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—— (5R)-N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-ethyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H20ClN5O2
(5R)-N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-ethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-9-[(4-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H20FNO2
(5S)-9-[(4-fluorophenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-chloropyridin-2-yl)-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C18H26ClN3O
(5-chloropyridin-2-yl)-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— (5-chloropyridin-2-yl)-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C18H26ClN3O
(5-chloropyridin-2-yl)-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— 5-[[(3R)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methylfuran-2-carboxamide —— C19H29N3O3
5-[[(3R)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methylfuran-2-carboxamide
—— 5-[[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine —— C20H26F2N4
5-[[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine
—— [5-[1-[(2R)-1-indol-1-ylpropan-2-yl]imidazol-2-yl]furan-2-yl]methanol —— C19H19N3O2
[5-[1-[(2R)-1-indol-1-ylpropan-2-yl]imidazol-2-yl]furan-2-yl]methanol
—— 5-[(2R)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C16H23N3O2
5-[(2R)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— [5-[1-[(2S)-1-indol-1-ylpropan-2-yl]imidazol-2-yl]furan-2-yl]methanol —— C19H19N3O2
[5-[1-[(2S)-1-indol-1-ylpropan-2-yl]imidazol-2-yl]furan-2-yl]methanol
—— 5-[(4S)-5-(1H-benzimidazol-2-ylmethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-ethylpyrimidin-2-amine —— C20H22N8
5-[(4S)-5-(1H-benzimidazol-2-ylmethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-N-ethylpyrimidin-2-amine
—— 5-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C19H21FN2O2
5-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (5S)-3-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-ethyl-5-(4-methoxyphenyl)imidazolidine-2,4-dione —— C21H29N3O4
(5S)-3-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-ethyl-5-(4-methoxyphenyl)imidazolidine-2,4-dione
—— 5-[(2S)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C16H23N3O2
5-[(2S)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— (5S)-N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-ethyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H20ClN5O2
(5S)-N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-ethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(1S)-1-(2-chlorophenyl)ethyl]sulfanyl-1-(3-fluorophenyl)tetrazole —— C15H12ClFN4S
5-[(1S)-1-(2-chlorophenyl)ethyl]sulfanyl-1-(3-fluorophenyl)tetrazole
—— 5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C20H32N4O2
5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(4-Chlorophenyl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole —— C14H10ClFN4S
5-[(4-Chlorophenyl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole
—— 5-(1,3-Benzodioxol-5-ylmethylsulfanyl)-1-(3-fluorophenyl)tetrazole —— C15H11FN4O2S
5-(1,3-Benzodioxol-5-ylmethylsulfanyl)-1-(3-fluorophenyl)tetrazole
—— (5R)-5-(1-adamantyl)-3-ethyl-2-sulfanylideneimidazolidin-4-one —— C15H22N2OS
(5R)-5-(1-adamantyl)-3-ethyl-2-sulfanylideneimidazolidin-4-one
—— 5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C20H32N4O2
5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(6-chloro-4H-1,3-benzodioxin-8-yl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole —— C16H12ClFN4O2S
5-[(6-chloro-4H-1,3-benzodioxin-8-yl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole
—— 5-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C19H21FN2O2
5-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5-[(2-Bromophenyl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole —— C14H10BrFN4S
5-[(2-Bromophenyl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole
—— 5-[[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C20H25FN4O3
5-[[(3R)-4-[(4-fluorophenyl)methyl]-5-oxo-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— 5-[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C21H21F2N3O2
5-[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[[(2R)-2-[(2-chlorophenyl)methyl]morpholin-4-yl]methyl]-2-hydroxybenzoic acid —— C19H20ClNO4
5-[[(2R)-2-[(2-chlorophenyl)methyl]morpholin-4-yl]methyl]-2-hydroxybenzoic acid
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-ethylsulfinylbenzoate —— C16H14N2O4S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-ethylsulfinylbenzoate
—— 5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H23N5O3
5-[[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5R)-9-[[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C20H23FN2O3
(5R)-9-[[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— [5-[(E)-but-2-enyl]-1,3,4-oxadiazol-2-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone —— C17H20N4O2
[5-[(E)-but-2-enyl]-1,3,4-oxadiazol-2-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone
—— 5-[[(2S)-2-[(2-chlorophenyl)methyl]morpholin-4-yl]methyl]-2-hydroxybenzoic acid —— C19H20ClNO4
5-[[(2S)-2-[(2-chlorophenyl)methyl]morpholin-4-yl]methyl]-2-hydroxybenzoic acid
—— 5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C17H26N4O2
5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— (5R)-5-(2,5-difluorophenyl)-5-methyl-3-(2-oxo-2-pyrrolidin-1-ylethyl)imidazolidine-2,4-dione —— C16H17F2N3O3
(5R)-5-(2,5-difluorophenyl)-5-methyl-3-(2-oxo-2-pyrrolidin-1-ylethyl)imidazolidine-2,4-dione
—— 5-(imidazol-1-ylmethyl)-N-methyl-N-[(1R)-1-pyridin-3-ylethyl]furan-2-carboxamide —— C17H18N4O2
5-(imidazol-1-ylmethyl)-N-methyl-N-[(1R)-1-pyridin-3-ylethyl]furan-2-carboxamide
—— (5E)-2-phenyl-5-[(Z)-3-phenylprop-2-enylidene]-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one —— C27H27N3O
(5E)-2-phenyl-5-[(Z)-3-phenylprop-2-enylidene]-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one
—— [5-[(E)-but-2-enyl]-1,3,4-oxadiazol-2-yl]-[(3S)-3-phenylpiperazin-1-yl]methanone —— C17H20N4O2
[5-[(E)-but-2-enyl]-1,3,4-oxadiazol-2-yl]-[(3S)-3-phenylpiperazin-1-yl]methanone
—— (5S)-9-[[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C20H23FN2O3
(5S)-9-[[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(2-methoxyphenoxy)methyl]-N-[(3S)-1-methyl-2-oxopyrrolidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H20N4O4
5-[(2-methoxyphenoxy)methyl]-N-[(3S)-1-methyl-2-oxopyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C21H21F2N3O2
5-[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5R)-5-(2,5-difluorophenyl)-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-methylimidazolidine-2,4-dione —— C18H21F2N3O4
(5R)-5-(2,5-difluorophenyl)-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-methylimidazolidine-2,4-dione
—— 5-[(1S)-1-[2-(2-butyl-5-chloro-1H-imidazol-4-yl)imidazol-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole —— C16H21ClN6O
5-[(1S)-1-[2-(2-butyl-5-chloro-1H-imidazol-4-yl)imidazol-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-ethyl-5-methylthiophene-2-carboxylate —— C17H15N3O5S
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-ethyl-5-methylthiophene-2-carboxylate
—— 5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C17H26N4O2
5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— 5-[[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine —— C20H26FN3O
5-[[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine
—— 5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine —— C20H26FN3O
5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine
—— 5-methoxy-2-[(2S)-2-(2-phenylethyl)morpholine-4-carbonyl]-1H-pyridin-4-one —— C19H22N2O4
5-methoxy-2-[(2S)-2-(2-phenylethyl)morpholine-4-carbonyl]-1H-pyridin-4-one
—— 5-[(2-methoxyphenoxy)methyl]-N-[(3R)-1-methyl-2-oxopyrrolidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H20N4O4
5-[(2-methoxyphenoxy)methyl]-N-[(3R)-1-methyl-2-oxopyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-methyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-3-carboxamide —— C11H18N4O4S
5-methyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-3-carboxamide
—— 5-methyl-N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-3-carboxamide —— C11H18N4O4S
5-methyl-N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-3-carboxamide