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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(4-fluorophenyl)methyl]-2-methyl-6-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]pyridine-3-carboxamide —— C23H22FN5O2
N-[(4-fluorophenyl)methyl]-2-methyl-6-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]pyridine-3-carboxamide
—— N-[(4-fluorophenyl)methyl]-2-methyl-6-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]pyridine-3-carboxamide —— C23H22FN5O2
N-[(4-fluorophenyl)methyl]-2-methyl-6-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]pyridine-3-carboxamide
—— (6R)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H35N5O3
(6R)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H35N5O3
(6S)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— N,N-dimethyl-3-[[(2S)-1-(5-methylpyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C24H28N4O2S
N,N-dimethyl-3-[[(2S)-1-(5-methylpyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— N,N-dimethyl-3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C24H28N4O2S
N,N-dimethyl-3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— N-propan-2-yl-3-[[(2S)-1-(pyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C24H28N4O2S
N-propan-2-yl-3-[[(2S)-1-(pyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— N-propan-2-yl-3-[[(2R)-1-(pyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C24H28N4O2S
N-propan-2-yl-3-[[(2R)-1-(pyrazine-2-carbonyl)azepan-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— N-(2-methoxyethyl)-3-[[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C23H26N4O3S
N-(2-methoxyethyl)-3-[[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— 3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C20H20N4O2S
3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— 3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]methyl]-N-propan-2-yl-1-benzothiophene-2-carboxamide —— C24H28N4O2S
3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]methyl]-N-propan-2-yl-1-benzothiophene-2-carboxamide
—— N-(2-methoxyethyl)-3-[[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C23H26N4O3S
N-(2-methoxyethyl)-3-[[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— N-(2-methoxyethyl)-3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C23H26N4O3S
N-(2-methoxyethyl)-3-[[(2R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— 3-[[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide —— C20H20N4O2S
3-[[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]methyl]-1-benzothiophene-2-carboxamide
—— 4-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide —— C14H22N4O
4-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-amine —— C14H25N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-amine
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine —— C16H29N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine —— C16H29N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine
—— N-[[4-[(3R)-1-(diethylsulfamoyl)piperidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide —— C18H32N6O3S
N-[[4-[(3R)-1-(diethylsulfamoyl)piperidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-amine —— C14H25N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-amine
—— N-[[4-[(3S)-1-(diethylsulfamoyl)piperidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide —— C18H32N6O3S
N-[[4-[(3S)-1-(diethylsulfamoyl)piperidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide
—— N,N,4-trimethyl-2-[(3S)-1-methylpiperidin-3-yl]pyrimidine-5-carboxamide —— C14H22N4O
N,N,4-trimethyl-2-[(3S)-1-methylpiperidin-3-yl]pyrimidine-5-carboxamide
—— 4-methyl-2-[(2S)-1-pyrimidin-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide —— C15H18N6O
4-methyl-2-[(2S)-1-pyrimidin-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide
—— N,N,4-trimethyl-2-[(3R)-1-methylpiperidin-3-yl]pyrimidine-5-carboxamide —— C14H22N4O
N,N,4-trimethyl-2-[(3R)-1-methylpiperidin-3-yl]pyrimidine-5-carboxamide
—— 4-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide —— C14H22N4O
4-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide
—— 2-[(2S)-1-acetylpiperidin-2-yl]-4-methylpyrimidine-5-carboxamide —— C13H18N4O2
2-[(2S)-1-acetylpiperidin-2-yl]-4-methylpyrimidine-5-carboxamide
—— 2-[(3R)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpyrrolidin-3-yl]-4,6-dimethylpyrimidine —— C16H23N5O2S
2-[(3R)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpyrrolidin-3-yl]-4,6-dimethylpyrimidine
—— 2-[(2R)-1-acetylpiperidin-2-yl]-4-methylpyrimidine-5-carboxamide —— C13H18N4O2
2-[(2R)-1-acetylpiperidin-2-yl]-4-methylpyrimidine-5-carboxamide
—— 2-[(3R)-1-(1,3-dimethylpyrazol-4-yl)sulfonylpyrrolidin-3-yl]-4,6-dimethylpyrimidine —— C15H21N5O2S
2-[(3R)-1-(1,3-dimethylpyrazol-4-yl)sulfonylpyrrolidin-3-yl]-4,6-dimethylpyrimidine
—— 6-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H21N5O3
6-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 4-methyl-2-[(2R)-1-pyrimidin-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide —— C15H18N6O
4-methyl-2-[(2R)-1-pyrimidin-2-ylpiperidin-2-yl]pyrimidine-5-carboxamide
—— 4-methyl-2-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-6-(trifluoromethyl)pyrimidine —— C11H14F3N3O2S
4-methyl-2-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-6-(trifluoromethyl)pyrimidine
—— N,1,3-trimethyl-2,4-dioxo-N-(thiophen-2-ylmethyl)pyrimidine-5-sulfonamide —— C12H15N3O4S2
N,1,3-trimethyl-2,4-dioxo-N-(thiophen-2-ylmethyl)pyrimidine-5-sulfonamide
—— [(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(4-methylpyrimidin-5-yl)methanone —— C16H19N5O
[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(4-methylpyrimidin-5-yl)methanone
—— [(3S)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]-pyrazin-2-ylmethanone —— C14H17N5O3S
[(3S)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]-pyrazin-2-ylmethanone
—— 4-methyl-2-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-6-(trifluoromethyl)pyrimidine —— C11H14F3N3O2S
4-methyl-2-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-6-(trifluoromethyl)pyrimidine
—— 6-[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H21N5O3
6-[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 4-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]sulfonylmorpholine —— C14H22N4O3S
4-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]sulfonylmorpholine
—— [2-(dimethylamino)pyrimidin-5-yl]-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methanone —— C17H22N6O
[2-(dimethylamino)pyrimidin-5-yl]-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methanone
—— 2-[(3S)-1-(1,3-dimethylpyrazol-4-yl)sulfonylpyrrolidin-3-yl]-4,6-dimethylpyrimidine —— C15H21N5O2S
2-[(3S)-1-(1,3-dimethylpyrazol-4-yl)sulfonylpyrrolidin-3-yl]-4,6-dimethylpyrimidine
—— [(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(4-methylpyrimidin-5-yl)methanone —— C16H19N5O
[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(4-methylpyrimidin-5-yl)methanone
—— [(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C16H19N5O
[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— (5-methylpyrazin-2-yl)-[(3R)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C15H19N5O3S
(5-methylpyrazin-2-yl)-[(3R)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— [2-(dimethylamino)pyrimidin-5-yl]-[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methanone —— C17H22N6O
[2-(dimethylamino)pyrimidin-5-yl]-[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methanone
—— [(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C16H19N5O
[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3R)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]-pyrimidin-5-ylmethanone —— C14H17N5O3S
[(3R)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]-pyrimidin-5-ylmethanone
—— pyrazin-2-yl-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C13H15N5O
pyrazin-2-yl-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— [(3S)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]-pyrimidin-5-ylmethanone —— C14H17N5O3S
[(3S)-3-(4-methylsulfonyl-1H-pyrazol-5-yl)piperidin-1-yl]-pyrimidin-5-ylmethanone
—— pyrazin-2-yl-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C13H15N5O
pyrazin-2-yl-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— 2-methyl-6-[(3R)-1-thiophen-2-ylsulfonylpiperidin-3-yl]pyrazine —— C14H17N3O2S2
2-methyl-6-[(3R)-1-thiophen-2-ylsulfonylpiperidin-3-yl]pyrazine