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中文名称 英文名称 CAS号 化学式 结构式图片
—— diethyl-[(1R)-2-[[2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylacetyl]amino]-1-(furan-2-yl)ethyl]azanium —— C19H24FN6O2S+
diethyl-[(1R)-2-[[2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylacetyl]amino]-1-(furan-2-yl)ethyl]azanium
—— 1-phenyl-3-thiophen-2-yl-1H-pyrazole-4-carboxylic acid (furan-2-ylmethyl)-amide —— C19H15N3O2S
1-phenyl-3-thiophen-2-yl-1H-pyrazole-4-carboxylic acid (furan-2-ylmethyl)-amide
—— 5-amino-4-(3,4-dihydro-2H-pyrrol-5-yl)-1-methyl-2-phenyl-1,2-dihydro-3H-pyrazol-3-one 923681-80-5 C14H16N4O
5-amino-4-(3,4-dihydro-2H-pyrrol-5-yl)-1-methyl-2-phenyl-1,2-dihydro-3H-pyrazol-3-one
—— 1-benzyl-N-[(1R)-1-cyclopropylethyl]-3-(3,4-dimethoxyphenyl)pyrazole-4-carboxamide —— C24H27N3O3
1-benzyl-N-[(1R)-1-cyclopropylethyl]-3-(3,4-dimethoxyphenyl)pyrazole-4-carboxamide
—— N-[(3R)-1-benzylpyrrolidin-3-yl]-4-pyrazol-1-ylbenzamide —— C21H22N4O
N-[(3R)-1-benzylpyrrolidin-3-yl]-4-pyrazol-1-ylbenzamide
—— (2Z,4S)-2-(3H-1,3-benzothiazol-2-ylidene)-4-[1-(2-ethoxyphenyl)tetrazol-5-yl]sulfanyl-3-oxopentanenitrile —— C21H18N6O2S2
(2Z,4S)-2-(3H-1,3-benzothiazol-2-ylidene)-4-[1-(2-ethoxyphenyl)tetrazol-5-yl]sulfanyl-3-oxopentanenitrile
—— (3R)-1-[3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanoyl]piperidine-3-carboxamide —— C20H26N4O2
(3R)-1-[3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanoyl]piperidine-3-carboxamide
—— ATX inhibitor 3 —— C17H12ClFN2O5S
ATX inhibitor 3
—— (2S)-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[[(2R)-oxolan-2-yl]methyl]propanamide —— C20H26N4O3S
(2S)-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[[(2R)-oxolan-2-yl]methyl]propanamide
—— [1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone —— C27H25N3O2
[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— 1-(2-Ethoxyphenyl)-5-[(2-methoxy-5-methylphenyl)methylsulfanyl]tetrazole —— C18H20N4O2S
1-(2-Ethoxyphenyl)-5-[(2-methoxy-5-methylphenyl)methylsulfanyl]tetrazole
—— N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C18H21BrN2O2S
N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— (2S)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2S)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— N-[[2-(morpholin-4-ium-4-ylmethyl)phenyl]methyl]-2-thiophen-2-yl-1,3-thiazole-4-carboxamide —— C20H22N3O2S2+
N-[[2-(morpholin-4-ium-4-ylmethyl)phenyl]methyl]-2-thiophen-2-yl-1,3-thiazole-4-carboxamide
—— 3-benzyl-5-[[(4R)-1,3-dioxan-4-yl]methylsulfanyl]-4-(4-fluorophenyl)-1,2,4-triazole —— C20H20FN3O2S
3-benzyl-5-[[(4R)-1,3-dioxan-4-yl]methylsulfanyl]-4-(4-fluorophenyl)-1,2,4-triazole
—— 1-[(2S)-2-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(1-phenylpyrazol-4-yl)propan-1-one —— C24H24N4OS
1-[(2S)-2-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(1-phenylpyrazol-4-yl)propan-1-one
—— (2R)-N,N,3-trimethyl-7-phenyl-2H-imidazo[2,1-b][1,3,4]thiadiazine-2-carboxamide —— C15H16N4OS
(2R)-N,N,3-trimethyl-7-phenyl-2H-imidazo[2,1-b][1,3,4]thiadiazine-2-carboxamide
—— N-(furan-2-ylmethyl)-N-methyl-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylacetamide —— C19H17N5O2S
N-(furan-2-ylmethyl)-N-methyl-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylacetamide
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2S)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2S)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— N-(3-tert-butyl-1,2-oxazol-5-yl)-2-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylacetamide —— C19H24N6O2S
N-(3-tert-butyl-1,2-oxazol-5-yl)-2-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylacetamide
—— N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C18H21BrN2O2S
N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— 3-(3,4-Dimethoxyphenyl)-5-(quinazolin-4-ylsulfanylmethyl)-1,2,4-oxadiazole —— C19H16N4O3S
3-(3,4-Dimethoxyphenyl)-5-(quinazolin-4-ylsulfanylmethyl)-1,2,4-oxadiazole
—— N-[2-[di(propan-2-yl)amino]ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide —— C25H32N4O2
N-[2-[di(propan-2-yl)amino]ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide
—— 2-(2,4-dimethyl-5-phenylimidazo[1,5-b]pyridazin-7-yl)sulfanyl-N-(2-methoxyphenyl)acetamide —— C23H22N4O2S
2-(2,4-dimethyl-5-phenylimidazo[1,5-b]pyridazin-7-yl)sulfanyl-N-(2-methoxyphenyl)acetamide
—— N-(1-cyanocyclopentyl)-2-({2,4-dimethyl-5-phenylimidazo[1,5-b]pyridazin-7-yl}sulfanyl)acetamide —— C22H23N5OS
N-(1-cyanocyclopentyl)-2-({2,4-dimethyl-5-phenylimidazo[1,5-b]pyridazin-7-yl}sulfanyl)acetamide
—— (2S)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2S)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2S)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2S)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— 3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-(2-methoxy-5-methylphenyl)ethyl]propanamide —— C21H22ClN3O3
3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-(2-methoxy-5-methylphenyl)ethyl]propanamide
—— 2,4-dimethyl-7-[[(2S)-oxolan-2-yl]methylsulfanyl]-5-phenylimidazo[1,5-b]pyridazine —— C19H21N3OS
2,4-dimethyl-7-[[(2S)-oxolan-2-yl]methylsulfanyl]-5-phenylimidazo[1,5-b]pyridazine
—— N-[(1S)-1-(2-methoxy-5-methylphenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide —— C25H31N3O3
N-[(1S)-1-(2-methoxy-5-methylphenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide
—— N-[(1R)-1-(2-methoxy-5-methylphenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide —— C25H31N3O3
N-[(1R)-1-(2-methoxy-5-methylphenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide
—— 2-[1-(2-Methoxyphenyl)tetrazol-5-yl]sulfanylethanol —— C10H12N4O2S
2-[1-(2-Methoxyphenyl)tetrazol-5-yl]sulfanylethanol
—— (Z)-3-amino-2-[2-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile —— C19H20ClN5O2S
(Z)-3-amino-2-[2-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile
—— 4-[(6,7-Dimethyl-2-oxochromen-4-yl)methylamino]-1,5-dimethyl-2-phenylpyrazol-3-one —— C23H23N3O3
4-[(6,7-Dimethyl-2-oxochromen-4-yl)methylamino]-1,5-dimethyl-2-phenylpyrazol-3-one
—— 1-(3-chlorophenyl)-5-[(1S)-1-(4-fluorophenyl)ethyl]sulfanyltetrazole —— C15H12ClFN4S
1-(3-chlorophenyl)-5-[(1S)-1-(4-fluorophenyl)ethyl]sulfanyltetrazole
—— (2R)-2-[[5-(3-bromophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-propan-2-ylpropanamide —— C15H19BrN4OS
(2R)-2-[[5-(3-bromophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-propan-2-ylpropanamide
—— N-[(1S)-1-cyclopropylethyl]-1-(4-fluorophenyl)-3-(4-methylphenyl)pyrazole-4-carboxamide —— C22H22FN3O
N-[(1S)-1-cyclopropylethyl]-1-(4-fluorophenyl)-3-(4-methylphenyl)pyrazole-4-carboxamide
—— 6-chloro-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-2H-chromene-3-carboxamide —— C23H21ClN4O2
6-chloro-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-2H-chromene-3-carboxamide
—— (Z)-3-amino-2-[2-[[5-(4-chlorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile —— C19H20ClN5O2S
(Z)-3-amino-2-[2-[[5-(4-chlorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile
—— (Z)-3-amino-2-[2-[[5-(4-chlorophenyl)-4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile —— C17H18ClN5O2S
(Z)-3-amino-2-[2-[[5-(4-chlorophenyl)-4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile
—— 3-methyl-1-phenyl-N-(1-propylpiperidin-1-ium-4-yl)thieno[2,3-c]pyrazole-5-carboxamide —— C21H27N4OS+
3-methyl-1-phenyl-N-(1-propylpiperidin-1-ium-4-yl)thieno[2,3-c]pyrazole-5-carboxamide
—— (2R)-1-[(2S)-2-ethylpiperidin-1-yl]-2-[[4-phenyl-5-(pyrrolidin-1-ium-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propan-1-one —— C23H34N5OS+
(2R)-1-[(2S)-2-ethylpiperidin-1-yl]-2-[[4-phenyl-5-(pyrrolidin-1-ium-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propan-1-one
—— N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[5-(2-fluorophenyl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C25H21FN4O3S
N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[5-(2-fluorophenyl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 1-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-(5-phenyltetrazol-2-yl)ethanone —— C16H21N5O
1-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-(5-phenyltetrazol-2-yl)ethanone
—— ethyl N-[2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]carbamate —— C14H17N5O3S
ethyl N-[2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]carbamate
—— 1-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-(5-phenyltetrazol-2-yl)ethanone —— C16H21N5O
1-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-(5-phenyltetrazol-2-yl)ethanone