-yl]pyrimidine
—— 5-methoxy-2-[[(3R)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]methyl]pyran-4-one —— C21H27NO3
5-methoxy-2-[[(3R)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]methyl]pyran-4-one
—— (5S)-9-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O3S
(5S)-9-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-2-(2H-benzotriazole-5-carbonyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H27N5O2
(5R)-2-(2H-benzotriazole-5-carbonyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O3S
(5R)-9-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-7-(2-methyl-5-propan-2-ylfuran-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H22N2O4
(5R)-3-methyl-7-(2-methyl-5-propan-2-ylfuran-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methyl-N-[(4-morpholin-4-ylsulfonylphenyl)methyl]-1,2-oxazole-3-carboxamide —— C16H19N3O5S
5-methyl-N-[(4-morpholin-4-ylsulfonylphenyl)methyl]-1,2-oxazole-3-carboxamide
—— 5-[[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine —— C21H27N5
5-[[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine
—— 5-propan-2-yl-4-[(3R)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]pyrimidine —— C22H31N5
5-propan-2-yl-4-[(3R)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]pyrimidine
—— 5-methyl-2-[(E)-2-[4-(3-methylbutoxy)phenyl]ethenyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C21H21N2O4S-
5-methyl-2-[(E)-2-[4-(3-methylbutoxy)phenyl]ethenyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— (5S)-2-(2H-benzotriazole-5-carbonyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H27N5O2
(5S)-2-(2H-benzotriazole-5-carbonyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide —— C19H23FN2O2
5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide
—— (5S)-3-methyl-7-(2-methyl-5-propan-2-ylfuran-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H22N2O4
(5S)-3-methyl-7-(2-methyl-5-propan-2-ylfuran-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H20N4O4
(5S)-7-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-propyl-4-[(3R)-3-(1-pyrimidin-2-ylpiperidin-4-yl)pyrrolidin-1-yl]pyrimidine —— C20H28N6
5-propyl-4-[(3R)-3-(1-pyrimidin-2-ylpiperidin-4-yl)pyrrolidin-1-yl]pyrimidine
—— (5S)-3-methyl-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5S)-3-methyl-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pentyl-[(3S)-thiolan-3-yl]azanium —— C18H26N3O2S+
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pentyl-[(3S)-thiolan-3-yl]azanium
—— (5R)-3-methyl-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5R)-3-methyl-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H24N4O3
(5R)-3-methyl-9-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[3-(benzenesulfonyl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H20N2O5S
(5S)-9-[3-(benzenesulfonyl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H20N4O2
(5R)-9-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H21N5O3
(5S)-3-methyl-9-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-N-(benzylsulfamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine —— C14H18N4O2S
(5R)-N-(benzylsulfamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O3
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[2-(2-fluorophenoxy)ethylsulfanyl]-N-(3-methoxyphenyl)-1,3,4-thiadiazol-2-amine —— C17H16FN3O2S2
5-[2-(2-fluorophenoxy)ethylsulfanyl]-N-(3-methoxyphenyl)-1,3,4-thiadiazol-2-amine
—— (5R)-5-[[(1R)-2,2-dichlorocyclopropyl]methyliminomethyl]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C12H15Cl2N3O3S
(5R)-5-[[(1R)-2,2-dichlorocyclopropyl]methyliminomethyl]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-ethyl-3-[[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C17H21N5O
5-ethyl-3-[[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-ethyl-3-[[(2R)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C17H21N5O
5-ethyl-3-[[(2R)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5-ethyl-1H-pyrazol-4-yl)-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone —— C16H26N4O2
(5-ethyl-1H-pyrazol-4-yl)-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone
—— (5R)-3-methyl-9-[(1-propylimidazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H26N4O2
(5R)-3-methyl-9-[(1-propylimidazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H21N3O3S
(5R)-3-methyl-9-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(1S)-2,2-dichlorocyclopropyl]methyliminomethyl]-1,3-diethyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C13H17Cl2N3O2S
5-[[(1S)-2,2-dichlorocyclopropyl]methyliminomethyl]-1,3-diethyl-2-sulfanylidene-1,3-diazinane-4,6-dione