抑制剂简介
抑制剂是一类能够降低或阻止生物体内的酶活性、受体的活性或是细胞内特定反应过程的小分子化合物。它们在有机化学、化学化工和生物医药领域中有着广泛的应用,尤其是在药物研发方面。
分类与作用机制
应用领域
总结
抑制剂的研究和发展对于理解生命过程至关重要,并在药物开发、基础科学研究等多个领域发挥着重要作用。随着技术的进步,新的抑制剂不断被发现和开发出来,为医学治疗提供了更多的可能性。
中文名称 | 英文名称 | CAS号 | 化学式 | 结构式图片 |
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罗美昔布 | lumiracoxib | 220991-20-8 | C15H13ClFNO2 |
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罗米鲁曲 | 6-((4-bromothiophen-2-yl)methoxy)-9H-purin-2-amine | 192441-08-0 | C10H8BrN5OS |
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罗米地辛 | (1S,7Z,10S,16E,21R)-7-ethylidene-4,21-di(propan-2-yl)-2-oxa-12,13-dithia-5,8,20,23-tetrazabicyclo[8.7.6]tricos-16-ene-3,6,9,19,22-pentone | 128517-07-7 | C24H36N4O6S2 |
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罗替戈汀 | 5-hydroxy-2-(N-n-propyl-N-2-[2-thienyl]ethylamino)tetralin | 92206-54-7 | C19H25NOS |
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罗替戈汀 | rotigotine | 99755-59-6 | C19H25NOS |
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罗斯匹莫 | Losmapimod | 585543-15-3 | C22H26FN3O2 |
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维特克拉 | venetoclax | 1257044-40-8 | C45H50ClN7O7S |
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维利帕尼盐酸盐 | Veliparib dihydrochloride | 912445-05-7 | C13H18Cl2N4O |
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组织蛋白酶抑制剂1 | Cathepsin inhibitor 1 | 225120-65-0 | C20H24ClN5O2 |
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红斑素 | rubropunctatin | 514-67-0 | C21H22O5 |
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米氮平 | Mirtazapine | 85650-52-8 | C17H19N3 |
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米拉贝隆 | (R)-2-(2-aminothiazol-4-yl)-4'-[2-[(2-hydroxy-2-phenylethyl)amino]ethyl]acetanilide | 223673-61-8 | C21H24N4O2S |
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米屈肼(二水合物) | Meldonium dihydrate | 86426-17-7 | C6H18N2O4 |
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福美司坦 | Formestaqne | 848-35-1 | C19H28O3 |
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福美司坦 | 4-hydroxyandrost-4-ene-3,17-dione | 566-48-3 | C19H26O3 |
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福他替尼 | fostamatinib | 901119-35-5 | C23H26FN6O9P |
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磷酸组胺 | histamine diphosphate | 51-74-1 | C5H9N3*2H3O4P |
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硫锌酸硫胺 | sulbutiamine | 3286-46-2 | C32H46N8O6S2 |
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硫酸氯吡格雷 | (S)-(+)-clopidogrel bisulfate | 120202-66-6 | C16H16ClNO2S*H2O4S |
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硫酸单[(1R,2S,5R)-7-氧代-2-[(4-哌啶基氨基)羰基]-1,6-二氮杂双环[3.2.1]辛-6-基]酯 | relebactam | 1174018-99-5 | C12H20N4O6S |
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硫唑嘌呤 | Azathioprin | 446-86-6 | C9H7N7O2S |
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硝替卡朋 | nitecapone | 116313-94-1 | C12H11NO6 |
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石斛酚 | gigantol | 67884-30-4 | C16H18O4 |
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盐酸齐拉西酮 | ziprasidone hydrochloride | 122883-93-6 | C21H21ClN4OS*ClH |
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盐酸雷洛昔芬 | raloxifene hydrochloride | 82640-04-8 | C28H27NO4S*ClH |
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盐酸阿那格雷 | anagrelide hydrochloride | 58579-51-4 | C10H7Cl2N3O*ClH |
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盐酸阿莫伦特 | almorexant hydrochloride | 913358-93-7 | C29H31F3N2O3*ClH |
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盐酸阿米洛利二水合物 | 3,5-diamino-6-chloro-N-(diaminomethylidene)pyrazine-2-carboxamide;dihydrate;hydrochloride | 17440-83-4 | C6H13Cl2N7O3 |
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盐酸那拉曲坦 | naratriptan hydrochloride | 143388-64-1 | C17H25N3O2S*ClH |
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盐酸莫昔普利 | moexipril hydrochloride | 82586-52-5 | C27H34N2O7*ClH |
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盐酸芬司必利 | Fenspiride hydrochloride | 5053-08-7 | C15H20N2O2*ClH |
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盐酸美金刚 | memantine hydrochloride | 41100-52-1 | C12H21N*ClH |
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盐酸美托咪啶 | medetomidine hydrochloride | 86347-15-1 | C13H16N2*ClH |
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盐酸罗沙替丁醋酸酯 | Gastralgin | 93793-83-0 | C19H28N2O4*ClH |
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盐酸罗格列酮 | (+)-5-(4-[2-(N-methyl-N-(pyridin-2-yl)amino)ethoxy]-benzyl)thiazolidine-2,4-dione hydrochloride | 302543-62-0 | C18H19N3O3S*ClH |
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盐酸维拉唑酮 | vilazodone hydrochloride | 163521-08-2 | C26H27N5O2*ClH |
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盐酸甲状旁腺激素 | cinacalcet hydrochloride | 364782-34-3 | C22H22F3N*ClH |
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盐酸甲基苄肼 | matulane | 366-70-1 | C12H19N3O*ClH |
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盐酸枢复宁 | Ondansetron hydrochloride | 99614-01-4 | C18H19N3O*ClH |
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盐酸替莫普利 | temocapril Hydrochloride | 110221-44-8 | C23H28N2O5S2*ClH |
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盐酸文拉法辛 | venlafaxine hydrochloride | 99300-78-4 | C17H27NO2*ClH |
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盐酸托莫西汀 | atomoxetine hydrochloride | 82248-59-7 | C17H21NO*ClH |
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盐酸度洛西汀 | duloxetine hydrochloride | 136434-34-9 | C18H19NOS*ClH |
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盐酸帕洛诺司琼 | palonosetron hydrochloride | 135729-62-3 | C19H24N2O*ClH |
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盐酸帕唑帕尼 | pazopanib hydrochloride | 635702-64-6 | C21H23N7O2S*ClH |
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盐酸布比卡因 | bupivacaine hydrochloride | 18010-40-7 | C18H28N2O*ClH |
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盐酸巴多昔芬 | 1-[4-(2-azepan-1-yl-ethoxy)-benzyl]-2-(4-hydroxy-phenyl)-3-methyl-1H-indol-5-ol hydrochloride | 198480-56-7 | C30H34N2O3*ClH |
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盐酸奥洛他定 | olopatadine hydrochloride | 140462-76-6 | C21H23NO3*ClH |
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盐酸奥扎格雷 | ozagrel hydrochloride | 78712-43-3 | C13H12N2O2*ClH |
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盐酸多奈哌齐 | donepezil hydrochloride | 120011-70-3 | C24H29NO3*ClH |
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