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—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone —— C16H19ClN4O
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone
—— (5-fluoro-2-methoxyphenyl)methyl (E)-3-(4-nitrophenyl)prop-2-enoate —— C17H14FNO5
(5-fluoro-2-methoxyphenyl)methyl (E)-3-(4-nitrophenyl)prop-2-enoate
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone —— C16H19ClN4O
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone
—— [5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-nitrophenyl)prop-2-enoate —— C18H12ClN3O5
[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-nitrophenyl)prop-2-enoate
—— 5-chloro-6-[(3S)-3-[methyl(propan-2-yl)carbamoyl]piperidin-1-yl]pyridine-3-carboxamide —— C16H23ClN4O2
5-chloro-6-[(3S)-3-[methyl(propan-2-yl)carbamoyl]piperidin-1-yl]pyridine-3-carboxamide
—— 5,6-dimethyl-3-[(3R)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]pyridazine-4-carbonitrile —— C15H20N6O
5,6-dimethyl-3-[(3R)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]pyridazine-4-carbonitrile
—— 5-chloro-6-[(3R)-3-[methyl(propan-2-yl)carbamoyl]piperidin-1-yl]pyridine-3-carboxamide —— C16H23ClN4O2
5-chloro-6-[(3R)-3-[methyl(propan-2-yl)carbamoyl]piperidin-1-yl]pyridine-3-carboxamide
—— 5,6-dimethyl-3-[(3S)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]pyridazine-4-carbonitrile —— C15H20N6O
5,6-dimethyl-3-[(3S)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]pyridazine-4-carbonitrile
—— 5-ethyl-6-methyl-3-[[(2R)-oxolan-2-yl]methyl]-2-(4-oxopentylsulfanyl)thieno[2,3-d]pyrimidin-4-one —— C19H26N2O3S2
5-ethyl-6-methyl-3-[[(2R)-oxolan-2-yl]methyl]-2-(4-oxopentylsulfanyl)thieno[2,3-d]pyrimidin-4-one
—— 5-[[5-[(5R)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]pentan-2-one —— C18H25N3OS2
5-[[5-[(5R)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]pentan-2-one
—— (5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(furan-2-yl)prop-2-enoate —— C17H13NO4
(5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(furan-2-yl)prop-2-enoate
—— 5-ethyl-6-methyl-3-[[(2S)-oxolan-2-yl]methyl]-2-(4-oxopentylsulfanyl)thieno[2,3-d]pyrimidin-4-one —— C19H26N2O3S2
5-ethyl-6-methyl-3-[[(2S)-oxolan-2-yl]methyl]-2-(4-oxopentylsulfanyl)thieno[2,3-d]pyrimidin-4-one
—— [5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-nitrophenyl)prop-2-enoate —— C16H11N3O6
[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-nitrophenyl)prop-2-enoate
—— [5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate —— C14H10N2O5
[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate
—— 5-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1-[3-(trifluoromethyl)phenyl]pyrazolo[3,4-d]pyrimidin-4-one —— C20H20F3N5O3
5-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1-[3-(trifluoromethyl)phenyl]pyrazolo[3,4-d]pyrimidin-4-one
—— [5-(2-bromophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate —— C16H11BrN2O4
[5-(2-bromophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate
—— 5-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1-[3-(trifluoromethyl)phenyl]pyrazolo[3,4-d]pyrimidin-4-one —— C20H20F3N5O3
5-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1-[3-(trifluoromethyl)phenyl]pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1-[3-(trifluoromethyl)phenyl]pyrazolo[3,4-d]pyrimidin-4-one —— C20H20F3N5O3
5-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1-[3-(trifluoromethyl)phenyl]pyrazolo[3,4-d]pyrimidin-4-one
—— [5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate —— C19H18N2O7
[5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate
—— [5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate —— C16H11N3O6
[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(furan-2-yl)prop-2-enoate
—— 5-[3-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,6-dimethyl-2-oxo-1H-pyridine-3-carbonitrile —— C19H26N4O2
5-[3-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,6-dimethyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 3,4,5-triethoxybenzoate —— C23H25NO6
(5-Phenyl-1,3-oxazol-2-yl)methyl 3,4,5-triethoxybenzoate
—— 5-[3-[(9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,6-dimethyl-2-oxo-1H-pyridine-3-carbonitrile —— C19H26N4O2
5-[3-[(9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,6-dimethyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[3-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-3-oxopropyl]-6-methyl-1H-pyrimidine-2,4-dione —— C16H24N4O3
5-[3-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-3-oxopropyl]-6-methyl-1H-pyrimidine-2,4-dione
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-chloro-2-nitrobenzoate —— C16H9Cl2N3O5
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-chloro-2-nitrobenzoate
—— 5-[2-[(9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C16H22N6O2
5-[2-[(9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-[2-[(9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-2,6-dimethyl-1H-pyrimidin-4-one —— C16H24N4O2
5-[2-[(9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-2,6-dimethyl-1H-pyrimidin-4-one
—— 5-[2-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-2,6-dimethyl-1H-pyrimidin-4-one —— C16H24N4O2
5-[2-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-2,6-dimethyl-1H-pyrimidin-4-one
—— 5-[2-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C16H22N6O2
5-[2-[(9aS)-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-2-oxoethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3R)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C16H20ClN5O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3R)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3S)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C16H20ClN5O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3S)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone —— C16H19ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone —— C16H19ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone —— C16H19ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone
—— 5-[(2S)-3-[bis(4-fluorophenyl)methoxy]-2-hydroxypropyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C22H20F2N4O3
5-[(2S)-3-[bis(4-fluorophenyl)methoxy]-2-hydroxypropyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-chloro-N-[(5S)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]-2-propan-2-ylpyrimidine-4-carboxamide —— C17H19ClN4O2
5-chloro-N-[(5S)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]-2-propan-2-ylpyrimidine-4-carboxamide
—— 5-chloro-N-[(5R)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]-2-propan-2-ylpyrimidine-4-carboxamide —— C17H19ClN4O2
5-chloro-N-[(5R)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]-2-propan-2-ylpyrimidine-4-carboxamide
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone —— C16H19ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone
—— (5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate —— C21H19NO4
(5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate
—— 5-[(2R)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H15Cl2FN4O3
5-[(2R)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2R)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C24H24ClFN4O3
5-[(2R)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2R)-3-[bis(4-fluorophenyl)methoxy]-2-hydroxypropyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C22H20F2N4O3
5-[(2R)-3-[bis(4-fluorophenyl)methoxy]-2-hydroxypropyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2S)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H15Cl2FN4O3
5-[(2S)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2S)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C24H24ClFN4O3
5-[(2S)-3-(4-chloro-5-methyl-2-propan-2-ylphenoxy)-2-hydroxypropyl]-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— (5-acetyl-2-methoxyphenyl)methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate —— C21H22O5
(5-acetyl-2-methoxyphenyl)methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate
—— [5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate —— C20H17ClN2O4
[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate —— C20H18N2O4
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (E)-3-(2-ethoxyphenyl)prop-2-enoate
—— (5R)-5-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methylamino]-5,6,7,8-tetrahydro-1H-quinolin-2-one —— C17H17N3O2S
(5R)-5-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methylamino]-5,6,7,8-tetrahydro-1H-quinolin-2-one
—— (5S)-5-[(4-imidazol-1-ylphenyl)methylamino]-5,6,7,8-tetrahydro-1H-quinolin-2-one —— C19H20N4O
(5S)-5-[(4-imidazol-1-ylphenyl)methylamino]-5,6,7,8-tetrahydro-1H-quinolin-2-one
—— (5S)-5-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methylamino]-5,6,7,8-tetrahydro-1H-quinolin-2-one —— C17H17N3O2S
(5S)-5-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methylamino]-5,6,7,8-tetrahydro-1H-quinolin-2-one