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—— (5-bromothiophen-3-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C13H14BrN3OS
(5-bromothiophen-3-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-methyl-1H-indazol-7-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C17H19N5O
(5-methyl-1H-indazol-7-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-bromothiophen-3-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C13H14BrN3OS
(5-bromothiophen-3-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— [5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C16H23N5O
[5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-methyl-1-benzofuran-2-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C18H19N3O2
(5-methyl-1-benzofuran-2-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— [5-(diethylaminomethyl)furan-2-yl]-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C18H26N4O2
[5-(diethylaminomethyl)furan-2-yl]-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-bromofuran-3-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C13H14BrN3O2
(5-bromofuran-3-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— [5-(diethylaminomethyl)furan-2-yl]-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C18H26N4O2
[5-(diethylaminomethyl)furan-2-yl]-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— 5-(4-methoxyphenyl)-1-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]pentan-1-one —— C20H27N3O2
5-(4-methoxyphenyl)-1-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]pentan-1-one
—— [5-methyl-1-(4-methylphenyl)pyrazol-4-yl]-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C20H23N5O
[5-methyl-1-(4-methylphenyl)pyrazol-4-yl]-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C17H21ClN4O2
(5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-methyl-1H-indazol-7-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C17H19N5O
(5-methyl-1H-indazol-7-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C16H20ClN5O
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C17H21ClN4O2
(5-chloro-6-propan-2-yloxypyridin-3-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-methyl-1H-pyrazol-3-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C13H17N5O
(5-methyl-1H-pyrazol-3-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— 5-(4-methoxyphenyl)-1-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]pentan-1-one —— C20H27N3O2
5-(4-methoxyphenyl)-1-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]pentan-1-one
—— 5-[(3S)-3-imidazol-1-ylpiperidine-1-carbonyl]-1H-pyridin-2-one —— C14H16N4O2
5-[(3S)-3-imidazol-1-ylpiperidine-1-carbonyl]-1H-pyridin-2-one
—— 5-[(3R)-3-imidazol-1-ylpiperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one —— C16H17N5O2
5-[(3R)-3-imidazol-1-ylpiperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one
—— 5-phenyl-2-[[(2S)-2-pyrazol-1-ylpropanoyl]amino]thiophene-3-carboxamide —— C17H16N4O2S
5-phenyl-2-[[(2S)-2-pyrazol-1-ylpropanoyl]amino]thiophene-3-carboxamide
—— 5-phenyl-2-[[(2R)-2-pyrazol-1-ylpropanoyl]amino]thiophene-3-carboxamide —— C17H16N4O2S
5-phenyl-2-[[(2R)-2-pyrazol-1-ylpropanoyl]amino]thiophene-3-carboxamide
—— (5-chloro-6-propan-2-yloxypyridin-3-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C17H21ClN4O2
(5-chloro-6-propan-2-yloxypyridin-3-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— 5-chloro-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[[(2R)-oxolan-2-yl]methoxy]aniline —— C16H20ClN3O3
5-chloro-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[[(2R)-oxolan-2-yl]methoxy]aniline
—— 5-chloro-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[[(2S)-oxolan-2-yl]methoxy]aniline —— C16H20ClN3O3
5-chloro-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[[(2S)-oxolan-2-yl]methoxy]aniline
—— 5-chloro-N-[(5R)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]furan-2-carboxamide —— C14H13ClN2O3
5-chloro-N-[(5R)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]furan-2-carboxamide
—— 5-chloro-N-[(5S)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]furan-2-carboxamide —— C14H13ClN2O3
5-chloro-N-[(5S)-2-oxo-5,6,7,8-tetrahydro-1H-quinolin-5-yl]furan-2-carboxamide
—— (5S)-2-[[(2-fluorophenyl)methyl-methylamino]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C16H19FN2O2S
(5S)-2-[[(2-fluorophenyl)methyl-methylamino]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— (5R)-2-[[(2-fluorophenyl)methyl-methylamino]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C16H19FN2O2S
(5R)-2-[[(2-fluorophenyl)methyl-methylamino]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— (5R)-5-phenyl-N-(2H-tetrazol-5-yl)-4,5-dihydro-1,2-oxazole-3-carboxamide —— C11H10N6O2
(5R)-5-phenyl-N-(2H-tetrazol-5-yl)-4,5-dihydro-1,2-oxazole-3-carboxamide
—— [5-chloro-2-(furan-2-ylmethylamino)pyrimidin-4-yl]-[(3S)-3-methylmorpholin-4-yl]methanone —— C15H17ClN4O3
[5-chloro-2-(furan-2-ylmethylamino)pyrimidin-4-yl]-[(3S)-3-methylmorpholin-4-yl]methanone
—— (5S)-5-phenyl-N-(2H-tetrazol-5-yl)-4,5-dihydro-1,2-oxazole-3-carboxamide —— C11H10N6O2
(5S)-5-phenyl-N-(2H-tetrazol-5-yl)-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5-(2-fluorophenyl)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]furan-2-carboxamide —— C16H16FNO4S
5-(2-fluorophenyl)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]furan-2-carboxamide
—— 5-[[(2S)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-ethyl-1,2,4-oxadiazole —— C17H23N3O3
5-[[(2S)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-ethyl-1,2,4-oxadiazole
—— 5-[[(2R)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C15H22N4O
5-[[(2R)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-(4-fluorophenyl)-N-[4-[[(2R)-1-methoxypropan-2-yl]sulfamoyl]phenyl]thiophene-2-carboxamide —— C21H21FN2O4S2
5-(4-fluorophenyl)-N-[4-[[(2R)-1-methoxypropan-2-yl]sulfamoyl]phenyl]thiophene-2-carboxamide
—— 5-(2-fluorophenyl)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]furan-2-carboxamide —— C16H16FNO4S
5-(2-fluorophenyl)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]furan-2-carboxamide
—— (5-phenyl-1,3-oxazol-2-yl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C18H18N2O4S
(5-phenyl-1,3-oxazol-2-yl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— 5-[[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C15H22N4O
5-[[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5-phenyl-1,3-oxazol-2-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C18H18N2O4S
(5-phenyl-1,3-oxazol-2-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (5-phenyl-1,3-oxazol-2-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C18H18N2O4S
(5-phenyl-1,3-oxazol-2-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— 5-[[(2R)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-ethyl-1,2,4-oxadiazole —— C17H23N3O3
5-[[(2R)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-ethyl-1,2,4-oxadiazole
—— 5-(4-chlorophenyl)-3-[[(2R)-oxolan-2-yl]methylsulfanyl]-1H-1,2,4-triazole —— C13H14ClN3OS
5-(4-chlorophenyl)-3-[[(2R)-oxolan-2-yl]methylsulfanyl]-1H-1,2,4-triazole
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C17H17N3O4S
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C15H15N3O4S2
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (5-acetyl-2-methoxyphenyl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C18H21NO5S
(5-acetyl-2-methoxyphenyl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (5R)-N-[(3R)-1,1-dioxothiolan-3-yl]-5-methyl-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H25NO3S2
(5R)-N-[(3R)-1,1-dioxothiolan-3-yl]-5-methyl-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C15H15N3O4S2
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (5S)-N-[(3R)-1,1-dioxothiolan-3-yl]-5-methyl-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H25NO3S2
(5S)-N-[(3R)-1,1-dioxothiolan-3-yl]-5-methyl-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-N-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5-methyl-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C22H24ClN3O2S
(5S)-N-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5-methyl-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-(2-chlorophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylfuran-2-carboxamide —— C17H18ClNO4S
5-(2-chlorophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylfuran-2-carboxamide
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C15H15N3O4S2
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate