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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol —— C19H21N5O2
(3S)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol
—— 7-[(1-Acetylindol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H21N5O2
7-[(1-Acetylindol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-(furan-2-ylmethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-methylpyridin-3-yl)pyrimidin-2-amine —— C19H17N5O2
N-(furan-2-ylmethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-methylpyridin-3-yl)pyrimidin-2-amine
—— 7-[(2,5-Dimethyl-1-pyridin-2-ylpyrrol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[(2,5-Dimethyl-1-pyridin-2-ylpyrrol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Methylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H18N6O
7-[(1-Methylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [(3S)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-yl]methanol —— C20H23N5O2
[(3S)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-yl]methanol
—— 7-[(2,5-Dimethoxy-4-pyrrolidin-1-ylphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O3
7-[(2,5-Dimethoxy-4-pyrrolidin-1-ylphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-morpholin-4-ylethyl)pyrimidin-2-amine —— C19H23N7O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-morpholin-4-ylethyl)pyrimidin-2-amine
—— 7-[(1-Ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N6O
7-[(1-Ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-(3-ethoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine —— C19H23N5O2
N-(3-ethoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine
—— 7-[(1-Benzylbenzimidazol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C27H24N6O
7-[(1-Benzylbenzimidazol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 1-[3-[[5-(3-Methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]amino]propyl]pyrrolidin-2-one —— C21H24N6O2
1-[3-[[5-(3-Methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]amino]propyl]pyrrolidin-2-one
—— N-(3-methoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine —— C18H21N5O2
N-(3-methoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine
—— 2-Pyridin-2-yl-7-[[2-(pyridin-2-ylmethoxy)phenyl]methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H23N5O2
2-Pyridin-2-yl-7-[[2-(pyridin-2-ylmethoxy)phenyl]methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-Pyridin-2-yl-7-[(2-thiomorpholin-4-ylpyrimidin-4-yl)methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H23N7OS
2-Pyridin-2-yl-7-[(2-thiomorpholin-4-ylpyrimidin-4-yl)methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-Pyridin-2-yl-7-[[4-(trifluoromethoxy)phenyl]methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H17F3N4O2
2-Pyridin-2-yl-7-[[4-(trifluoromethoxy)phenyl]methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19ClN6O
7-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C18H20N6O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— 7-[(7-ethyl-1H-indol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H23N5O
7-[(7-ethyl-1H-indol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-[(5-methylfuran-2-yl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine —— C20H19N5O2
N-[(5-methylfuran-2-yl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine
—— 5-[2-(4-Ethylpiperazin-1-yl)-4-(6-methylpyridin-3-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole —— C20H24N6O
5-[2-(4-Ethylpiperazin-1-yl)-4-(6-methylpyridin-3-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole
—— N-methyl-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-(2-pyridin-2-ylethyl)pyrimidin-2-amine —— C22H22N6O
N-methyl-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-(2-pyridin-2-ylethyl)pyrimidin-2-amine
—— 7-[[4-Methoxy-3-(pyrazol-1-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O2
7-[[4-Methoxy-3-(pyrazol-1-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 3-[3-[(4-Oxo-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-7-yl)methyl]indol-1-yl]propanamide —— C24H24N6O2
3-[3-[(4-Oxo-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-7-yl)methyl]indol-1-yl]propanamide
—— N-(2-methoxyethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine —— C16H18N6O2
N-(2-methoxyethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine
—— 7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-Methoxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O3
7-[[4-Methoxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-Pyridin-4-yl-7-(quinolin-4-ylmethyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19N5O
2-Pyridin-4-yl-7-(quinolin-4-ylmethyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-(2-methoxyethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine —— C17H19N5O2
N-(2-methoxyethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine
—— N-(1,3-benzodioxol-5-ylmethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine —— C22H19N5O3
N-(1,3-benzodioxol-5-ylmethyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine
—— 7-[(1-Methylpyrrol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H19N5O
7-[(1-Methylpyrrol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-(Diethylamino)-2-methoxyphenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H29N5O2
7-[[4-(Diethylamino)-2-methoxyphenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 5-methyl-3-[(4-oxo-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-7-yl)methyl]-1H-indole-2-carboxylic acid —— C23H21N5O3
5-methyl-3-[(4-oxo-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-7-yl)methyl]-1H-indole-2-carboxylic acid
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine —— C20H18N6O
5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
—— 3-Methyl-5-[4-(2-methylpyridin-3-yl)-2-thiomorpholin-4-ylpyrimidin-5-yl]-1,2-oxazole —— C18H19N5OS
3-Methyl-5-[4-(2-methylpyridin-3-yl)-2-thiomorpholin-4-ylpyrimidin-5-yl]-1,2-oxazole
—— (3R)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol —— C19H21N5O2
(3R)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol
—— 7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H26N6O
7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-Methyl-4-morpholin-4-ylphenyl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27N5O2
7-[(2-Methyl-4-morpholin-4-ylphenyl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C18H20N6O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— 7-[(2,7-Dimethoxyquinolin-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H23N5O3
7-[(2,7-Dimethoxyquinolin-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine —— C19H17N5OS
5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine
—— 7-[[4-Methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O2
7-[[4-Methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Ethyl-5-methoxyindol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H25N5O2
7-[(1-Ethyl-5-methoxyindol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(6-methylpyridin-3-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C19H21N5O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(6-methylpyridin-3-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— 7-[[1-(4-Fluorophenyl)pyrazol-4-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19FN6O
7-[[1-(4-Fluorophenyl)pyrazol-4-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(6-Bromo-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H17BrN4O3
7-[(6-Bromo-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[1-(4-Methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H27N5O2
7-[[1-(4-Methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27N5O
7-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [(3R)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-yl]methanol —— C20H23N5O2
[(3R)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-yl]methanol
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-propan-2-ylpyrimidin-2-amine —— C17H19N5O
5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)-N-propan-2-ylpyrimidin-2-amine