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—— 5-ethyl-N-[(2R)-2-methyl-3-[3-(5-methyl-1H-pyrazol-4-yl)propylamino]-3-oxopropyl]furan-2-carboxamide —— C18H26N4O3
5-ethyl-N-[(2R)-2-methyl-3-[3-(5-methyl-1H-pyrazol-4-yl)propylamino]-3-oxopropyl]furan-2-carboxamide
—— [5-[[(1S)-1-(2-methoxyphenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-yl]-pyrrolidin-1-ylmethanone —— C24H27N3O3
[5-[[(1S)-1-(2-methoxyphenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-yl]-pyrrolidin-1-ylmethanone
—— [5-[[(1S)-1-(2-methoxyphenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-yl]-morpholin-4-ylmethanone —— C24H28N3O4+
[5-[[(1S)-1-(2-methoxyphenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-yl]-morpholin-4-ylmethanone
—— 5-chloro-6-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C14H14ClN5O
5-chloro-6-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 5-chloro-6-[(2R)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C14H14ClN5O
5-chloro-6-[(2R)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— [5-[[Cyclopropyl(ethylcarbamoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C15H22N2O5S
[5-[[Cyclopropyl(ethylcarbamoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— [5-[[Furan-2-carbonyl(2-methylpropyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C18H23NO6S
[5-[[Furan-2-carbonyl(2-methylpropyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— 5-methyl-2-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-1,3-benzoxazole —— C16H18N4O2
5-methyl-2-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-1,3-benzoxazole
—— [5-[[furan-2-carbonyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate —— C19H23NO7S
[5-[[furan-2-carbonyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate
—— [5-[[(1R)-1-(2-methoxyphenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-yl]-morpholin-4-ylmethanone —— C24H28N3O4+
[5-[[(1R)-1-(2-methoxyphenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-yl]-morpholin-4-ylmethanone
—— 5-[[(1S)-1-(2,4-difluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid —— C19H16F2N2O3
5-[[(1S)-1-(2,4-difluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid
—— 5-[[(1S)-1-(2,4-difluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate —— C19H16F2N2O3
5-[[(1S)-1-(2,4-difluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate
—— [5-[[(1R)-1-(2-methoxyphenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-yl]-pyrrolidin-1-ylmethanone —— C24H27N3O3
[5-[[(1R)-1-(2-methoxyphenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-yl]-pyrrolidin-1-ylmethanone
—— [5-[[ethylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate —— C17H26N2O6S
[5-[[ethylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate
—— [5-[[Cyclopropyl-(2-methoxyacetyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C15H21NO6S
[5-[[Cyclopropyl-(2-methoxyacetyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— [5-[[ethylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate —— C17H26N2O6S
[5-[[ethylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate
—— 5-[[(1R)-1-(2,4-difluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid —— C19H16F2N2O3
5-[[(1R)-1-(2,4-difluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid
—— 5-[[(1R)-1-(2,4-difluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate —— C19H16F2N2O3
5-[[(1R)-1-(2,4-difluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate
—— 5-{[(Tert-butylcarbamoyl)(2-methoxyethyl)amino]methyl}-2-methoxyphenyl propane-2-sulfonate —— C19H32N2O6S
5-{[(Tert-butylcarbamoyl)(2-methoxyethyl)amino]methyl}-2-methoxyphenyl propane-2-sulfonate
—— [5-[[(1R)-1-(2-methoxyphenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-yl]-pyrrolidin-1-ylmethanone —— C24H28N3O3+
[5-[[(1R)-1-(2-methoxyphenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-yl]-pyrrolidin-1-ylmethanone
—— 5-chloro-6-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C16H18ClN5O
5-chloro-6-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 5-[(2S)-oxolan-2-yl]-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-oxazole-4-carboxamide —— C15H18N4O3
5-[(2S)-oxolan-2-yl]-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-oxazole-4-carboxamide
—— 5-[(2R)-oxolan-2-yl]-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-oxazole-4-carboxamide —— C15H18N4O3
5-[(2R)-oxolan-2-yl]-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-oxazole-4-carboxamide
—— 5-[(2S)-oxolan-2-yl]-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-oxazole-4-carboxamide —— C15H18N4O3
5-[(2S)-oxolan-2-yl]-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-oxazole-4-carboxamide
—— [5-[[cyclobutanecarbonyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate —— C19H27NO6S
[5-[[cyclobutanecarbonyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate
—— 5-{[1-Cyclopropyl(ethylcarbamoyl)amino]methyl}-2-methoxyphenyl ethane-1-sulfonate —— C16H24N2O5S
5-{[1-Cyclopropyl(ethylcarbamoyl)amino]methyl}-2-methoxyphenyl ethane-1-sulfonate
—— 5-Chloro-2-(5-methyl-1,3-benzoxazol-2-yl)phenyl methanesulfonate —— C15H12ClNO4S
5-Chloro-2-(5-methyl-1,3-benzoxazol-2-yl)phenyl methanesulfonate
—— 5-methyl-2-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-1,3-benzoxazole —— C16H18N4O2
5-methyl-2-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-1,3-benzoxazole
—— 5-{[(Tert-butylcarbamoyl)[(furan-2-YL)methyl]amino]methyl}-2-methoxyphenyl methanesulfonate —— C19H26N2O6S
5-{[(Tert-butylcarbamoyl)[(furan-2-YL)methyl]amino]methyl}-2-methoxyphenyl methanesulfonate
—— 5-methyl-N-[(2R)-2-methyl-3-[3-(5-methyl-1H-pyrazol-4-yl)propylamino]-3-oxopropyl]thiophene-2-carboxamide —— C17H24N4O2S
5-methyl-N-[(2R)-2-methyl-3-[3-(5-methyl-1H-pyrazol-4-yl)propylamino]-3-oxopropyl]thiophene-2-carboxamide
—— 5-chloro-6-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C14H14ClN5O
5-chloro-6-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 5-methyl-2-[(2R)-2-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-1,3-benzoxazole —— C17H20N4O2
5-methyl-2-[(2R)-2-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-1,3-benzoxazole
—— 5-(4-fluorophenyl)-N-[(1R)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-oxopentanamide —— C20H20FNO3
5-(4-fluorophenyl)-N-[(1R)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-oxopentanamide
—— (5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2S)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C17H19N5OS
(5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2S)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— 5-[(2-Fluorophenyl)methyl]-4-(methoxymethyl)-2-methyl-6-(4-methylsulfonylpiperazin-1-yl)pyrimidine —— C19H25FN4O3S
5-[(2-Fluorophenyl)methyl]-4-(methoxymethyl)-2-methyl-6-(4-methylsulfonylpiperazin-1-yl)pyrimidine
—— 5-({1-Cyclopropyl[(propan-2-YL)carbamoyl]amino}methyl)-2-methoxyphenyl ethane-1-sulfonate —— C17H26N2O5S
5-({1-Cyclopropyl[(propan-2-YL)carbamoyl]amino}methyl)-2-methoxyphenyl ethane-1-sulfonate
—— 5-[(2-Fluorophenyl)methyl]-4-(4-methanesulfonylpiperazin-1-YL)-2,6-dimethylpyrimidine —— C18H23FN4O2S
5-[(2-Fluorophenyl)methyl]-4-(4-methanesulfonylpiperazin-1-YL)-2,6-dimethylpyrimidine
—— [5-Chloro-2-(5-methyl-1,3-benzoxazol-2-yl)phenyl] 4-methylbenzenesulfonate —— C21H16ClNO4S
[5-Chloro-2-(5-methyl-1,3-benzoxazol-2-yl)phenyl] 4-methylbenzenesulfonate
—— 5-(4-fluorophenyl)-N-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-oxopentanamide —— C20H20FNO3
5-(4-fluorophenyl)-N-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-oxopentanamide
—— 5-{[1-(Furan-2-YL)-N-(propan-2-YL)formamido]methyl}-2-methoxyphenyl propane-2-sulfonate —— C19H25NO6S
5-{[1-(Furan-2-YL)-N-(propan-2-YL)formamido]methyl}-2-methoxyphenyl propane-2-sulfonate
—— 5-[(2-Chloro-6-fluorophenyl)methyl]-2,4-dimethyl-6-(4-methylsulfonylpiperazin-1-yl)pyrimidine —— C18H22ClFN4O2S
5-[(2-Chloro-6-fluorophenyl)methyl]-2,4-dimethyl-6-(4-methylsulfonylpiperazin-1-yl)pyrimidine
—— 5-{[1-Cyclopropyl(tert-butylcarbamoyl)amino]methyl}-2-methoxyphenyl methanesulfonate —— C17H26N2O5S
5-{[1-Cyclopropyl(tert-butylcarbamoyl)amino]methyl}-2-methoxyphenyl methanesulfonate
—— (5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C17H19N5OS
(5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— [5-[[4-[Cyclohexyl(methyl)amino]-6-methylpyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-pyrrolidin-1-ylmethanone —— C22H30N4O2S
[5-[[4-[Cyclohexyl(methyl)amino]-6-methylpyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-pyrrolidin-1-ylmethanone
—— 5-[[(1S)-1-(2-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid —— C19H17FN2O3
5-[[(1S)-1-(2-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid
—— 5-[[(1S)-1-(2-fluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate —— C19H17FN2O3
5-[[(1S)-1-(2-fluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate
—— 5-[(2,5-Dimethylphenyl)methyl]-2,4-dimethyl-6-(4-propylsulfonylpiperazin-1-yl)pyrimidine —— C22H32N4O2S
5-[(2,5-Dimethylphenyl)methyl]-2,4-dimethyl-6-(4-propylsulfonylpiperazin-1-yl)pyrimidine
—— 5-bromo-1-[(2R)-oxan-2-yl]indazole —— C12H13BrN2O
5-bromo-1-[(2R)-oxan-2-yl]indazole
—— 5-bromo-1-[(2S)-oxan-2-yl]indazole —— C12H13BrN2O
5-bromo-1-[(2S)-oxan-2-yl]indazole
—— 5-chloro-2-methoxy-N-[(2R)-4-morpholin-4-ylbutan-2-yl]benzamide —— C16H23ClN2O3
5-chloro-2-methoxy-N-[(2R)-4-morpholin-4-ylbutan-2-yl]benzamide