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—— 5-[(1R)-1-[4-(4-methylpiperazin-1-yl)sulfonylpiperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C19H28N6O3S
5-[(1R)-1-[4-(4-methylpiperazin-1-yl)sulfonylpiperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[[(1S)-6,7-dimethoxy-1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-N,N-dimethylfuran-2-sulfonamide —— C24H28N2O5S
5-[[(1S)-6,7-dimethoxy-1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-N,N-dimethylfuran-2-sulfonamide
—— 5-[[(1R)-6,7-dimethoxy-1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-N,N-dimethylfuran-2-sulfonamide —— C24H28N2O5S
5-[[(1R)-6,7-dimethoxy-1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-N,N-dimethylfuran-2-sulfonamide
—— 5-[[(1S)-6,7-dimethoxy-1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-3-(4-nitrophenyl)-1,2,4-oxadiazole —— C26H24N4O5
5-[[(1S)-6,7-dimethoxy-1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-3-(4-nitrophenyl)-1,2,4-oxadiazole
—— (5S,7R)-3-chloro-N-[(2,4-dichlorophenyl)methyl]adamantane-1-carboxamide —— C18H20Cl3NO
(5S,7R)-3-chloro-N-[(2,4-dichlorophenyl)methyl]adamantane-1-carboxamide
—— 5,6-dichloro-N-(3-phenylpropyl)pyridine-3-carboxamide —— C15H14Cl2N2O
5,6-dichloro-N-(3-phenylpropyl)pyridine-3-carboxamide
—— 5-bromo-N-methyl-N-[2-oxo-2-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methylamino]ethyl]thiophene-2-carboxamide —— C25H23BrN2O2S
5-bromo-N-methyl-N-[2-oxo-2-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methylamino]ethyl]thiophene-2-carboxamide
—— (5S,7R)-3-bromo-N-[(2,4-dichlorophenyl)methyl]adamantane-1-carboxamide —— C18H20BrCl2NO
(5S,7R)-3-bromo-N-[(2,4-dichlorophenyl)methyl]adamantane-1-carboxamide
—— 5-bromo-N-[2-[[(2R)-3-ethyl-2-morpholin-4-ylpentyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C19H30BrN3O3S
5-bromo-N-[2-[[(2R)-3-ethyl-2-morpholin-4-ylpentyl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-bromo-N-[2-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propylamino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C17H26BrN3O3S
5-bromo-N-[2-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propylamino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— (5Z)-5-[(3-methylthiophen-2-yl)methylidene]-2-thioxoimidazolidin-4-one —— C9H8N2OS2
(5Z)-5-[(3-methylthiophen-2-yl)methylidene]-2-thioxoimidazolidin-4-one
—— 5-bromo-N-[2-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propylamino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C17H26BrN3O3S
5-bromo-N-[2-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propylamino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— (5Z)-5-[(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C18H13N5OS
(5Z)-5-[(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— 5-bromo-N-[2-[[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C18H23BrN4O3S2
5-bromo-N-[2-[[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— (5Z)-5-[[3,4-bis(phenylmethoxy)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C24H20N2O3S
(5Z)-5-[[3,4-bis(phenylmethoxy)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— 5-[(2S)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C19H17N5O5S
5-[(2S)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2R)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C24H24ClN5O5
5-[(2R)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— (5S,7R)-3-bromo-N-cycloheptyladamantane-1-carboxamide —— C18H28BrNO
(5S,7R)-3-bromo-N-cycloheptyladamantane-1-carboxamide
—— 5-[(2-cyanophenoxy)methyl]-N-[4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]furan-2-carboxamide —— C23H24N4O4S
5-[(2-cyanophenoxy)methyl]-N-[4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]furan-2-carboxamide
—— 5-[(2R)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H15Cl2N5O5
5-[(2R)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— (5S)-N-[(2,4-dichlorophenyl)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H17Cl2NOS
(5S)-N-[(2,4-dichlorophenyl)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-bromo-N-[2-[3-[(2S,6R)-2,6-dimethylmorpholin-4-yl]propylamino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C17H26BrN3O3S
5-bromo-N-[2-[3-[(2S,6R)-2,6-dimethylmorpholin-4-yl]propylamino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-[(2R)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C19H17N5O5S
5-[(2R)-2-hydroxy-3-(thiophen-2-ylmethoxy)propyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-chloro-N-[(2,4-dichlorophenyl)methyl]thiophene-2-carboxamide —— C12H8Cl3NOS
5-chloro-N-[(2,4-dichlorophenyl)methyl]thiophene-2-carboxamide
—— 5-[(2S)-3-(5,6-dimethylbenzimidazol-1-yl)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C23H21FN6O2
5-[(2S)-3-(5,6-dimethylbenzimidazol-1-yl)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— (5Z)-5-[[3-ethoxy-4-(2-methylpropoxy)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C16H20N2O3S
(5Z)-5-[[3-ethoxy-4-(2-methylpropoxy)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— 5-[(2R)-3-(3,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C22H21N5O5
5-[(2R)-3-(3,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2S)-3-(2,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C22H21N5O5
5-[(2S)-3-(2,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-2-chloro-N-[(2,4-dichlorophenyl)methyl]benzamide —— C14H9BrCl3NO
5-bromo-2-chloro-N-[(2,4-dichlorophenyl)methyl]benzamide
—— 5,6-dichloro-N-[2-(4-chlorophenyl)ethyl]pyridine-3-carboxamide —— C14H11Cl3N2O
5,6-dichloro-N-[2-(4-chlorophenyl)ethyl]pyridine-3-carboxamide
—— 5-[(2R)-3-(2,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C22H21N5O5
5-[(2R)-3-(2,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-N-[(2R)-1-oxo-1-[[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]amino]propan-2-yl]thiophene-2-carboxamide —— C17H21BrN4O2S2
5-bromo-N-[(2R)-1-oxo-1-[[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]amino]propan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-[[4-[(4-methylpiperidin-1-yl)methyl]-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H23BrN4O2S2
5-bromo-N-[(2S)-1-[[4-[(4-methylpiperidin-1-yl)methyl]-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-1-[[4-[(4-methylpiperidin-1-yl)methyl]-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H23BrN4O2S2
5-bromo-N-[(2R)-1-[[4-[(4-methylpiperidin-1-yl)methyl]-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-[(2-cyanophenoxy)methyl]-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]furan-2-carboxamide —— C23H24N4O4S
5-[(2-cyanophenoxy)methyl]-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]furan-2-carboxamide
—— 5-[(2-cyanophenoxy)methyl]-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]furan-2-carboxamide —— C23H24N4O4S
5-[(2-cyanophenoxy)methyl]-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]furan-2-carboxamide
—— 5-[(2S)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C24H24ClN5O5
5-[(2S)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2S)-3-(3,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C22H21N5O5
5-[(2S)-3-(3,5-dimethylphenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2S)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H15Cl2N5O5
5-[(2S)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-N-[2-[[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C18H23BrN4O3S2
5-bromo-N-[2-[[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-bromo-N-[2-[[4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C18H23BrN4O3S2
5-bromo-N-[2-[[4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]amino]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-oxo-1-[[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]amino]propan-2-yl]thiophene-2-carboxamide —— C17H21BrN4O2S2
5-bromo-N-[(2S)-1-oxo-1-[[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]amino]propan-2-yl]thiophene-2-carboxamide
—— (5S)-5-(2,3-dihydro-1H-inden-5-yl)-3-[(2R)-3-(5,6-dimethylbenzimidazol-1-yl)-2-hydroxypropyl]-5-methylimidazolidine-2,4-dione —— C25H28N4O3
(5S)-5-(2,3-dihydro-1H-inden-5-yl)-3-[(2R)-3-(5,6-dimethylbenzimidazol-1-yl)-2-hydroxypropyl]-5-methylimidazolidine-2,4-dione
—— 5-bromo-N-[(2R)-1-[3-(cyclopropylcarbamoyl)anilino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H18BrN3O3S
5-bromo-N-[(2R)-1-[3-(cyclopropylcarbamoyl)anilino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— (5R)-N-[(2,4-dichlorophenyl)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H17Cl2NOS
(5R)-N-[(2,4-dichlorophenyl)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5Z)-5-[(3-chloro-5-ethoxy-4-methoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C13H13ClN2O3S
(5Z)-5-[(3-chloro-5-ethoxy-4-methoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— 5-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-N-[(1R,2S)-2-methylcyclohexyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C24H32N4S
5-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-N-[(1R,2S)-2-methylcyclohexyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— 5-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-N-[(1S,2R)-2-methylcyclohexyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C24H32N4S
5-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-N-[(1S,2R)-2-methylcyclohexyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— 5-[(2Z)-2-[(5-methylfuran-2-yl)methylidene]hydrazinyl]-1,2-dihydro-1,2,4-triazole-3-thione —— C8H9N5OS
5-[(2Z)-2-[(5-methylfuran-2-yl)methylidene]hydrazinyl]-1,2-dihydro-1,2,4-triazole-3-thione
—— 5,6-dichloro-N-[2-(2,6-difluoroanilino)-2-oxoethyl]-N-ethylpyridine-3-carboxamide —— C16H13Cl2F2N3O2
5,6-dichloro-N-[2-(2,6-difluoroanilino)-2-oxoethyl]-N-ethylpyridine-3-carboxamide