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—— [5-[[(3S)-3-hydroxypiperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone —— C16H22N4O2S
[5-[[(3S)-3-hydroxypiperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone
—— 5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C19H24N4O3
5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— (5-fluoro-2-methoxyphenyl)-[(3R)-1-(6-methylpyridazin-3-yl)piperidin-3-yl]methanone —— C18H20FN3O2
(5-fluoro-2-methoxyphenyl)-[(3R)-1-(6-methylpyridazin-3-yl)piperidin-3-yl]methanone
—— 5-[2-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H30N4O3
5-[2-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-[3-[(2R)-2-(3,4-dichlorophenyl)morpholin-4-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C16H16Cl2N2O4
5-[3-[(2R)-2-(3,4-dichlorophenyl)morpholin-4-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C19H24N4O3
5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— 5-methoxy-2-[(3R)-3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-4-one —— C21H26N2O4
5-methoxy-2-[(3R)-3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-4-one
—— (5-Acetyl-2-methoxyphenyl)methyl 2-(thiophene-2-carbonylamino)acetate —— C17H17NO5S
(5-Acetyl-2-methoxyphenyl)methyl 2-(thiophene-2-carbonylamino)acetate
—— 5-methoxy-2-[(3S)-3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-4-one —— C21H26N2O4
5-methoxy-2-[(3S)-3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-4-one
—— [(5R)-3-ethyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-(3-methylpyridin-2-yl)piperazin-1-yl]methanone —— C16H22N4O2
[(5R)-3-ethyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-(3-methylpyridin-2-yl)piperazin-1-yl]methanone
—— (5R)-N-[2-(2-fluorophenoxy)ethyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C13H15FN2O3
(5R)-N-[2-(2-fluorophenoxy)ethyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[1-[(1S)-1-pyridin-4-ylpropyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C19H17N5S
5-[1-[(1S)-1-pyridin-4-ylpropyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-[(2-ethoxybenzoyl)amino]acetate —— C20H19N3O5
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-[(2-ethoxybenzoyl)amino]acetate
—— (5S)-N-[2-(2-fluorophenoxy)ethyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C13H15FN2O3
(5S)-N-[2-(2-fluorophenoxy)ethyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-9-(pyridin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H20N2O2
(5R)-9-(pyridin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-N-[3-(1,3-benzothiazol-2-yl)propyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H17N3O2S
(5R)-N-[3-(1,3-benzothiazol-2-yl)propyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [(5S)-3-ethyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-(3-methylpyridin-2-yl)piperazin-1-yl]methanone —— C16H22N4O2
[(5S)-3-ethyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-(3-methylpyridin-2-yl)piperazin-1-yl]methanone
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate —— C20H15NO5
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate
—— (5-Acetyl-2-ethoxyphenyl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate —— C21H20O6
(5-Acetyl-2-ethoxyphenyl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate
—— (5-Fluoro-2-methoxyphenyl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate —— C18H15FO5
(5-Fluoro-2-methoxyphenyl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate —— C17H12N2O5S
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate
—— (5-Acetyl-2-methoxyphenyl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate —— C20H18O6
(5-Acetyl-2-methoxyphenyl)methyl 2-(6-hydroxy-1-benzofuran-3-yl)acetate
—— 5-[[2-[(3R)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole —— C17H26N4O
5-[[2-[(3R)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole
—— (5S)-9-(pyridin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H20N2O2
(5S)-9-(pyridin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-N-[3-(1,3-benzothiazol-2-yl)propyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H17N3O2S
(5S)-N-[3-(1,3-benzothiazol-2-yl)propyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[1-[[(1R)-3,4-dihydro-1H-isochromen-1-yl]methyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine —— C20H22N4O
5-[1-[[(1R)-3,4-dihydro-1H-isochromen-1-yl]methyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine
—— 5-[1-[(1R)-1-pyridin-4-ylpropyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C19H17N5S
5-[1-[(1R)-1-pyridin-4-ylpropyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— (5S)-N-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C12H17N3O3
(5S)-N-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[1-[[(1S)-3,4-dihydro-1H-isochromen-1-yl]methyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine —— C20H22N4O
5-[1-[[(1S)-3,4-dihydro-1H-isochromen-1-yl]methyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine
—— 5-[[2-[(3S)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole —— C17H26N4O
5-[[2-[(3S)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole
—— (5-methyl-1H-imidazol-4-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C19H22F3N3O
(5-methyl-1H-imidazol-4-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (5R)-N-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C12H17N3O3
(5R)-N-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5-methyl-1H-imidazol-4-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C19H22F3N3O
(5-methyl-1H-imidazol-4-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— 5-amino-1-[(2S)-2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pentan-1-one —— C20H26N2O3
5-amino-1-[(2S)-2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pentan-1-one
—— 5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine —— C20H26F2N4
5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-piperidin-1-ylsulfonylbenzoate —— C19H19N3O6S
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-piperidin-1-ylsulfonylbenzoate
—— 5-amino-1-[(2R)-2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pentan-1-one —— C20H26N2O3
5-amino-1-[(2R)-2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pentan-1-one
—— (5R)-9-[(2,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H19F2NO2
(5R)-9-[(2,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine —— C20H26F2N4
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine
—— 5-tert-butyl-4-[[(2R)-2-(4-fluorophenyl)morpholin-4-yl]methyl]furan-2-carboxamide —— C20H25FN2O3
5-tert-butyl-4-[[(2R)-2-(4-fluorophenyl)morpholin-4-yl]methyl]furan-2-carboxamide
—— 5-tert-butyl-4-[[(2S)-2-(4-fluorophenyl)morpholin-4-yl]methyl]furan-2-carboxamide —— C20H25FN2O3
5-tert-butyl-4-[[(2S)-2-(4-fluorophenyl)morpholin-4-yl]methyl]furan-2-carboxamide
—— (5S)-9-[(2,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H19F2NO2
(5S)-9-[(2,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-phenylsulfanylpropanoate —— C18H16N2O3S
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-phenylsulfanylpropanoate
—— [5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (2S)-2-phenylsulfanylpropanoate —— C16H14N2O4S
[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (2S)-2-phenylsulfanylpropanoate
—— (5R)-5-[2-(2-methyl-4-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-2-oxoethyl]pyrrolidin-2-one —— C18H25N5O2
(5R)-5-[2-(2-methyl-4-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-2-oxoethyl]pyrrolidin-2-one
—— [5-[[methyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone —— C18H26N4O2S
[5-[[methyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone
—— 5-[1-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine —— C17H22N6
5-[1-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2R)-2-acetamido-3-methylbutanoate —— C16H19N3O4
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2R)-2-acetamido-3-methylbutanoate
—— (5R)-9-[(6-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H22N2O2
(5R)-9-[(6-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[1-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine —— C17H22N6
5-[1-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]imidazol-2-yl]-N,N-dimethylpyridin-2-amine