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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide —— C20H27N5OS
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide —— C20H27N5OS
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide —— C20H27N5OS
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(3,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide
—— (2Z,5E)-2-(3,3-dimethyl-2-oxobutylidene)-5-[[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-thiazolidin-4-one —— C20H21N3O3S
(2Z,5E)-2-(3,3-dimethyl-2-oxobutylidene)-5-[[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-thiazolidin-4-one
—— N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(1-phenylpyrazol-4-yl)propanamide —— C21H27N3O
N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(1-phenylpyrazol-4-yl)propanamide
—— N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(1-phenylpyrazol-4-yl)propanamide —— C21H27N3O
N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(1-phenylpyrazol-4-yl)propanamide
—— N-[(1R)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(1-phenylpyrazol-4-yl)propanamide —— C21H27N3O
N-[(1R)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(1-phenylpyrazol-4-yl)propanamide
—— ethyl (4R)-6-[[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H24N6O3S
ethyl (4R)-6-[[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide —— C20H25N3O
2-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide
—— [(Z)-4-amino-3-cyano-2-oxopent-3-enyl] 1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazole-3-carboxylate —— C20H19FN4O3
[(Z)-4-amino-3-cyano-2-oxopent-3-enyl] 1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazole-3-carboxylate
—— (2R)-N-tert-butyl-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C16H23N5OS
(2R)-N-tert-butyl-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— 2-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide —— C20H25N3O
2-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide
—— (2S)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(2-phenylethyl)propanamide —— C20H23N5OS
(2S)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(2-phenylethyl)propanamide
—— [(1R)-1-(2-chlorophenyl)ethyl]-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]azanium —— C17H17ClN3O+
[(1R)-1-(2-chlorophenyl)ethyl]-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]azanium
—— (Z)-3-amino-2-[2-[[5-(4-fluorophenyl)-1,3-oxazol-2-yl]sulfanyl]acetyl]but-2-enenitrile —— C15H12FN3O2S
(Z)-3-amino-2-[2-[[5-(4-fluorophenyl)-1,3-oxazol-2-yl]sulfanyl]acetyl]but-2-enenitrile
—— N-[2-(dimethylamino)ethyl]-2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C29H30FN5O2S2
N-[2-(dimethylamino)ethyl]-2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— (4R)-2-(1,3-dihydrobenzimidazol-2-ylidene)-4-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-3-oxopentanenitrile —— C21H19N7OS
(4R)-2-(1,3-dihydrobenzimidazol-2-ylidene)-4-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-3-oxopentanenitrile
—— (2S)-N-(2,5-dimethylphenyl)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C20H23N5OS
(2S)-N-(2,5-dimethylphenyl)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— 2-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide —— C20H25N3O
2-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide
—— 2-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide —— C20H25N3O
2-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-N-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]acetamide
—— (2S)-N-benzyl-N-tert-butyl-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C23H29N5OS
(2S)-N-benzyl-N-tert-butyl-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— N-[2-(dimethylamino)ethyl]-2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C29H30FN5O2S2
N-[2-(dimethylamino)ethyl]-2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— [(1R)-1-(2-chlorophenyl)ethyl]-[[2-(4-methylphenyl)-1,3-thiazol-4-yl]methyl]azanium —— C19H20ClN2S+
[(1R)-1-(2-chlorophenyl)ethyl]-[[2-(4-methylphenyl)-1,3-thiazol-4-yl]methyl]azanium
—— 4-[(2S)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanoyl]-1,3-dihydroquinoxalin-2-one —— C20H20N6O2S
4-[(2S)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanoyl]-1,3-dihydroquinoxalin-2-one
—— 2-[4,5-dimethyl-1-(2-methylpropyl)imidazol-2-yl]sulfanyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide —— C19H33N3O3S2
2-[4,5-dimethyl-1-(2-methylpropyl)imidazol-2-yl]sulfanyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide
—— (2S)-N-(2-chlorophenyl)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C18H18ClN5OS
(2S)-N-(2-chlorophenyl)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2S)-N-tert-butyl-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C16H23N5OS
(2S)-N-tert-butyl-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2R)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-propylpropanamide —— C15H21N5OS
(2R)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-propylpropanamide
—— 2-[4,5-dimethyl-1-(2-methylpropyl)imidazol-2-yl]sulfanyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide —— C19H33N3O3S2
2-[4,5-dimethyl-1-(2-methylpropyl)imidazol-2-yl]sulfanyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide
—— (2S)-N-(2,3-dihydro-1H-inden-5-yl)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H23N5OS
(2S)-N-(2,3-dihydro-1H-inden-5-yl)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— N-[[4-(dimethylamino)phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide —— C23H28N4O
N-[[4-(dimethylamino)phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide
—— (2R)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(2-oxo-1,3-dihydrobenzimidazol-5-yl)propanamide —— C19H19N7O2S
(2R)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(2-oxo-1,3-dihydrobenzimidazol-5-yl)propanamide
—— [3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (5R,7R)-3-bromoadamantane-1-carboxylate —— C22H25BrN2O5
[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (5R,7R)-3-bromoadamantane-1-carboxylate
—— (2S)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-phenylbutyl]propanamide —— C26H31FN4O2S
(2S)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-phenylbutyl]propanamide
—— [(1S)-1-(2-chlorophenyl)ethyl]-[[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl]azanium —— C18H17Cl2N2S+
[(1S)-1-(2-chlorophenyl)ethyl]-[[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl]azanium
—— (1S)-1-(2-chlorophenyl)-N-[[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl]ethanamine —— C18H16Cl2N2S
(1S)-1-(2-chlorophenyl)-N-[[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl]ethanamine
—— N-methyl-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C24H23N5O2S
N-methyl-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— 1-benzyl-N-[[4-(dimethylamino)phenyl]methyl]pyrazole-4-carboxamide —— C20H22N4O
1-benzyl-N-[[4-(dimethylamino)phenyl]methyl]pyrazole-4-carboxamide
—— (2R)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-phenylbutyl]propanamide —— C26H31FN4O2S
(2R)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-phenylbutyl]propanamide
—— N-[[4-(dimethylamino)phenyl]methyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide —— C22H26N4O
N-[[4-(dimethylamino)phenyl]methyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide
—— 1-butyl-5-chloro-N-[[4-(dimethylamino)phenyl]methyl]-3-methylpyrazole-4-carboxamide —— C18H25ClN4O
1-butyl-5-chloro-N-[[4-(dimethylamino)phenyl]methyl]-3-methylpyrazole-4-carboxamide
—— (1S,2S)-N,2-dimethyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]cyclopropane-1-carboxamide —— C16H20N4O
(1S,2S)-N,2-dimethyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]cyclopropane-1-carboxamide
—— (4-pyrazol-1-ylphenyl)methyl 2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetate —— C19H22N2O2
(4-pyrazol-1-ylphenyl)methyl 2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetate
—— [2-[methyl-[(1R)-1-phenylethyl]amino]-2-oxoethyl] 2-[(4,5-diphenyl-1,2,4-triazol-3-yl)sulfanyl]acetate —— C27H26N4O3S
[2-[methyl-[(1R)-1-phenylethyl]amino]-2-oxoethyl] 2-[(4,5-diphenyl-1,2,4-triazol-3-yl)sulfanyl]acetate
—— (2S)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-phenylbutyl]propanamide —— C26H31FN4O2S
(2S)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-phenylbutyl]propanamide
—— (2R)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-phenylbutyl]propanamide —— C26H31FN4O2S
(2R)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-phenylbutyl]propanamide
—— 2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]acetamide —— C25H29FN4O2S
2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]acetamide
—— (4-pyrazol-1-ylphenyl)methyl 2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetate —— C19H22N2O2
(4-pyrazol-1-ylphenyl)methyl 2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetate
—— [2-[methyl-[(1S)-1-phenylethyl]amino]-2-oxoethyl] 2-[(4,5-diphenyl-1,2,4-triazol-3-yl)sulfanyl]acetate —— C27H26N4O3S
[2-[methyl-[(1S)-1-phenylethyl]amino]-2-oxoethyl] 2-[(4,5-diphenyl-1,2,4-triazol-3-yl)sulfanyl]acetate
—— [(2S)-1-[[(1R,2S,3S)-2,3-dimethylcyclohexyl]amino]-1-oxopropan-2-yl] 1-methylpyrazole-4-carboxylate —— C16H25N3O3
[(2S)-1-[[(1R,2S,3S)-2,3-dimethylcyclohexyl]amino]-1-oxopropan-2-yl] 1-methylpyrazole-4-carboxylate