抑制剂简介
抑制剂是一类能够降低或阻止生物体内的酶活性、受体的活性或是细胞内特定反应过程的小分子化合物。它们在有机化学、化学化工和生物医药领域中有着广泛的应用,尤其是在药物研发方面。
分类与作用机制
应用领域
总结
抑制剂的研究和发展对于理解生命过程至关重要,并在药物开发、基础科学研究等多个领域发挥着重要作用。随着技术的进步,新的抑制剂不断被发现和开发出来,为医学治疗提供了更多的可能性。
中文名称 | 英文名称 | CAS号 | 化学式 | 结构式图片 |
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泊马度胺 | pomalidomide | 19171-19-8 | C13H11N3O4 |
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沙芬酰胺甲磺酸盐 | safinamide mesylate | 202825-46-5 | CH4O3S*C17H19FN2O2 |
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沙芬酰胺 | safinamide | 133865-89-1 | C17H19FN2O2 |
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沙库巴曲 | sacubitril | 149709-62-6 | C24H29NO5 |
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氯贝胆碱 | bethanechol chloride | 590-63-6 | C7H17N2O2*Cl |
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氨萘非特 | amonafide | 69408-81-7 | C16H17N3O2 |
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氨芬酸钠 | 61618-27-7 | C15H15NNaO4 |
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氢溴酸达非那新 | (S)-darifenacin hydrobromide | 133099-07-7 | BrH*C28H30N2O2 |
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氢溴酸替格列汀 | Teneligliptin hydrobromide anhydrous | 906093-29-6 | C44H65Br5N12O2S2 |
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氢化白果酸 | 6-Pentadecylsalicylic Acid | 16611-84-0 | C22H36O3 |
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氟米龙醋酸酯 | fluorometholone acetate | 3801-06-7 | C24H31FO5 |
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氟米松 | flumetasone | 2135-17-3 | C22H28F2O5 |
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比瑞那帕 | birinapant | 1260251-31-7 | C42H56F2N8O6 |
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比尼替尼 | binimetinib | 606143-89-9 | C17H15BrF2N4O3 |
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比卡格韦 | bictegravir sodium | 1807988-02-8 | C21H17F3N3O5*Na |
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毒黄素 | toxoflavin | 84-82-2 | C7H7N5O2 |
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欧司哌米 | ospemifene | 128607-22-7 | C24H23ClO2 |
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桑霉素 | sangivamycin | 18417-89-5 | C12H15N5O5 |
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格拉斯吉布 | glasdegib | 1095173-27-5 | C21H22N6O |
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枸橼酸艾沙佐米 | ixazomib citrate | 1239908-20-3 | C20H23BCl2N2O9 |
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枸橼酸托瑞米芬 | toremifene citrate | 89778-27-8 | C6H8O7*C26H28ClNO |
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林扎戈利 | 3-[2-fluoro-5-(2,3-difluoro-6-methoxybenzyloxy)-4-methoxyphenyl]-2,4-dioxo-1,2,3,4-tetrahydrothieno[3,4-d]pyrimidine-5-carboxylic acid | 935283-04-8 | C22H15F3N2O7S |
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月桂41-2272 | 5-cyclopropyl-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyrimidin-4-ylamine | 256376-24-6 | C20H17FN6 |
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替泊沙林 | tepoxalin | 103475-41-8 | C20H20ClN3O3 |
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替拉鲁替尼 | 6-amino-9-[(3R)-1-(2-butynoyl)-3-pyrrolidinyl]-7-(4-phenoxyphenyl)-7,9-dihydro-8H-purin-8-one | 1351636-18-4 | C25H22N6O3 |
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替拉替尼 | 17-allylamino-17-demethoxygeldanamycin | 75747-14-7 | C31H43N3O8 |
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替吡法尼 | tipifarnib | 192185-72-1 | C27H22Cl2N4O |
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曲西瑞宾 | triciribine | 35943-35-2 | C13H16N6O4 |
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曲美替尼 | trametinib | 871700-17-3 | C26H23FIN5O4 |
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曲法罗汀 | trifarotene | 895542-09-3 | C29H33NO4 |
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曲格列汀 | Trelagliptin | 865759-25-7 | C18H20FN5O2 |
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曲帕拉醇 | triparanol | 78-41-1 | C27H32ClNO2 |
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普纳替尼 | ponatinib | 943319-70-8 | C29H27F3N6O |
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普卡必利 | prucalopride | 179474-81-8 | C18H26ClN3O3 |
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普乐沙福 | 1-[4-(1,4,8,11-tetraazacyclotetradecan-1-ylmethyl)benzyl]-1,4,8,11-tetraazacyclotetradecane | 110078-46-1 | C28H54N8 |
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昂丹司琼 | ondanserton | 99614-02-5 | C18H19N3O |
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拮抗剂多肽BALIXAFORTIDE | Balixafortide | 1051366-32-5 | C84H118N24O21S2 |
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粉蝶霉素A | piericidin A | 2738-64-9 | C25H37NO4 |
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托莫西汀 | (R)-Tomoxetine | 83015-26-3 | C17H21NO |
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托法替尼 | tasocitinib | 477600-75-2 | C16H20N6O |
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托彻普 | ethyl cis-4-((3,5-bis(trifluoromethyl)benzyl)(methoxycarbonyl)amino)-2-ethyl-6-(trifluoromethyl)-3,4-dihydroquinoline-1(2H)-carboxylate | 262352-17-0 | C26H25F9N2O4 |
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托卡朋 | tolcapone | 134308-13-7 | C14H11NO5 |
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托伐普坦 | tolvaptan | 150683-30-0 | C26H25ClN2O3 |
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扎托布洛芬 | zaltoprofen | 74711-43-6 | C17H14O3S |
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恩替诺特 | Entinostat | 209783-80-2 | C21H20N4O3 |
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异环磷酰胺 | ilfosfamide | 3778-73-2 | C7H15Cl2N2O2P |
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异烟棒曲霉素C | roquefortine C | 58735-64-1 | C22H23N5O2 |
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异戊酰胺 | isobutylamide | 541-46-8 | C5H11NO |
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康奈非尼 | encorafenib | 1269440-17-6 | C22H27ClFN7O4S |
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度鲁特韦钠盐 | (4R,12AS)-N-(2,4-difluorobenzyl)-7-hydroxy-4-methyl-6,8-dioxo-3,4,6,8,12,12a-hexahydro-2H-pyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxamide, sodium sa | 1051375-19-9 | C20H19F2N3NaO5 |
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