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—— 5-methyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide —— C17H22N2O3S
5-methyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-[[(2S)-2-methylpiperidin-1-yl]methyl]phenyl]pentanamide —— C23H34N4O2S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-[[(2S)-2-methylpiperidin-1-yl]methyl]phenyl]pentanamide
—— 5-methyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide —— C17H22N2O3S
5-methyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-[[(2R)-2-methylpiperidin-1-yl]methyl]phenyl]pentanamide —— C23H34N4O2S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-[[(2R)-2-methylpiperidin-1-yl]methyl]phenyl]pentanamide
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-nitrobenzoate —— C16H10ClN3O5
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-nitrobenzoate
—— (5-ethyl-4-methylthiophen-2-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C18H21NOS2
(5-ethyl-4-methylthiophen-2-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (5-Amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 1-oxidopyridin-1-ium-4-carboxylate —— C15H13N3O5S
(5-Amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 1-oxidopyridin-1-ium-4-carboxylate
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 1-oxidopyridin-1-ium-4-carboxylate —— C15H10N4O6
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 1-oxidopyridin-1-ium-4-carboxylate
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 1-oxidopyridin-1-ium-4-carboxylate —— C15H11N3O4
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 1-oxidopyridin-1-ium-4-carboxylate
—— 5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]pyridin-1-ium-2-amine —— C22H30N3O3S+
5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]pyridin-1-ium-2-amine
—— (5-ethyl-4-methylthiophen-2-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C18H21NOS2
(5-ethyl-4-methylthiophen-2-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 5-(furan-2-yl)-3-[2-[(3S)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-1,3,4-oxadiazol-2-one —— C24H20N4O5
5-(furan-2-yl)-3-[2-[(3S)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-1,3,4-oxadiazol-2-one
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-phenoxypropanoate —— C16H14N2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-phenoxypropanoate
—— 5-[(2S)-1-(2,4-difluorophenyl)-1-oxopropan-2-yl]sulfanyl-3-methyl-7-propan-2-yl-1-propylpyrimido[4,5-d]pyrimidine-2,4-dione —— C22H24F2N4O3S
5-[(2S)-1-(2,4-difluorophenyl)-1-oxopropan-2-yl]sulfanyl-3-methyl-7-propan-2-yl-1-propylpyrimido[4,5-d]pyrimidine-2,4-dione
—— 5-(4-methylphenyl)-4-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine —— C21H21N5S
5-(4-methylphenyl)-4-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine
—— 5-[(2R)-1-(2,4-difluorophenyl)-1-oxopropan-2-yl]sulfanyl-3-methyl-7-propan-2-yl-1-propylpyrimido[4,5-d]pyrimidine-2,4-dione —— C22H24F2N4O3S
5-[(2R)-1-(2,4-difluorophenyl)-1-oxopropan-2-yl]sulfanyl-3-methyl-7-propan-2-yl-1-propylpyrimido[4,5-d]pyrimidine-2,4-dione
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-2-phenoxypropanoate —— C16H14N2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-2-phenoxypropanoate
—— 5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]pyridin-1-ium-2-amine —— C22H30N3O3S+
5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]pyridin-1-ium-2-amine
—— (5S)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H31NO4S2
(5S)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]pyridin-2-amine —— C22H29N3O3S
5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]pyridin-2-amine
—— (5R)-5-tert-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H31NO4S2
(5R)-5-tert-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-(4-methylphenyl)-4-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine —— C21H21N5S
5-(4-methylphenyl)-4-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine
—— (5R)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H31NO4S2
(5R)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]pyridin-2-amine —— C22H29N3O3S
5-(4-benzylpiperidin-1-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]pyridin-2-amine
—— 5-(furan-2-yl)-3-[2-[(3R)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-1,3,4-oxadiazol-2-one —— C24H20N4O5
5-(furan-2-yl)-3-[2-[(3R)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-1,3,4-oxadiazol-2-one
—— 5-[(1R)-1-(2-bromophenyl)sulfanylethyl]-3-phenyl-1,2,4-oxadiazole —— C16H13BrN2OS
5-[(1R)-1-(2-bromophenyl)sulfanylethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-tert-butyl-3-[[(2R)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H24N4O
5-tert-butyl-3-[[(2R)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-ethyl-7-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C16H24N6
5-ethyl-7-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-methyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H23N5O
5-methyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-methyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H23N5O
5-methyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-7-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C16H24N6
5-ethyl-7-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-methyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H23N5O
5-methyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-[(1R)-1-[4-(2,6-dimethoxyphenoxy)piperidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C18H25N3O4
5-[(1R)-1-[4-(2,6-dimethoxyphenoxy)piperidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(1S)-1-(2-bromophenyl)sulfanylethyl]-3-phenyl-1,2,4-oxadiazole —— C16H13BrN2OS
5-[(1S)-1-(2-bromophenyl)sulfanylethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(2,4,5-Trichlorophenoxy)methyl]-1,3-benzodioxole —— C14H9Cl3O3
5-[(2,4,5-Trichlorophenoxy)methyl]-1,3-benzodioxole
—— 5-tert-butyl-3-[[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H24N4O
5-tert-butyl-3-[[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[(1S)-1-[4-(2,6-dimethoxyphenoxy)piperidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C18H25N3O4
5-[(1S)-1-[4-(2,6-dimethoxyphenoxy)piperidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-methyl-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H23N5O
5-methyl-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-(trifluoromethyl)-7-[(3R)-3-(trifluoromethyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C12H11F6N5
5-(trifluoromethyl)-7-[(3R)-3-(trifluoromethyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-bromo-N-[2-[4-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]-2-oxoethyl]furan-2-carboxamide —— C20H29BrN4O4
5-bromo-N-[2-[4-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]-2-oxoethyl]furan-2-carboxamide
—— 5-(trifluoromethyl)-7-[(3S)-3-(trifluoromethyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C12H11F6N5
5-(trifluoromethyl)-7-[(3S)-3-(trifluoromethyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-methyl-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]thiophene-2-carboxamide —— C16H18N4OS2
5-methyl-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]thiophene-2-carboxamide
—— 5-(4-Ethoxyphenyl)-3-(pyrrolidin-1-ium-1-ylmethyl)-1,3,4-oxadiazole-2-thione —— C15H20N3O2S+
5-(4-Ethoxyphenyl)-3-(pyrrolidin-1-ium-1-ylmethyl)-1,3,4-oxadiazole-2-thione
—— (5R)-7-amino-5-(2-ethoxyphenyl)-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C16H14N4O4
(5R)-7-amino-5-(2-ethoxyphenyl)-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— (5E)-5-[(3-chlorophenyl)methylidene]-3-(2-ethoxyphenyl)-2-phenylimidazol-4-one —— C24H19ClN2O2
(5E)-5-[(3-chlorophenyl)methylidene]-3-(2-ethoxyphenyl)-2-phenylimidazol-4-one
—— (5E)-5-[(3-chlorophenyl)methylidene]-3-(4-ethoxyphenyl)-2-phenylimidazol-4-one —— C24H19ClN2O2
(5E)-5-[(3-chlorophenyl)methylidene]-3-(4-ethoxyphenyl)-2-phenylimidazol-4-one
—— 5-[[4-(4-Chlorophenyl)-3-ethoxycarbonylthiophen-2-yl]amino]-5-oxopentanoate —— C18H17ClNO5S-
5-[[4-(4-Chlorophenyl)-3-ethoxycarbonylthiophen-2-yl]amino]-5-oxopentanoate
—— 5-chloro-4-(4-methylphenyl)sulfonyl-2-[(3R)-3-methylpiperidin-1-yl]-1,3-thiazole —— C16H19ClN2O2S2
5-chloro-4-(4-methylphenyl)sulfonyl-2-[(3R)-3-methylpiperidin-1-yl]-1,3-thiazole
—— 5-[[4-(4-Chlorophenyl)-3-ethoxycarbonylthiophen-2-yl]amino]-5-oxopentanoic acid —— C18H18ClNO5S
5-[[4-(4-Chlorophenyl)-3-ethoxycarbonylthiophen-2-yl]amino]-5-oxopentanoic acid
—— 5-[(1R)-1-[[4-(2-methoxyphenyl)-5-piperidin-1-yl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C24H26N6O2S
5-[(1R)-1-[[4-(2-methoxyphenyl)-5-piperidin-1-yl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole