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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-ethyl-5-[(1S)-1-[2-[2-(furan-2-yl)pyrimidin-5-yl]imidazol-1-yl]ethyl]-1,2,4-oxadiazole —— C17H16N6O2
3-ethyl-5-[(1S)-1-[2-[2-(furan-2-yl)pyrimidin-5-yl]imidazol-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-[(1S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-hydroxyethyl]phenol —— C17H21N3O2
3-[(1S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-hydroxyethyl]phenol
—— 4-cyclobutyl-6-methyl-N-[(1R)-1-(2-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine —— C14H20N6
4-cyclobutyl-6-methyl-N-[(1R)-1-(2-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
—— 1-[4-[[(2S)-2-ethoxypropyl]-methylamino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H27N5O2
1-[4-[[(2S)-2-ethoxypropyl]-methylamino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 1-[4-[[(2S)-2,3-dihydroxypropyl]-methylamino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H23N5O3
1-[4-[[(2S)-2,3-dihydroxypropyl]-methylamino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 2-[(1R)-1-[[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino]ethyl]phenol —— C15H16F3N3O
2-[(1R)-1-[[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino]ethyl]phenol
—— (3S)-4-(cyclopropylmethyl)-1-(4-methyl-2-propan-2-ylpyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C21H32N4O2
(3S)-4-(cyclopropylmethyl)-1-(4-methyl-2-propan-2-ylpyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— [(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-pyrazin-2-ylmethanone —— C17H26N4O
[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-pyrazin-2-ylmethanone
—— methyl (4S)-4-(2-chloro-6-fluorophenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C13H12ClFN2O2S
methyl (4S)-4-(2-chloro-6-fluorophenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H18F2N2O4S
ethyl (4S)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-[4-[[(3S)-3-(dimethylamino)butyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H28N6O
1-[4-[[(3S)-3-(dimethylamino)butyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— methyl (4R)-6-methyl-2-sulfanylidene-4-(2,3,4-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H20N2O5S
methyl (4R)-6-methyl-2-sulfanylidene-4-(2,3,4-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 4-cyclobutyl-6-methyl-N-[(1S)-1-(2-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine —— C14H20N6
4-cyclobutyl-6-methyl-N-[(1S)-1-(2-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
—— N-[(S)-cyclopropyl-(4-methylpyridin-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C17H19F3N4
N-[(S)-cyclopropyl-(4-methylpyridin-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 2-[(1S)-1-[[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino]ethyl]phenol —— C15H16F3N3O
2-[(1S)-1-[[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino]ethyl]phenol
—— [(3S)-1-[2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl]piperidin-3-yl]methanol —— C17H28N4O
[(3S)-1-[2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl]piperidin-3-yl]methanol
—— 1-[4-[[(3R)-3-(dimethylamino)butyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H28N6O
1-[4-[[(3R)-3-(dimethylamino)butyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 2-methoxyethyl (4R)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H20F2N2O5S
2-methoxyethyl (4R)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-methyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C21H30N6
N-methyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— 2-methoxyethyl (4S)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H20F2N2O5S
2-methoxyethyl (4S)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-[4-[[(2R)-2,3-dihydroxypropyl]-methylamino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H23N5O3
1-[4-[[(2R)-2,3-dihydroxypropyl]-methylamino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 6-(1-methylimidazol-2-yl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine —— C15H17N7
6-(1-methylimidazol-2-yl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine
—— 6-(1-methylimidazol-2-yl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine —— C15H17N7
6-(1-methylimidazol-2-yl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine
—— methyl (4S)-6-methyl-2-sulfanylidene-4-(2,3,4-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H20N2O5S
methyl (4S)-6-methyl-2-sulfanylidene-4-(2,3,4-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (2R)-2-(6-methoxynaphthalen-2-yl)-4-(6-phenylpyridazin-3-yl)morpholine —— C25H23N3O2
(2R)-2-(6-methoxynaphthalen-2-yl)-4-(6-phenylpyridazin-3-yl)morpholine
—— [(3R)-1-[2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl]piperidin-3-yl]methanol —— C17H28N4O
[(3R)-1-[2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl]piperidin-3-yl]methanol
—— 5-[2-[(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione —— C15H21N3O3
5-[2-[(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione
—— 7-[(2S)-1,4-dioxane-2-carbonyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H18N4O4
7-[(2S)-1,4-dioxane-2-carbonyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H30N4O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— (2S)-2-(6-methoxynaphthalen-2-yl)-4-(6-phenylpyridazin-3-yl)morpholine —— C25H23N3O2
(2S)-2-(6-methoxynaphthalen-2-yl)-4-(6-phenylpyridazin-3-yl)morpholine
—— 6-[(3R)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H24N4O4
6-[(3R)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H30N4O2
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— 5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H29FN4
5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— (3S)-4-benzyl-3-ethyl-1-(4-methylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H24N4O2
(3S)-4-benzyl-3-ethyl-1-(4-methylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— ethyl (4R)-4-ethyl-2-oxo-6-[(4-oxo-4-thiophen-2-ylbutanoyl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H22N2O6S
ethyl (4R)-4-ethyl-2-oxo-6-[(4-oxo-4-thiophen-2-ylbutanoyl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (3R)-4-benzyl-3-ethyl-1-(4-methylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H24N4O2
(3R)-4-benzyl-3-ethyl-1-(4-methylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— 6-[(3S)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H24N4O4
6-[(3S)-4-(cyclopropylmethyl)-5-oxo-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione
—— [(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone —— C21H25F2N3O
[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone
—— ethyl (4S)-4-ethyl-2-oxo-6-[(4-oxo-4-thiophen-2-ylbutanoyl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H22N2O6S
ethyl (4S)-4-ethyl-2-oxo-6-[(4-oxo-4-thiophen-2-ylbutanoyl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-methyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C21H30N6
N-methyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— [(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone —— C21H25F2N3O
[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone
—— (4S)-1-tert-butyl-4-[[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-methylamino]methyl]pyrrolidin-2-one —— C21H29N5O
(4S)-1-tert-butyl-4-[[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-methylamino]methyl]pyrrolidin-2-one
—— 4-cyclobutyl-6-methyl-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrimidin-2-amine —— C17H25N5
4-cyclobutyl-6-methyl-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrimidin-2-amine
—— (4R)-1-tert-butyl-4-[[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-methylamino]methyl]pyrrolidin-2-one —— C21H29N5O
(4R)-1-tert-butyl-4-[[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-methylamino]methyl]pyrrolidin-2-one
—— 7-[(2R)-1,4-dioxane-2-carbonyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H18N4O4
7-[(2R)-1,4-dioxane-2-carbonyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [(3R)-1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-3-yl]-pyridin-2-ylmethanone —— C22H22N4O2
[(3R)-1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-3-yl]-pyridin-2-ylmethanone
—— 2-methyl-5-[[2-[(1S)-1-phenylethyl]imidazol-1-yl]methyl]pyrazine —— C17H18N4
2-methyl-5-[[2-[(1S)-1-phenylethyl]imidazol-1-yl]methyl]pyrazine
—— [(3S)-1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-3-yl]-pyridin-2-ylmethanone —— C22H22N4O2
[(3S)-1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-3-yl]-pyridin-2-ylmethanone
—— methyl (4S)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H16F2N2O4S
methyl (4S)-4-[4-(difluoromethoxy)-3-methoxyphenyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 5-[2-[(3R)-3-aminopyrrolidin-1-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid —— C17H20N4O3
5-[2-[(3R)-3-aminopyrrolidin-1-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid