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—— [5-[(E)-but-2-enyl]-1,3,4-oxadiazol-2-yl]-[(2R)-2-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]morpholin-4-yl]methanone —— C16H21N5O5
[5-[(E)-but-2-enyl]-1,3,4-oxadiazol-2-yl]-[(2R)-2-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]morpholin-4-yl]methanone
—— 5-[2-[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C20H23F2N3O2
5-[2-[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-2-phenyl-1,3-thiazole —— C17H17N3OS
5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-2-phenyl-1,3-thiazole
—— 5-[[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C21H30N4O
5-[[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— 5-[(2S)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C18H20FN3O3
5-[(2S)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(2R)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C18H20FN3O3
5-[(2R)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(1S)-1-[2-(3-ethoxy-4-methoxyphenyl)imidazol-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole —— C18H22N4O3
5-[(1S)-1-[2-(3-ethoxy-4-methoxyphenyl)imidazol-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole
—— 5-[[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C21H30N4O
5-[[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— (5R)-9-[(3-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H22N2O2
(5R)-9-[(3-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(1R)-1-[2-(3-ethoxy-4-methoxyphenyl)imidazol-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole —— C18H22N4O3
5-[(1R)-1-[2-(3-ethoxy-4-methoxyphenyl)imidazol-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole
—— (5S)-9-[(3-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H22N2O2
(5S)-9-[(3-methylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]-2-phenyl-1,3-thiazole —— C17H17N3OS
5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]-2-phenyl-1,3-thiazole
—— 5-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C18H20F3N3O2
5-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— (5-Methyl-1,3,4-oxadiazol-2-yl)methyl 5-(diethylsulfamoyl)-2-fluorobenzoate —— C15H18FN3O5S
(5-Methyl-1,3,4-oxadiazol-2-yl)methyl 5-(diethylsulfamoyl)-2-fluorobenzoate
—— (5-Fluoro-2-methoxyphenyl)methyl 5-(diethylsulfamoyl)-2-fluorobenzoate —— C19H21F2NO5S
(5-Fluoro-2-methoxyphenyl)methyl 5-(diethylsulfamoyl)-2-fluorobenzoate
—— (5S)-3-methyl-N-[[1-[(2-methylimidazol-1-yl)methyl]cyclopropyl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H20N4O2
(5S)-3-methyl-N-[[1-[(2-methylimidazol-1-yl)methyl]cyclopropyl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-methyl-N-[[1-[(2-methylimidazol-1-yl)methyl]cyclopropyl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H20N4O2
(5R)-3-methyl-N-[[1-[(2-methylimidazol-1-yl)methyl]cyclopropyl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5-Amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 1-oxidopyridin-1-ium-2-carboxylate —— C15H13N3O5S
(5-Amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 1-oxidopyridin-1-ium-2-carboxylate
—— 5-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyrazol-3-one —— C9H10F3N3O3
5-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyrazol-3-one
—— [5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl 1-oxidopyridin-1-ium-2-carboxylate —— C16H17N3O6S
[5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl 1-oxidopyridin-1-ium-2-carboxylate
—— (5-Acetyl-2-ethoxyphenyl)methyl 1-oxidopyridin-1-ium-2-carboxylate —— C17H17NO5
(5-Acetyl-2-ethoxyphenyl)methyl 1-oxidopyridin-1-ium-2-carboxylate
—— 5-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyrazol-3-one —— C9H10F3N3O3
5-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyrazol-3-one
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide —— C13H19N5O2S2
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide
—— 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide —— C13H19N5O2S2
5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide
—— 5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C20H25FN4O2
5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide —— C13H19N5O2S2
5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(2S)-2-(trifluoromethyl)morpholin-4-yl]methanone —— C15H13ClF3NO4
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(2S)-2-(trifluoromethyl)morpholin-4-yl]methanone
—— [5-[1-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazol-2-yl]furan-2-yl]methanol —— C19H22N4O3
[5-[1-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazol-2-yl]furan-2-yl]methanol
—— (5-propyl-1,3,4-oxadiazol-2-yl)-[(2S)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methanone —— C16H26N4O3
(5-propyl-1,3,4-oxadiazol-2-yl)-[(2S)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methanone
—— 5-[[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C19H24FN5O3
5-[[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(2R)-2-(trifluoromethyl)morpholin-4-yl]methanone —— C15H13ClF3NO4
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(2R)-2-(trifluoromethyl)morpholin-4-yl]methanone
—— [5-[1-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazol-2-yl]furan-2-yl]methanol —— C19H22N4O3
[5-[1-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazol-2-yl]furan-2-yl]methanol
—— 5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C20H25FN4O2
5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— (5-propyl-1,3,4-oxadiazol-2-yl)-[(2R)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methanone —— C16H26N4O3
(5-propyl-1,3,4-oxadiazol-2-yl)-[(2R)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methanone
—— 5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-4-hydroxy-1H-pyridin-2-one —— C18H27N3O3
5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-4-hydroxy-1H-pyridin-2-one
—— (5S)-9-[(3,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H19F2NO2
(5S)-9-[(3,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-methyl-3-[4-[2-[(1R)-1-phenylethyl]imidazol-1-yl]phenyl]-1H-1,2,4-triazole —— C20H19N5
5-methyl-3-[4-[2-[(1R)-1-phenylethyl]imidazol-1-yl]phenyl]-1H-1,2,4-triazole
—— (5R)-9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H26N2O3
(5R)-9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-chloro-N-[(2R)-1-imidazol-1-ylbutan-2-yl]pyridine-2-carboxamide —— C13H15ClN4O
5-chloro-N-[(2R)-1-imidazol-1-ylbutan-2-yl]pyridine-2-carboxamide
—— 5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-4-hydroxy-1H-pyridin-2-one —— C18H27N3O3
5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-4-hydroxy-1H-pyridin-2-one
—— (5R)-9-[(3,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H19F2NO2
(5R)-9-[(3,5-difluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-methoxy-2-[[(3R)-3-(4-methylsulfanylbenzoyl)piperidin-1-yl]methyl]-1H-pyridin-4-one —— C20H24N2O3S
5-methoxy-2-[[(3R)-3-(4-methylsulfanylbenzoyl)piperidin-1-yl]methyl]-1H-pyridin-4-one
—— 5-methyl-3-[4-[2-[(1S)-1-phenylethyl]imidazol-1-yl]phenyl]-1H-1,2,4-triazole —— C20H19N5
5-methyl-3-[4-[2-[(1S)-1-phenylethyl]imidazol-1-yl]phenyl]-1H-1,2,4-triazole
—— 5-chloro-N-[(2S)-1-imidazol-1-ylbutan-2-yl]pyridine-2-carboxamide —— C13H15ClN4O
5-chloro-N-[(2S)-1-imidazol-1-ylbutan-2-yl]pyridine-2-carboxamide
—— 5-methoxy-2-[[(3S)-3-(4-methylsulfanylbenzoyl)piperidin-1-yl]methyl]-1H-pyridin-4-one —— C20H24N2O3S
5-methoxy-2-[[(3S)-3-(4-methylsulfanylbenzoyl)piperidin-1-yl]methyl]-1H-pyridin-4-one
—— 5-[[(2R)-2-(4-chlorophenyl)morpholin-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H19ClN4O2
5-[[(2R)-2-(4-chlorophenyl)morpholin-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[[(3S)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methylfuran-2-carboxamide —— C19H29N3O3
5-[[(3S)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methylfuran-2-carboxamide
—— 5-[(4R)-5-(1H-benzimidazol-2-ylmethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-ethylpyrimidin-2-amine —— C20H22N8
5-[(4R)-5-(1H-benzimidazol-2-ylmethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-ethylpyrimidin-2-amine
—— (5R)-9-[(4-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H20FNO2
(5R)-9-[(4-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one