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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-cyclopropyl-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide —— C16H19N3O
N-cyclopropyl-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide
—— ethyl (4R)-4-methyl-2-oxo-6-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H30N6O3S
ethyl (4R)-4-methyl-2-oxo-6-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-methyl-2-oxo-6-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H30N6O3S
ethyl (4S)-4-methyl-2-oxo-6-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-cyclopropyl-1-(4-fluorophenyl)-3-(3-methylphenyl)pyrazole-4-carboxamide —— C20H18FN3O
N-cyclopropyl-1-(4-fluorophenyl)-3-(3-methylphenyl)pyrazole-4-carboxamide
—— (2R)-N-[(1S)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H26F2N4O2S
(2R)-N-[(1S)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(2-chlorophenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)-1,3-thiazol-4-yl]acetamide —— C16H16ClN3O2S
N-[(2-chlorophenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)-1,3-thiazol-4-yl]acetamide
—— 2-chloro-N'-[2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]benzohydrazide —— C21H22Cl2N6O2S
2-chloro-N'-[2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]benzohydrazide
—— 2-[(2R)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-1-(2-methylpropyl)piperazin-2-yl]ethanol —— C20H29FN4O
2-[(2R)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-1-(2-methylpropyl)piperazin-2-yl]ethanol
—— [2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate —— C21H19ClFN3O3S
[2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate
—— 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3-methoxyphenyl)methyl]-N-methylacetamide —— C24H27FN4O3S
2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3-methoxyphenyl)methyl]-N-methylacetamide
—— 2-[(3-Phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-azaspiro[4.4]nonane-1,3-dione —— C17H17N3O3
2-[(3-Phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-azaspiro[4.4]nonane-1,3-dione
—— ethyl 1-[(2R)-2-[3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carbonyl]oxypropanoyl]piperidine-4-carboxylate —— C22H26FN3O5S
ethyl 1-[(2R)-2-[3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carbonyl]oxypropanoyl]piperidine-4-carboxylate
—— (2S)-N-[(1S)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H26F2N4O2S
(2S)-N-[(1S)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 4-methyl-N-[[2-(pyrrolidin-1-ylmethyl)phenyl]methyl]-2-thiophen-2-yl-1,3-thiazole-5-carboxamide —— C21H23N3OS2
4-methyl-N-[[2-(pyrrolidin-1-ylmethyl)phenyl]methyl]-2-thiophen-2-yl-1,3-thiazole-5-carboxamide
—— (1S)-1-[4-(4-chlorophenyl)-5-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]-N,N-dimethylethanamine —— C21H20ClN7O3S
(1S)-1-[4-(4-chlorophenyl)-5-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]-N,N-dimethylethanamine
—— (2S)-2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide —— C21H22ClFN6O3S
(2S)-2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide
—— 3-(4-acetyl-5-methylfuran-2-yl)-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]propanamide —— C23H26N4O3
3-(4-acetyl-5-methylfuran-2-yl)-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]propanamide
—— (2R)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H26F2N4O2S
(2R)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— ethyl (4S)-4-methyl-2-oxo-6-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H28N6O3S
ethyl (4S)-4-methyl-2-oxo-6-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[(2R)-1-(1-methylpiperidin-4-yl)-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl]ethanol —— C22H32N4OS
2-[(2R)-1-(1-methylpiperidin-4-yl)-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl]ethanol
—— Methyl 3-[1-[4-(cyclopentylcarbamoyl)phenyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C21H27N3O3
Methyl 3-[1-[4-(cyclopentylcarbamoyl)phenyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— [2-oxo-2-[(2E)-2-[(1S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate —— C20H24N6O3
[2-oxo-2-[(2E)-2-[(1S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate
—— N-cyclopentyl-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide —— C18H23N3O
N-cyclopentyl-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide
—— N-cyclopentyl-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C16H18FN3O2
N-cyclopentyl-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— [(2S)-1-[4-(dimethylamino)anilino]-1-oxopropan-2-yl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate —— C22H23FN4O3S
[(2S)-1-[4-(dimethylamino)anilino]-1-oxopropan-2-yl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate
—— 2-[(2R)-4-[(1-methyl-3-phenylpyrazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethanol —— C24H31N5O
2-[(2R)-4-[(1-methyl-3-phenylpyrazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethanol
—— ethyl (4R)-4-methyl-2-oxo-6-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H28N6O3S
ethyl (4R)-4-methyl-2-oxo-6-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-benzyl-N-cyclopentyl-3-(3,4-dimethoxyphenyl)pyrazole-4-carboxamide —— C24H27N3O3
1-benzyl-N-cyclopentyl-3-(3,4-dimethoxyphenyl)pyrazole-4-carboxamide
—— [2-oxo-2-[(2E)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate —— C20H24N6O3
[2-oxo-2-[(2E)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate
—— ethyl (4S)-6-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H29FN6O3S
ethyl (4S)-6-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [2-oxo-2-[(2E)-2-[(1R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate —— C20H24N6O3
[2-oxo-2-[(2E)-2-[(1R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate
—— [2-[[(1R)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate —— C21H19ClFN3O3S
[2-[[(1R)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methoxy-5-methylphenyl)propanamide —— C19H18FN3O3
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methoxy-5-methylphenyl)propanamide
—— (2R)-2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide —— C21H22ClFN6O3S
(2R)-2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide
—— N-cyclopentyl-3-(3,4-dimethoxyphenyl)-1-phenylpyrazole-4-carboxamide —— C23H25N3O3
N-cyclopentyl-3-(3,4-dimethoxyphenyl)-1-phenylpyrazole-4-carboxamide
—— 2-[(2R)-1-[(2-ethoxyphenyl)methyl]-4-[(4-pyrazol-1-ylphenyl)methyl]piperazin-2-yl]ethanol —— C25H32N4O2
2-[(2R)-1-[(2-ethoxyphenyl)methyl]-4-[(4-pyrazol-1-ylphenyl)methyl]piperazin-2-yl]ethanol
—— (2S)-2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide —— C21H22ClFN6O3S
(2S)-2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide
—— 2-chloro-N'-[2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]benzohydrazide —— C21H22Cl2N6O2S
2-chloro-N'-[2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]benzohydrazide
—— [2-oxo-2-[(2E)-2-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate —— C20H24N6O3
[2-oxo-2-[(2E)-2-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]ethyl] 3-(tetrazol-1-yl)benzoate
—— (2R)-2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide —— C21H22ClFN6O3S
(2R)-2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-fluoro-3-nitrophenyl)propanamide
—— 4-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-N-phenyl-1,3-thiazol-2-amine —— C22H23ClN6S2
4-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-N-phenyl-1,3-thiazol-2-amine
—— 2-(4-chlorophenyl)-5-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole —— C22H19ClFN5O2S
2-(4-chlorophenyl)-5-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole
—— 4-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-N-phenyl-1,3-thiazol-2-amine —— C22H23ClN6S2
4-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-N-phenyl-1,3-thiazol-2-amine
—— (2S)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H26F2N4O2S
(2S)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-(4-chlorophenyl)-5-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole —— C22H19ClFN5O2S
2-(4-chlorophenyl)-5-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole
—— N'-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-4-(tetrazol-1-yl)benzohydrazide —— C17H20N6O2
N'-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-4-(tetrazol-1-yl)benzohydrazide
—— 2-[(2R)-1-[(3-methoxyphenyl)methyl]-4-[(3-pyrazol-1-ylphenyl)methyl]piperazin-2-yl]ethanol —— C24H30N4O2
2-[(2R)-1-[(3-methoxyphenyl)methyl]-4-[(3-pyrazol-1-ylphenyl)methyl]piperazin-2-yl]ethanol
—— (1R)-1-[4-(4-chlorophenyl)-5-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]-N,N-dimethylethanamine —— C21H20ClN7O3S
(1R)-1-[4-(4-chlorophenyl)-5-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]-N,N-dimethylethanamine
—— 2-(4-methoxyphenyl)-4-methyl-N-[[2-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]-1,3-thiazole-5-carboxamide —— C24H28N3O2S+
2-(4-methoxyphenyl)-4-methyl-N-[[2-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]-1,3-thiazole-5-carboxamide
—— 2-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]-N-prop-2-enylacetamide —— C20H18ClN3O
2-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]-N-prop-2-enylacetamide