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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-9-(3-phenylpropyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H25NO2
(5R)-9-(3-phenylpropyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-ethyl-1H-pyrazol-4-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H24F3N3O
(5-ethyl-1H-pyrazol-4-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (5S)-9-[(2-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H20FNO2
(5S)-9-[(2-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-methoxy-2-[[(2R)-2-(trifluoromethyl)morpholin-4-yl]methyl]pyran-4-one —— C12H14F3NO4
5-methoxy-2-[[(2R)-2-(trifluoromethyl)morpholin-4-yl]methyl]pyran-4-one
—— (5-chloropyridin-2-yl)-[(2S)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C17H14ClN5O2
(5-chloropyridin-2-yl)-[(2S)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— 5-[[2-[5-[(2S)-oxan-2-yl]furan-2-yl]imidazol-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C20H19N5O3
5-[[2-[5-[(2S)-oxan-2-yl]furan-2-yl]imidazol-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5R)-1-[4-(benzylsulfamoylamino)phenyl]-5-methylpyrrolidin-2-one —— C18H21N3O3S
(5R)-1-[4-(benzylsulfamoylamino)phenyl]-5-methylpyrrolidin-2-one
—— 5-[4-[(3S)-3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl]-5-oxopentanamide —— C21H37N5O3
5-[4-[(3S)-3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl]-5-oxopentanamide
—— (5R)-9-[(2-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H20FNO2
(5R)-9-[(2-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(4R)-5-[(1-methylimidazol-2-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-propylpyrimidin-2-amine —— C18H24N8
5-[(4R)-5-[(1-methylimidazol-2-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-propylpyrimidin-2-amine
—— (5-ethyl-1H-pyrazol-4-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H24F3N3O
(5-ethyl-1H-pyrazol-4-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (5-chloropyridin-2-yl)-[(2R)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C17H14ClN5O2
(5-chloropyridin-2-yl)-[(2R)-2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (5S)-9-(3-phenylpropyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H25NO2
(5S)-9-(3-phenylpropyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-oxo-4-thiophen-2-ylbutanoate —— C15H12N2O5S
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-oxo-4-thiophen-2-ylbutanoate
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(3-phenylpropyl)morpholin-4-yl]methanone —— C22H26N4O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(3-phenylpropyl)morpholin-4-yl]methanone
—— (5-Acetyl-2-ethoxyphenyl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate —— C19H22N2O6S
(5-Acetyl-2-ethoxyphenyl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate
—— 5-[(4S)-5-[(1-methylimidazol-2-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-propylpyrimidin-2-amine —— C18H24N8
5-[(4S)-5-[(1-methylimidazol-2-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-propylpyrimidin-2-amine
—— (5-Acetyl-2-methoxyphenyl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate —— C18H20N2O6S
(5-Acetyl-2-methoxyphenyl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(3-phenylpropyl)morpholin-4-yl]methanone —— C22H26N4O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(3-phenylpropyl)morpholin-4-yl]methanone
—— 5-methoxy-2-[[(2S)-2-(trifluoromethyl)morpholin-4-yl]methyl]pyran-4-one —— C12H14F3NO4
5-methoxy-2-[[(2S)-2-(trifluoromethyl)morpholin-4-yl]methyl]pyran-4-one
—— 5-[(3R)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C24H27N3O2
5-[(3R)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate —— C18H17N3O5S
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate
—— 5-[6-amino-5-cyano-4-(2-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-1H-pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid —— C20H18N4O4
5-[6-amino-5-cyano-4-(2-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-1H-pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
—— 5-[[(2R)-2-(3,4-dichlorophenyl)morpholin-4-yl]methyl]-2-methoxyphenol —— C18H19Cl2NO3
5-[[(2R)-2-(3,4-dichlorophenyl)morpholin-4-yl]methyl]-2-methoxyphenol
—— (5S)-9-[(3,4-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H19F2NO2
(5S)-9-[(3,4-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-phenyl-1,3-oxazol-2-yl)methyl (3S)-1-(2-ethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H22N2O4
(5-phenyl-1,3-oxazol-2-yl)methyl (3S)-1-(2-ethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— [5-[[[(2S)-2-hydroxypropyl]-methylamino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone —— C15H22N4O2S
[5-[[[(2S)-2-hydroxypropyl]-methylamino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone
—— 5-[(3S)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C24H27N3O2
5-[(3S)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— (5-fluoropyridin-3-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H20F4N2O
(5-fluoropyridin-3-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-thiophen-2-ylacetate —— C13H10N2O3S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-thiophen-2-ylacetate
—— [5-[[[(2R)-2-hydroxypropyl]-methylamino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone —— C15H22N4O2S
[5-[[[(2R)-2-hydroxypropyl]-methylamino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone
—— (5-phenyl-1,3-oxazol-2-yl)methyl (3R)-1-(2-ethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H22N2O4
(5-phenyl-1,3-oxazol-2-yl)methyl (3R)-1-(2-ethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— 5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C20H26N4O3
5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-acetyl-6-methyl-3-[(3R)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C23H28N2O3
5-acetyl-6-methyl-3-[(3R)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
—— 5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C20H26N4O3
5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (5-fluoropyridin-3-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H20F4N2O
(5-fluoropyridin-3-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— [5-[[(3R)-3-(hydroxymethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone —— C18H26N4O2S
[5-[[(3R)-3-(hydroxymethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone
—— 5-[(4,5-dimethoxy-2-methylphenyl)methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C15H19N3O2S2
5-[(4,5-dimethoxy-2-methylphenyl)methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— [5-[[(3S)-3-(hydroxymethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone —— C18H26N4O2S
[5-[[(3S)-3-(hydroxymethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone
—— (5S)-2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O
(5S)-2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1S)-1-(2-chlorophenyl)ethyl]sulfanyl-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C13H14ClN3S2
5-[(1S)-1-(2-chlorophenyl)ethyl]sulfanyl-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— [(5R)-2,9-diazaspiro[4.5]decan-2-yl]-[2-(1,2,4-triazol-1-yl)phenyl]methanone —— C17H21N5O
[(5R)-2,9-diazaspiro[4.5]decan-2-yl]-[2-(1,2,4-triazol-1-yl)phenyl]methanone
—— [(5S)-2,9-diazaspiro[4.5]decan-2-yl]-[2-(1,2,4-triazol-1-yl)phenyl]methanone —— C17H21N5O
[(5S)-2,9-diazaspiro[4.5]decan-2-yl]-[2-(1,2,4-triazol-1-yl)phenyl]methanone
—— 5-[2-(4-methoxyphenyl)ethylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C14H17N3OS2
5-[2-(4-methoxyphenyl)ethylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— 5-[(2-bromophenyl)methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C12H12BrN3S2
5-[(2-bromophenyl)methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— 5-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C15H13FN4S3
5-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— 5-[[2-(2-chlorophenyl)-1,3-thiazol-4-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C15H13ClN4S3
5-[[2-(2-chlorophenyl)-1,3-thiazol-4-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— (5R)-N-[3-(3,5-dimethylpyrazol-1-yl)propyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H22N4O2
(5R)-N-[3-(3,5-dimethylpyrazol-1-yl)propyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide