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—— (5-fluoro-2-methoxyphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C18H15FN2O3
(5-fluoro-2-methoxyphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— 5-[(2R)-1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]-4-(2-fluorophenyl)-1H-pyrazole —— C19H17ClFN3O2S
5-[(2R)-1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]-4-(2-fluorophenyl)-1H-pyrazole
—— 5-[(2S)-1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]-4-(2-fluorophenyl)-1H-pyrazole —— C19H17ClFN3O2S
5-[(2S)-1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]-4-(2-fluorophenyl)-1H-pyrazole
—— (5-Methyl-1,3,4-oxadiazol-2-yl)methyl 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C17H18N4O3
(5-Methyl-1,3,4-oxadiazol-2-yl)methyl 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— 5-[(2S)-pyrrolidin-2-yl]-4-[3-(trifluoromethyl)phenyl]-1H-pyrazole —— C14H14F3N3
5-[(2S)-pyrrolidin-2-yl]-4-[3-(trifluoromethyl)phenyl]-1H-pyrazole
—— (5-fluoro-3-methyl-1H-indol-2-yl)-[(3S)-3-[2-[(3-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone —— C25H25FN6O
(5-fluoro-3-methyl-1H-indol-2-yl)-[(3S)-3-[2-[(3-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone
—— (5-fluoro-3-methyl-1H-indol-2-yl)-[(3S)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C23H22FN7O
(5-fluoro-3-methyl-1H-indol-2-yl)-[(3S)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— (5-fluoro-3-methyl-1H-indol-2-yl)-[(3S)-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone —— C25H25FN6O
(5-fluoro-3-methyl-1H-indol-2-yl)-[(3S)-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone
—— (5-fluoro-3-methyl-1H-indol-2-yl)-[(3R)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C23H22FN7O
(5-fluoro-3-methyl-1H-indol-2-yl)-[(3R)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— (5-fluoro-3-methyl-1H-indol-2-yl)-[(3R)-3-[2-[(3-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone —— C25H25FN6O
(5-fluoro-3-methyl-1H-indol-2-yl)-[(3R)-3-[2-[(3-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone
—— 5-[(2R)-pyrrolidin-2-yl]-4-[3-(trifluoromethyl)phenyl]-1H-pyrazole —— C14H14F3N3
5-[(2R)-pyrrolidin-2-yl]-4-[3-(trifluoromethyl)phenyl]-1H-pyrazole
—— (5-fluoro-3-methyl-1H-indol-2-yl)-[(3R)-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone —— C25H25FN6O
(5-fluoro-3-methyl-1H-indol-2-yl)-[(3R)-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]methanone
—— (5-methoxycarbonylfuran-2-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C17H14N2O5
(5-methoxycarbonylfuran-2-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— (5-acetyl-2-ethoxyphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C21H20N2O4
(5-acetyl-2-ethoxyphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— 5,6-dimethyl-2-[[5-(2-methylpropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C15H19N5OS3
5,6-dimethyl-2-[[5-(2-methylpropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5-methyl-1H-pyrazol-4-yl)-[(3S)-3-[6-(2-propan-2-ylimidazol-1-yl)pyridin-2-yl]piperidin-1-yl]methanone —— C21H26N6O
(5-methyl-1H-pyrazol-4-yl)-[(3S)-3-[6-(2-propan-2-ylimidazol-1-yl)pyridin-2-yl]piperidin-1-yl]methanone
—— (5-methyl-1H-pyrazol-4-yl)-[(3R)-3-[6-(2-propan-2-ylimidazol-1-yl)pyridin-2-yl]piperidin-1-yl]methanone —— C21H26N6O
(5-methyl-1H-pyrazol-4-yl)-[(3R)-3-[6-(2-propan-2-ylimidazol-1-yl)pyridin-2-yl]piperidin-1-yl]methanone
—— (5-methyl-1H-pyrazol-4-yl)-[4-[6-(2-propan-2-ylimidazol-1-yl)pyridin-2-yl]piperidin-1-yl]methanone —— C21H26N6O
(5-methyl-1H-pyrazol-4-yl)-[4-[6-(2-propan-2-ylimidazol-1-yl)pyridin-2-yl]piperidin-1-yl]methanone
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(methanesulfonamido)benzoate —— C17H15N3O5S
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(methanesulfonamido)benzoate
—— 5-[[(2S)-2-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole —— C24H25FN4O
5-[[(2S)-2-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole
—— 5-[[(2S)-2-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole —— C24H25FN4O
5-[[(2S)-2-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole
—— 5-[(2R)-2-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one —— C22H23FN4O3
5-[(2R)-2-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-[[(2R)-2-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole —— C24H25FN4O
5-[[(2R)-2-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole
—— 5-[(2S)-2-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one —— C22H23FN4O3
5-[(2S)-2-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-[[(2R)-2-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole —— C24H24F2N4O
5-[[(2R)-2-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole
—— 5-[[(2S)-2-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole —— C24H24F2N4O
5-[[(2S)-2-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole
—— 5-[[(2R)-2-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole —— C24H25FN4O
5-[[(2R)-2-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole
—— 5-[[(3S)-3-[5-[2-(2-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole —— C24H25ClN4O
5-[[(3S)-3-[5-[2-(2-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]-1H-indole
—— 5-(4-Oxocinnolin-1-yl)pentanenitrile —— C13H13N3O
5-(4-Oxocinnolin-1-yl)pentanenitrile
—— 5-[3,5-Dimethyl-4-(4-methylpiperidin-1-yl)sulfonylpyrazol-1-yl]pentanenitrile —— C16H26N4O2S
5-[3,5-Dimethyl-4-(4-methylpiperidin-1-yl)sulfonylpyrazol-1-yl]pentanenitrile
—— 5-(3,5-Dimethyl-4-morpholin-4-ylsulfonylpyrazol-1-yl)pentanenitrile —— C14H22N4O3S
5-(3,5-Dimethyl-4-morpholin-4-ylsulfonylpyrazol-1-yl)pentanenitrile
—— 5-[[3,5-Dimethyl-4-(4-methylpiperidin-1-yl)sulfonylpyrazol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C20H25N5O3S
5-[[3,5-Dimethyl-4-(4-methylpiperidin-1-yl)sulfonylpyrazol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 5-(2-Methyl-4-oxo-3-phenoxychromen-7-yl)oxypentanenitrile —— C21H19NO4
5-(2-Methyl-4-oxo-3-phenoxychromen-7-yl)oxypentanenitrile
—— 5-[[3,5-Dimethyl-4-(4-methylpiperidin-1-yl)sulfonylpyrazol-1-yl]methyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C18H23N5O3S2
5-[[3,5-Dimethyl-4-(4-methylpiperidin-1-yl)sulfonylpyrazol-1-yl]methyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-methyl-N-[4-[(2R)-1-methylpiperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C14H19N5S
5-methyl-N-[4-[(2R)-1-methylpiperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— 5-(4-Acetylphenyl)-1-(5-chlorothiophen-2-yl)-3-(hydroxymethyl)-4,6-dioxo-1,2,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-3-carboxylic acid —— C20H17ClN2O6S
5-(4-Acetylphenyl)-1-(5-chlorothiophen-2-yl)-3-(hydroxymethyl)-4,6-dioxo-1,2,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-3-carboxylic acid
—— 5-[(4-Tert-butylphenyl)methyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C22H21FN4O
5-[(4-Tert-butylphenyl)methyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[2-(2-Fluorophenoxy)ethyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C19H14F2N4O2
5-[2-(2-Fluorophenoxy)ethyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-(5-Methylthiophen-2-yl)-3-[(4-nitrophenyl)methyl]thieno[2,3-d]pyrimidin-4-one —— C18H13N3O3S2
5-(5-Methylthiophen-2-yl)-3-[(4-nitrophenyl)methyl]thieno[2,3-d]pyrimidin-4-one
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 3-chloro-4-ethoxy-5-methoxybenzoate —— C20H18ClNO5
(5-Phenyl-1,2-oxazol-3-yl)methyl 3-chloro-4-ethoxy-5-methoxybenzoate
—— 5-(2-fluorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C19H21FN6O2S
5-(2-fluorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 5-(4-fluorophenyl)-4-[(2S)-1-(1H-indol-5-ylmethyl)piperidin-2-yl]pyrimidin-2-amine —— C24H24FN5
5-(4-fluorophenyl)-4-[(2S)-1-(1H-indol-5-ylmethyl)piperidin-2-yl]pyrimidin-2-amine
—— 5-(1,3-Benzothiazol-2-ylmethyl)-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C19H12FN5OS
5-(1,3-Benzothiazol-2-ylmethyl)-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(3,5-Dimethyl-4-piperidin-1-ylsulfonylpyrazol-1-yl)methyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C17H21N5O3S2
5-[(3,5-Dimethyl-4-piperidin-1-ylsulfonylpyrazol-1-yl)methyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-[(2,6-Dichlorophenyl)methyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C18H11Cl2FN4O
5-[(2,6-Dichlorophenyl)methyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-(4-chlorophenyl)-4-[(2R)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-2-yl]pyrimidin-2-amine —— C22H25ClN6
5-(4-chlorophenyl)-4-[(2R)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-2-yl]pyrimidin-2-amine
—— 5-[2-(4-Fluorophenoxy)ethyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C19H14F2N4O2
5-[2-(4-Fluorophenoxy)ethyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-(4-fluorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C19H21FN6O2S
5-(4-fluorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 5-(3-fluorophenyl)-4-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]pyrimidin-2-amine —— C18H17FN6
5-(3-fluorophenyl)-4-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]pyrimidin-2-amine
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 3-chloro-4-ethoxy-5-methoxybenzoate —— C18H16ClNO6
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 3-chloro-4-ethoxy-5-methoxybenzoate