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—— (5E)-5-[(4-chlorophenyl)methylidene]-2-phenyl-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one —— C25H24ClN3O
(5E)-5-[(4-chlorophenyl)methylidene]-2-phenyl-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one
—— (5R)-1-(2-methylpropyl)-5-(3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)piperidin-2-one —— C15H23N5OS
(5R)-1-(2-methylpropyl)-5-(3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)piperidin-2-one
—— 5-(imidazol-1-ylmethyl)-N-methyl-N-[(1S)-1-pyridin-3-ylethyl]furan-2-carboxamide —— C17H18N4O2
5-(imidazol-1-ylmethyl)-N-methyl-N-[(1S)-1-pyridin-3-ylethyl]furan-2-carboxamide
—— 5-[[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C17H29N5O2
5-[[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-ethyl-5-methylthiophene-2-carboxylate —— C15H14N2O4S
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-ethyl-5-methylthiophene-2-carboxylate
—— (5E)-5-[[4-(dimethylamino)phenyl]methylidene]-2-phenyl-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one —— C27H30N4O
(5E)-5-[[4-(dimethylamino)phenyl]methylidene]-2-phenyl-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one
—— 5-[[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C17H29N5O2
5-[[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— [5-(hydroxymethyl)furan-2-yl]-[(2S)-2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl]methanone —— C19H23NO4
[5-(hydroxymethyl)furan-2-yl]-[(2S)-2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl]methanone
—— [5-(hydroxymethyl)furan-2-yl]-[(2R)-2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl]methanone —— C19H23NO4
[5-(hydroxymethyl)furan-2-yl]-[(2R)-2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl]methanone
—— 5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H23N5O3
5-[[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-methyl-2-[[2-[5-[(2S)-oxan-2-yl]furan-2-yl]imidazol-1-yl]methyl]imidazo[1,2-a]pyridine —— C21H22N4O2
5-methyl-2-[[2-[5-[(2S)-oxan-2-yl]furan-2-yl]imidazol-1-yl]methyl]imidazo[1,2-a]pyridine
—— 5-methyl-2-[[2-[5-[(2R)-oxan-2-yl]furan-2-yl]imidazol-1-yl]methyl]imidazo[1,2-a]pyridine —— C21H22N4O2
5-methyl-2-[[2-[5-[(2R)-oxan-2-yl]furan-2-yl]imidazol-1-yl]methyl]imidazo[1,2-a]pyridine
—— (5S)-1-(2-methylpropyl)-5-(3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)piperidin-2-one —— C15H23N5OS
(5S)-1-(2-methylpropyl)-5-(3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)piperidin-2-one
—— 5-methoxy-2-[(2R)-2-(2-phenylethyl)morpholine-4-carbonyl]-1H-pyridin-4-one —— C19H22N2O4
5-methoxy-2-[(2R)-2-(2-phenylethyl)morpholine-4-carbonyl]-1H-pyridin-4-one
—— 5-[(1S)-1-[2-(2,3-difluoro-6-methoxyphenyl)imidazol-1-yl]ethyl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C19H15F2N5O2
5-[(1S)-1-[2-(2,3-difluoro-6-methoxyphenyl)imidazol-1-yl]ethyl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5S)-9-[(4-methylnaphthalen-1-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C21H25NO2
(5S)-9-[(4-methylnaphthalen-1-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-ethyl-1H-pyrazol-3-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H24F3N3O
(5-ethyl-1H-pyrazol-3-yl)-[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (5E)-5-[(2-chlorophenyl)methylidene]-2-phenyl-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one —— C25H24ClN3O
(5E)-5-[(2-chlorophenyl)methylidene]-2-phenyl-3-[(Z)-(3,5,5-trimethylcyclohex-3-en-1-ylidene)amino]imidazol-4-one
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 4-ethyl-5-methylthiophene-2-carboxylate —— C17H16N2O3S
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 4-ethyl-5-methylthiophene-2-carboxylate
—— 5-[[(3R)-3-(dimethylamino)pyrrolidin-1-yl]methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide —— C22H29N5OS
5-[[(3R)-3-(dimethylamino)pyrrolidin-1-yl]methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
—— (5-ethyl-1H-pyrazol-3-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H24F3N3O
(5-ethyl-1H-pyrazol-3-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (5-chloro-2-methoxyphenyl)-[(3R)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-3-yl]methanone —— C19H22ClN3O3
(5-chloro-2-methoxyphenyl)-[(3R)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-3-yl]methanone
—— 5-[(dimethylamino)methyl]-N-[(3R)-3-hydroxy-3-phenylpropyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide —— C16H22N4O3
5-[(dimethylamino)methyl]-N-[(3R)-3-hydroxy-3-phenylpropyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
—— (5R)-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H23N3O2
(5R)-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-chloro-2-methoxyphenyl)-[(3S)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-3-yl]methanone —— C19H22ClN3O3
(5-chloro-2-methoxyphenyl)-[(3S)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-3-yl]methanone
—— (5R)-9-[(4-methylnaphthalen-1-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C21H25NO2
(5R)-9-[(4-methylnaphthalen-1-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-hydroxypyridin-2-yl)-[(3R)-3-[2-[3-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H21F3N2O2
(5-hydroxypyridin-2-yl)-[(3R)-3-[2-[3-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (5S)-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H23N3O2
(5S)-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(1S)-1-[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole —— C21H17N7O
5-[(1S)-1-[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole
—— 5-acetyl-3-[(2S)-2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl]-6-methyl-1H-pyridin-2-one —— C20H21ClN2O4
5-acetyl-3-[(2S)-2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl]-6-methyl-1H-pyridin-2-one
—— 5-acetyl-3-[(2R)-2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl]-6-methyl-1H-pyridin-2-one —— C20H21ClN2O4
5-acetyl-3-[(2R)-2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl]-6-methyl-1H-pyridin-2-one
—— (5-methyl-1H-indazol-3-yl)-[(2S)-2-(4-methylpentyl)morpholin-4-yl]methanone —— C19H27N3O2
(5-methyl-1H-indazol-3-yl)-[(2S)-2-(4-methylpentyl)morpholin-4-yl]methanone
—— (5-Thiophen-2-yl-1,3,4-oxadiazol-2-yl)methyl 4-oxo-4-thiophen-2-ylbutanoate —— C15H12N2O4S2
(5-Thiophen-2-yl-1,3,4-oxadiazol-2-yl)methyl 4-oxo-4-thiophen-2-ylbutanoate
—— 5-[2-[(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione —— C15H21N3O3
5-[2-[(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione
—— 5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H29FN4
5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— 5-[(2-methoxyphenoxy)methyl]-N-[(2R)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide —— C16H20N4O4
5-[(2-methoxyphenoxy)methyl]-N-[(2R)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide
—— 5-[(1R)-1-[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole —— C21H17N7O
5-[(1R)-1-[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole
—— 5-[(2-methoxyphenoxy)methyl]-N-[(2S)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide —— C16H20N4O4
5-[(2-methoxyphenoxy)methyl]-N-[(2S)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide
—— (5-methyl-1H-pyrazol-3-yl)-[(3R)-3-phenylpiperidin-1-yl]methanone —— C16H19N3O
(5-methyl-1H-pyrazol-3-yl)-[(3R)-3-phenylpiperidin-1-yl]methanone
—— 5-[2-[(3R)-3-aminopyrrolidin-1-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid —— C17H20N4O3
5-[2-[(3R)-3-aminopyrrolidin-1-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid
—— (5-methyl-1H-pyrazol-3-yl)-[(3S)-3-phenylpiperidin-1-yl]methanone —— C16H19N3O
(5-methyl-1H-pyrazol-3-yl)-[(3S)-3-phenylpiperidin-1-yl]methanone
—— (5S)-1-[4-(benzylsulfamoylamino)phenyl]-5-methylpyrrolidin-2-one —— C18H21N3O3S
(5S)-1-[4-(benzylsulfamoylamino)phenyl]-5-methylpyrrolidin-2-one
—— 5-[2-[(3S)-3-aminopyrrolidin-1-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid —— C17H20N4O3
5-[2-[(3S)-3-aminopyrrolidin-1-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid
—— 5-[(2S)-2-benzylmorpholine-4-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C19H19N3O3
5-[(2S)-2-benzylmorpholine-4-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[[(2R)-2-[(3-fluorophenyl)methyl]morpholin-4-yl]methyl]-N-propylpyrimidin-2-amine —— C19H25FN4O
5-[[(2R)-2-[(3-fluorophenyl)methyl]morpholin-4-yl]methyl]-N-propylpyrimidin-2-amine
—— 5-[2-[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C20H24FN3O2
5-[2-[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[(2R)-2-benzylmorpholine-4-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C19H19N3O3
5-[(2R)-2-benzylmorpholine-4-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-oxo-4-thiophen-2-ylbutanoate —— C17H13ClN2O4S
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-oxo-4-thiophen-2-ylbutanoate
—— 5-[(2S)-2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C16H15Cl2N3O3
5-[(2S)-2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[(2R)-2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C16H15Cl2N3O3
5-[(2R)-2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methyl-1H-pyrimidin-6-one