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—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S)-1-(4-ethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C20H19N3O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S)-1-(4-ethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— 5-chloro-N-[(1R)-1-(furan-2-yl)ethyl]-N,3-dimethyl-1-benzofuran-2-carboxamide —— C17H16ClNO3
5-chloro-N-[(1R)-1-(furan-2-yl)ethyl]-N,3-dimethyl-1-benzofuran-2-carboxamide
—— 5-chloro-6-[(4S)-4-hydroxy-5,8-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile —— C17H16ClN3O3
5-chloro-6-[(4S)-4-hydroxy-5,8-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile
—— 5-chloro-2-fluoro-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]benzamide —— C15H21ClFN3O
5-chloro-2-fluoro-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]benzamide
—— 5-(4-fluorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylfuran-2-carboxamide —— C18H16FNO3
5-(4-fluorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylfuran-2-carboxamide
—— 5-bromo-2-chloro-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylbenzamide —— C14H13BrClNO2
5-bromo-2-chloro-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylbenzamide
—— 5-(4-fluorophenyl)-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylfuran-2-carboxamide —— C18H16FNO3
5-(4-fluorophenyl)-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylfuran-2-carboxamide
—— 5-chloro-6-[(4R)-4-hydroxy-5,8-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile —— C17H16ClN3O3
5-chloro-6-[(4R)-4-hydroxy-5,8-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile
—— 5-bromo-2-chloro-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylbenzamide —— C14H13BrClNO2
5-bromo-2-chloro-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylbenzamide
—— 5-bromo-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide —— C13H13BrN2O2
5-bromo-N-[(1S)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide
—— 5-chloro-N-[(1S)-1-(furan-2-yl)ethyl]-N,3-dimethyl-1-benzofuran-2-carboxamide —— C17H16ClNO3
5-chloro-N-[(1S)-1-(furan-2-yl)ethyl]-N,3-dimethyl-1-benzofuran-2-carboxamide
—— 5-bromo-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide —— C13H13BrN2O2
5-bromo-N-[(1R)-1-(furan-2-yl)ethyl]-N-methylpyridine-3-carboxamide
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C17H21N3OS
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5-acetyl-2-methoxyphenyl)methyl (3R)-1-(4-methylphenyl)-5-oxopyrrolidine-3-carboxylate —— C22H23NO5
(5-acetyl-2-methoxyphenyl)methyl (3R)-1-(4-methylphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5S,5aR)-3-methyl-1-phenyl-5-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)-5a,6,7,8-tetrahydro-4H-pyrazolo[3,4-e]indolizine-5-carbonitrile —— C24H27N7
(5S,5aR)-3-methyl-1-phenyl-5-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)-5a,6,7,8-tetrahydro-4H-pyrazolo[3,4-e]indolizine-5-carbonitrile
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C17H21N3OS
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5S,5aS)-3-methyl-1-phenyl-5-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)-5a,6,7,8-tetrahydro-4H-pyrazolo[3,4-e]indolizine-5-carbonitrile —— C24H27N7
(5S,5aS)-3-methyl-1-phenyl-5-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)-5a,6,7,8-tetrahydro-4H-pyrazolo[3,4-e]indolizine-5-carbonitrile
—— (5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H21ClN4O2
(5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H21ClN4O2
(5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-methylpyrazin-2-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C15H19N5O
(5-methylpyrazin-2-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5-ethyl-1-phenylpyrazol-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C20H23N5O
(5-ethyl-1-phenylpyrazol-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-bromofuran-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C13H14BrN3O2
(5-bromofuran-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C16H19N7O
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-methyl-1,2-oxazol-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C13H16N4O2
(5-methyl-1,2-oxazol-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— [5-methyl-1-(3-methylphenyl)pyrazol-4-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C20H23N5O
[5-methyl-1-(3-methylphenyl)pyrazol-4-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C16H19N3OS
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-methylpyrazin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C14H17N5O
(5-methylpyrazin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-methylimidazo[1,2-a]pyridin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H19N5O
(5-methylimidazo[1,2-a]pyridin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— [5-methyl-1-(3-methylphenyl)pyrazol-4-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C20H23N5O
[5-methyl-1-(3-methylphenyl)pyrazol-4-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H21N3O4
(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-methylimidazo[1,2-a]pyridin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H19N5O
(5-methylimidazo[1,2-a]pyridin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5Z)-5-[(2E)-2-(5-chloro-3-methyl-1,3-benzothiazol-2-ylidene)ethylidene]-3-propyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C16H15ClN2OS3
(5Z)-5-[(2E)-2-(5-chloro-3-methyl-1,3-benzothiazol-2-ylidene)ethylidene]-3-propyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]thiophene-2-carboxamide —— C16H20N4O2S
5-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]thiophene-2-carboxamide
—— (5-methyl-1H-indazol-7-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C19H23N5O
(5-methyl-1H-indazol-7-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (5-methylfuro[3,2-b]pyridin-2-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C19H22N4O2
(5-methylfuro[3,2-b]pyridin-2-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (5-methyl-1,2-oxazol-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C13H16N4O2
(5-methyl-1,2-oxazol-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one —— C18H21N5O2
5-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one
—— (5R)-5-[2-chloro-4-(dimethylamino)-5-nitrophenyl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C27H26ClN3O3
(5R)-5-[2-chloro-4-(dimethylamino)-5-nitrophenyl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C16H19N7O
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]thiophene-2-carboxamide —— C16H20N4O2S
5-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]thiophene-2-carboxamide
—— (5E)-5-[(4-tert-butylphenyl)methylidene]-1-methyl-3-propan-2-yl-2-sulfanylideneimidazolidin-4-one —— C18H24N2OS
(5E)-5-[(4-tert-butylphenyl)methylidene]-1-methyl-3-propan-2-yl-2-sulfanylideneimidazolidin-4-one
—— (5S)-5-[1-[(2-chlorophenyl)methyl]indol-3-yl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C34H29ClN2O
(5S)-5-[1-[(2-chlorophenyl)methyl]indol-3-yl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— (5Z)-5-[(2E)-2-(3-ethyl-6,7,8,9-tetrahydrobenzo[g][1,3]benzothiazol-2-ylidene)ethylidene]-3-propyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H24N2OS3
(5Z)-5-[(2E)-2-(3-ethyl-6,7,8,9-tetrahydrobenzo[g][1,3]benzothiazol-2-ylidene)ethylidene]-3-propyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5-methyl-1H-indazol-7-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C19H23N5O
(5-methyl-1H-indazol-7-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (5-methylpyrazin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C14H17N5O
(5-methylpyrazin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5S)-5-[2-chloro-4-(dimethylamino)-5-nitrophenyl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C27H26ClN3O3
(5S)-5-[2-chloro-4-(dimethylamino)-5-nitrophenyl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— (5R)-5-(2,4-dimorpholin-4-yl-5-nitrophenyl)-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C33H36N4O5
(5R)-5-(2,4-dimorpholin-4-yl-5-nitrophenyl)-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— (5S)-5-(3,5-dichloro-2-phenylmethoxyphenyl)-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C32H27Cl2NO2
(5S)-5-(3,5-dichloro-2-phenylmethoxyphenyl)-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— (5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C18H22N6O
(5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (5R)-5-(3-methoxy-4-propan-2-yloxyphenyl)-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C29H31NO3
(5R)-5-(3-methoxy-4-propan-2-yloxyphenyl)-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one