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—— 5-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole —— C17H21N5OS
5-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole
—— 5-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]pentanenitrile —— C14H22N4
5-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]pentanenitrile
—— 5-[(1R)-1-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C17H21N5OS
5-[(1R)-1-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-chloro-6-[[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pyridine-3-carbonitrile —— C13H13ClN6
5-chloro-6-[[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pyridine-3-carbonitrile
—— 5-chloro-6-[[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pyridine-3-carbonitrile —— C13H13ClN6
5-chloro-6-[[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pyridine-3-carbonitrile
—— 5,6-dimethyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine —— C15H18N6S
5,6-dimethyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine
—— 5-tert-butyl-2-[[(2R)-2-(4-methoxyphenyl)azepan-1-yl]methyl]-1,3-oxazole —— C21H30N2O2
5-tert-butyl-2-[[(2R)-2-(4-methoxyphenyl)azepan-1-yl]methyl]-1,3-oxazole
—— 5-fluoro-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]quinazolin-4-amine —— C15H15FN6
5-fluoro-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]quinazolin-4-amine
—— 5,6-dimethyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine —— C15H18N6S
5,6-dimethyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine
—— (5-cyclohexyl-1H-pyrazol-4-yl)-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone —— C19H27N5O
(5-cyclohexyl-1H-pyrazol-4-yl)-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone
—— (5S)-5-methyl-1-phenyl-3-[4-[(E)-3-phenylprop-2-enyl]piperazine-1-carbonyl]-2,5-dihydro-1,2,4-triazin-6-one —— C24H27N5O2
(5S)-5-methyl-1-phenyl-3-[4-[(E)-3-phenylprop-2-enyl]piperazine-1-carbonyl]-2,5-dihydro-1,2,4-triazin-6-one
—— (5R)-5-methyl-1-phenyl-3-[4-[(E)-3-phenylprop-2-enyl]piperazine-1-carbonyl]-2,5-dihydro-1,2,4-triazin-6-one —— C24H27N5O2
(5R)-5-methyl-1-phenyl-3-[4-[(E)-3-phenylprop-2-enyl]piperazine-1-carbonyl]-2,5-dihydro-1,2,4-triazin-6-one
—— 5-(azepan-1-ylsulfonyl)-N-[(2R)-butan-2-yl]-N-butyl-2-methoxybenzamide —— C22H36N2O4S
5-(azepan-1-ylsulfonyl)-N-[(2R)-butan-2-yl]-N-butyl-2-methoxybenzamide
—— 5-[[5-(4-Fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-phenyl-1,2,4-oxadiazole —— C20H16FN5OS
5-[[5-(4-Fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-(4-fluorophenyl)-N-[4-[[(2R)-oxolane-2-carbonyl]amino]phenyl]furan-2-carboxamide —— C22H19FN2O4
5-(4-fluorophenyl)-N-[4-[[(2R)-oxolane-2-carbonyl]amino]phenyl]furan-2-carboxamide
—— 5-(4-fluorophenyl)-N-[4-[[(2S)-oxolane-2-carbonyl]amino]phenyl]furan-2-carboxamide —— C22H19FN2O4
5-(4-fluorophenyl)-N-[4-[[(2S)-oxolane-2-carbonyl]amino]phenyl]furan-2-carboxamide
—— 5-[(4-Morpholin-4-yl-3-nitrophenyl)sulfonylamino]benzene-1,3-dicarboxylate —— C18H15N3O9S-2
5-[(4-Morpholin-4-yl-3-nitrophenyl)sulfonylamino]benzene-1,3-dicarboxylate
—— 5-(4-fluorophenyl)-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C20H20FN3O2S
5-(4-fluorophenyl)-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— [5-(4-fluorophenyl)-1H-pyrazol-4-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H18FN5O
[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-[[4-[(3R)-3-methylpiperidin-1-yl]sulfonylpiperazin-1-yl]methyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C20H26F3N5O3S
5-[[4-[(3R)-3-methylpiperidin-1-yl]sulfonylpiperazin-1-yl]methyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— (5-phenyl-1H-pyrazol-4-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H19N5O
(5-phenyl-1H-pyrazol-4-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— [5-(4-fluorophenyl)-1H-pyrazol-4-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H18FN5O
[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5,6-dimethyl-2-[(1S)-1-[2-(4-methylpyrazol-1-yl)ethylamino]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C16H21N5OS
5,6-dimethyl-2-[(1S)-1-[2-(4-methylpyrazol-1-yl)ethylamino]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5-phenyl-1H-pyrazol-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H19N5O
(5-phenyl-1H-pyrazol-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5,6-dimethyl-2-[(1R)-1-[2-(4-methylpyrazol-1-yl)ethylamino]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C16H21N5OS
5,6-dimethyl-2-[(1R)-1-[2-(4-methylpyrazol-1-yl)ethylamino]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5-cyclohexyl-1H-pyrazol-4-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C19H27N5O
(5-cyclohexyl-1H-pyrazol-4-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5-cyclohexyl-1H-pyrazol-4-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C19H27N5O
(5-cyclohexyl-1H-pyrazol-4-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— 5-(4-fluorophenyl)-3-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C20H20FN3O2S
5-(4-fluorophenyl)-3-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— [5-(4-fluorophenyl)-1-methylpyrrol-2-yl]-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C19H24FN3O2
[5-(4-fluorophenyl)-1-methylpyrrol-2-yl]-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-(4-Methylphenyl)-3-[(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl]thieno[2,3-d]pyrimidin-4-one —— C20H14N4O2S2
5-(4-Methylphenyl)-3-[(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl]thieno[2,3-d]pyrimidin-4-one
—— (5-fluoro-3-methyl-1-benzothiophen-2-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C17H21FN2O2S
(5-fluoro-3-methyl-1-benzothiophen-2-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-(4-fluorophenyl)-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C20H20FN3O2S
5-(4-fluorophenyl)-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— [5-(4-fluorophenyl)-1-methylpyrrol-2-yl]-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C19H24FN3O2
[5-(4-fluorophenyl)-1-methylpyrrol-2-yl]-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-(4-methylphenyl)-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C21H23N3O2S
5-(4-methylphenyl)-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 5-[4-[(2S)-2-hydroxypropyl]piperazine-1-carbonyl]-N-methylpyridine-2-carboxamide —— C15H22N4O3
5-[4-[(2S)-2-hydroxypropyl]piperazine-1-carbonyl]-N-methylpyridine-2-carboxamide
—— 5-(4-fluorophenyl)-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C20H20FN3O2S
5-(4-fluorophenyl)-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 5-[4-[(2R)-2-hydroxypropyl]piperazine-1-carbonyl]-N-methylpyridine-2-carboxamide —— C15H22N4O3
5-[4-[(2R)-2-hydroxypropyl]piperazine-1-carbonyl]-N-methylpyridine-2-carboxamide
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C15H23ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-[4-[(2S)-2-hydroxypropyl]piperazine-1-carbonyl]-4-methylthiophene-2-sulfonamide —— C13H21N3O4S2
5-[4-[(2S)-2-hydroxypropyl]piperazine-1-carbonyl]-4-methylthiophene-2-sulfonamide
—— (5-chloro-2-propan-2-yloxyphenyl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C17H25ClN2O3
(5-chloro-2-propan-2-yloxyphenyl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— (5-chloro-2-propan-2-yloxyphenyl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C17H25ClN2O3
(5-chloro-2-propan-2-yloxyphenyl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C15H23ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— (5-fluoro-3-methyl-1-benzothiophen-2-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C17H21FN2O2S
(5-fluoro-3-methyl-1-benzothiophen-2-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— (5-ethylfuran-2-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C14H22N2O3
(5-ethylfuran-2-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-[4-[(2R)-2-hydroxypropyl]piperazine-1-carbonyl]-4-methylthiophene-2-sulfonamide —— C13H21N3O4S2
5-[4-[(2R)-2-hydroxypropyl]piperazine-1-carbonyl]-4-methylthiophene-2-sulfonamide
—— 5,7-Dichloro-2-methyl-8-[2-(4-methylphenoxy)ethoxy]quinoline —— C19H17Cl2NO2
5,7-Dichloro-2-methyl-8-[2-(4-methylphenoxy)ethoxy]quinoline
—— 5,7-Dichloro-2-methyl-8-[(2-methylphenyl)methoxy]quinoline —— C18H15Cl2NO
5,7-Dichloro-2-methyl-8-[(2-methylphenyl)methoxy]quinoline
—— 5,7-Dichloro-8-[(2,5-dimethylphenyl)methoxy]-2-methylquinoline —— C19H17Cl2NO
5,7-Dichloro-8-[(2,5-dimethylphenyl)methoxy]-2-methylquinoline
—— (5-ethyl-1-pyridin-2-ylpyrazol-4-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C18H25N5O2
(5-ethyl-1-pyridin-2-ylpyrazol-4-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-[2-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]-2-oxoethyl]thiophene-2-sulfonamide —— C13H21N3O4S2
5-[2-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]-2-oxoethyl]thiophene-2-sulfonamide