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—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-phenylsulfanylpropanoate —— C16H14N2O3S2
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-phenylsulfanylpropanoate
—— [5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (2R)-2-phenylsulfanylpropanoate —— C16H14N2O4S
[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (2R)-2-phenylsulfanylpropanoate
—— (5S)-5-[2-(2-methyl-4-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-2-oxoethyl]pyrrolidin-2-one —— C18H25N5O2
(5S)-5-[2-(2-methyl-4-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-2-oxoethyl]pyrrolidin-2-one
—— 5-[(1R)-1-[2-(5-methylfuran-2-yl)imidazol-1-yl]ethyl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C17H15N5O2
5-[(1R)-1-[2-(5-methylfuran-2-yl)imidazol-1-yl]ethyl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(2S)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]methanone —— C21H23N3O4
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(2S)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]methanone
—— 5-[2-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C20H24FN3O2
5-[2-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— (5S)-9-[(6-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H22N2O2
(5S)-9-[(6-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(2R)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]methanone —— C21H23N3O4
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(2R)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]methanone
—— 5-[(1S)-1-[2-(5-methylfuran-2-yl)imidazol-1-yl]ethyl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C17H15N5O2
5-[(1S)-1-[2-(5-methylfuran-2-yl)imidazol-1-yl]ethyl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[2-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C20H24FN3O2
5-[2-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— [5-[[methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone —— C18H26N4O2S
[5-[[methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-piperidin-1-ylmethanone
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 1-ethylbenzotriazole-5-carboxylate —— C19H16N4O3
(5-Phenyl-1,3-oxazol-2-yl)methyl 1-ethylbenzotriazole-5-carboxylate
—— 5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H28F2N4
5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-3-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
—— [(5S)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]-(4-pyridin-4-ylpiperidin-1-yl)methanone —— C15H19N3O2
[(5S)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]-(4-pyridin-4-ylpiperidin-1-yl)methanone
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-3-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
—— 5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole —— C14H19N3O2
5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H28F2N4
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— 5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole —— C14H19N3O2
5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2-oxazole
—— (5-Acetyl-2-methoxyphenyl)methyl 2-(4,5-dihydro-1,3-thiazol-2-ylsulfanylmethyl)benzoate —— C21H21NO4S2
(5-Acetyl-2-methoxyphenyl)methyl 2-(4,5-dihydro-1,3-thiazol-2-ylsulfanylmethyl)benzoate
—— (5R)-9-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H23N3O2
(5R)-9-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H23N3O2
(5S)-9-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(3S)-1-(2-methyl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C20H23N7O
5-[(3S)-1-(2-methyl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— 5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine —— C20H25F2N3O
5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine
—— [5-[[(3R)-3-propylmorpholin-4-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone —— C18H26N4O2S
[5-[[(3R)-3-propylmorpholin-4-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine —— C20H25F2N3O
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine
—— 5-[[(2R)-2-(4-fluorophenyl)morpholin-4-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C14H15FN4O3
5-[[(2R)-2-(4-fluorophenyl)morpholin-4-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-[(3R)-1-(2-methyl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C20H23N7O
5-[(3R)-1-(2-methyl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— [5-[[(3S)-3-propylmorpholin-4-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone —— C18H26N4O2S
[5-[[(3S)-3-propylmorpholin-4-yl]methyl]imidazo[2,1-b][1,3]thiazol-6-yl]-pyrrolidin-1-ylmethanone
—— (5R)-9-[[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C21H26N2O4
(5R)-9-[[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[[2-[(4S)-2,2-dimethyloxan-4-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H24N4O2
5-[[2-[(4S)-2,2-dimethyloxan-4-yl]imidazol-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-(methoxymethyl)-N-methyl-N-[[(2R)-1-methylpiperidin-2-yl]methyl]-1,3,4-oxadiazole-2-carboxamide —— C13H22N4O3
5-(methoxymethyl)-N-methyl-N-[[(2R)-1-methylpiperidin-2-yl]methyl]-1,3,4-oxadiazole-2-carboxamide
—— 5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C15H15N5O2
5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— 5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C15H15N5O2
5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5S)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one —— C20H24N6O2
(5S)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one
—— (5R)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one —— C20H24N6O2
(5R)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one
—— (5-propyl-1H-pyrazol-4-yl)-[(2S)-2-(trifluoromethyl)morpholin-4-yl]methanone —— C12H16F3N3O2
(5-propyl-1H-pyrazol-4-yl)-[(2S)-2-(trifluoromethyl)morpholin-4-yl]methanone
—— 5-[(3S)-3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C22H25N3O3
5-[(3S)-3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-(4,5-dihydro-1,3-thiazol-2-ylsulfanylmethyl)benzoate —— C21H18N2O3S2
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-(4,5-dihydro-1,3-thiazol-2-ylsulfanylmethyl)benzoate
—— 5-[[(2S)-2-(4-fluorophenyl)morpholin-4-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C14H15FN4O3
5-[[(2S)-2-(4-fluorophenyl)morpholin-4-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5-Acetyl-2-methoxyphenyl)methyl 3-(phenylcarbamoylamino)propanoate —— C20H22N2O5
(5-Acetyl-2-methoxyphenyl)methyl 3-(phenylcarbamoylamino)propanoate
—— [5-[1-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]imidazol-2-yl]furan-2-yl]methanol —— C19H21N3O2
[5-[1-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]imidazol-2-yl]furan-2-yl]methanol
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 3-(phenylcarbamoylamino)propanoate —— C20H19N3O4
(5-Phenyl-1,3-oxazol-2-yl)methyl 3-(phenylcarbamoylamino)propanoate
—— (5-propyl-1H-pyrazol-4-yl)-[(2R)-2-(trifluoromethyl)morpholin-4-yl]methanone —— C12H16F3N3O2
(5-propyl-1H-pyrazol-4-yl)-[(2R)-2-(trifluoromethyl)morpholin-4-yl]methanone
—— (5S)-9-[[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C21H26N2O4
(5S)-9-[[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(3R)-3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C22H25N3O3
5-[(3R)-3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5-Fluoro-2-methoxyphenyl)methyl 2-(4,5-dihydro-1,3-thiazol-2-ylsulfanylmethyl)benzoate —— C19H18FNO3S2
(5-Fluoro-2-methoxyphenyl)methyl 2-(4,5-dihydro-1,3-thiazol-2-ylsulfanylmethyl)benzoate
—— [5-[[(4S)-4-(phenylmethoxymethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]furan-2-yl]methanol —— C20H23N3O3
[5-[[(4S)-4-(phenylmethoxymethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]furan-2-yl]methanol
—— 5-[[(2S)-2-benzylmorpholin-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H22N4O2
5-[[(2S)-2-benzylmorpholin-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[[(2R)-2-benzylmorpholin-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H22N4O2
5-[[(2R)-2-benzylmorpholin-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one