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—— 5-[(3S)-1-[(5,7-dimethylimidazo[1,2-a]pyrimidin-2-yl)methyl]piperidin-3-yl]-3-methyl-1,2,4-oxadiazole —— C17H22N6O
5-[(3S)-1-[(5,7-dimethylimidazo[1,2-a]pyrimidin-2-yl)methyl]piperidin-3-yl]-3-methyl-1,2,4-oxadiazole
—— 5,6-dimethyl-2-[[5-oxo-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C16H19N5O3S2
5,6-dimethyl-2-[[5-oxo-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5S)-2-oxo-5-(pyridine-2-carbonylamino)-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C16H16N4O3
(5S)-2-oxo-5-(pyridine-2-carbonylamino)-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 5,6-dimethyl-2-[[5-oxo-4-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C19H19N5O2S2
5,6-dimethyl-2-[[5-oxo-4-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5R)-5-[(5-ethyl-4-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C18H21N3O3S
(5R)-5-[(5-ethyl-4-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 5,6-dimethyl-2-[(1S)-1-[(5-oxo-4-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C15H19N5O2S2
5,6-dimethyl-2-[(1S)-1-[(5-oxo-4-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-(furan-2-yl)-3-[2-oxo-2-[(4R)-2-oxo-4-(trifluoromethyl)-3,4-dihydro-1H-1,5-benzodiazepin-5-yl]ethyl]-1,3,4-oxadiazol-2-one —— C18H13F3N4O5
5-(furan-2-yl)-3-[2-oxo-2-[(4R)-2-oxo-4-(trifluoromethyl)-3,4-dihydro-1H-1,5-benzodiazepin-5-yl]ethyl]-1,3,4-oxadiazol-2-one
—— (5S)-5-[[2-(6-methoxy-1-benzofuran-3-yl)acetyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C21H21N3O5
(5S)-5-[[2-(6-methoxy-1-benzofuran-3-yl)acetyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 5,6-dimethyl-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C16H14N4O3S2
5,6-dimethyl-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5R)-5-(1-benzofuran-2-carbonylamino)-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C19H17N3O4
(5R)-5-(1-benzofuran-2-carbonylamino)-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5S)-5-[[2-(2-fluorophenyl)acetyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C18H18FN3O3
(5S)-5-[[2-(2-fluorophenyl)acetyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5S)-2-oxo-5-[(1-phenylcyclopropanecarbonyl)amino]-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C20H21N3O3
(5S)-2-oxo-5-[(1-phenylcyclopropanecarbonyl)amino]-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 5-(furan-2-yl)-3-[2-oxo-2-[(4S)-2-oxo-4-(trifluoromethyl)-3,4-dihydro-1H-1,5-benzodiazepin-5-yl]ethyl]-1,3,4-oxadiazol-2-one —— C18H13F3N4O5
5-(furan-2-yl)-3-[2-oxo-2-[(4S)-2-oxo-4-(trifluoromethyl)-3,4-dihydro-1H-1,5-benzodiazepin-5-yl]ethyl]-1,3,4-oxadiazol-2-one
—— (5R)-5-[(2,4-dichlorobenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C17H15Cl2N3O3
(5R)-5-[(2,4-dichlorobenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5S)-5-(1-benzofuran-2-carbonylamino)-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C19H17N3O4
(5S)-5-(1-benzofuran-2-carbonylamino)-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5S)-5-[(5-ethyl-4-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C18H21N3O3S
(5S)-5-[(5-ethyl-4-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5R)-5-[(5-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C16H17N3O3S
(5R)-5-[(5-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5R)-5-[[2-(6-methoxy-1-benzofuran-3-yl)acetyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C21H21N3O5
(5R)-5-[[2-(6-methoxy-1-benzofuran-3-yl)acetyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5-Acetyl-2-methoxyphenyl)methyl 2-(5-methyl-2-propan-2-ylphenoxy)acetate —— C22H26O5
(5-Acetyl-2-methoxyphenyl)methyl 2-(5-methyl-2-propan-2-ylphenoxy)acetate
—— (5S)-5-[(3-cyanobenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C18H16N4O3
(5S)-5-[(3-cyanobenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5S)-5-[(5-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C16H17N3O3S
(5S)-5-[(5-methylthiophene-2-carbonyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5S)-5-[4-(1,3-benzothiazol-2-yl)butanoylamino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C21H22N4O3S
(5S)-5-[4-(1,3-benzothiazol-2-yl)butanoylamino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 5,6-dimethyl-2-[(1S)-1-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C17H16N4O3S2
5,6-dimethyl-2-[(1S)-1-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5S)-5-[(2,4-dichlorobenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C17H15Cl2N3O3
(5S)-5-[(2,4-dichlorobenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5-propyl-1H-pyrazol-3-yl)-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone —— C16H26N4O
(5-propyl-1H-pyrazol-3-yl)-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone
—— (5-methyl-1-benzofuran-2-yl)-[4-[(2R)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone —— C20H26N2O3
(5-methyl-1-benzofuran-2-yl)-[4-[(2R)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 3-(trifluoromethyl)benzoate —— C18H12F3NO3
(5-Phenyl-1,3-oxazol-2-yl)methyl 3-(trifluoromethyl)benzoate
—— 5,6-dimethyl-2-[(1R)-1-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C17H16N4O3S2
5,6-dimethyl-2-[(1R)-1-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5-propyl-1H-pyrazol-3-yl)-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone —— C16H26N4O
(5-propyl-1H-pyrazol-3-yl)-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone
—— 5-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]-N-(2-phenylethyl)-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C22H28N4OS
5-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]-N-(2-phenylethyl)-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— (5-methyl-1-benzofuran-2-yl)-[4-[(2S)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone —— C20H26N2O3
(5-methyl-1-benzofuran-2-yl)-[4-[(2S)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone
—— (5R)-5-methyl-1-phenyl-3-(thiomorpholine-4-carbonyl)-2,5-dihydro-1,2,4-triazin-6-one —— C15H18N4O2S
(5R)-5-methyl-1-phenyl-3-(thiomorpholine-4-carbonyl)-2,5-dihydro-1,2,4-triazin-6-one
—— (5S)-3-(2,4-dichlorophenyl)-N-[2-(1-methylpyrazol-4-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H16Cl2N4O2
(5S)-3-(2,4-dichlorophenyl)-N-[2-(1-methylpyrazol-4-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-5-methyl-1-phenyl-3-(thiomorpholine-4-carbonyl)-2,5-dihydro-1,2,4-triazin-6-one —— C15H18N4O2S
(5S)-5-methyl-1-phenyl-3-(thiomorpholine-4-carbonyl)-2,5-dihydro-1,2,4-triazin-6-one
—— 5-[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]-N-(2-phenylethyl)-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C22H28N4OS
5-[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]-N-(2-phenylethyl)-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— (5-propan-2-yl-1H-pyrazol-3-yl)-[(2R)-2-pyridin-4-ylazepan-1-yl]methanone —— C18H24N4O
(5-propan-2-yl-1H-pyrazol-3-yl)-[(2R)-2-pyridin-4-ylazepan-1-yl]methanone
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3-(trifluoromethyl)benzoate —— C15H9F3N2O4
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3-(trifluoromethyl)benzoate
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 3-(trifluoromethyl)benzoate —— C17H10ClF3N2O3
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 3-(trifluoromethyl)benzoate
—— (5-propan-2-yl-1H-pyrazol-3-yl)-[(2S)-2-pyridin-4-ylazepan-1-yl]methanone —— C18H24N4O
(5-propan-2-yl-1H-pyrazol-3-yl)-[(2S)-2-pyridin-4-ylazepan-1-yl]methanone
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 3-chlorobenzoate —— C17H12ClNO3
(5-Phenyl-1,3-oxazol-2-yl)methyl 3-chlorobenzoate
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone —— C16H18N2O2S
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone —— C16H18N2O2S
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 3-chlorobenzoate —— C16H10Cl2N2O3
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 3-chlorobenzoate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 4-(trifluoromethyl)benzoate —— C18H12F3NO3
(5-Phenyl-1,3-oxazol-2-yl)methyl 4-(trifluoromethyl)benzoate
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-(trifluoromethyl)benzoate —— C15H9F3N2O4
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-(trifluoromethyl)benzoate
—— (5-Methyl-1,3,4-oxadiazol-2-yl)methyl 4-phenoxybenzoate —— C17H14N2O4
(5-Methyl-1,3,4-oxadiazol-2-yl)methyl 4-phenoxybenzoate
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-phenoxybenzoate —— C20H14N2O5
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-phenoxybenzoate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-(trifluoromethyl)benzoate —— C18H12F3NO3
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-(trifluoromethyl)benzoate
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(trifluoromethyl)benzoate —— C17H10F3N3O5
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(trifluoromethyl)benzoate
—— 5-[2-[(2S)-2-[(4-fluorophenyl)methyl]pyrrolidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one —— C19H22FN3O2
5-[2-[(2S)-2-[(4-fluorophenyl)methyl]pyrrolidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one