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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-N-(4-fluorophenyl)acetamide —— C24H26FN5O2
2-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-N-(4-fluorophenyl)acetamide
—— 2-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-N,N-dimethylacetamide —— C20H27N5O2
2-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-N,N-dimethylacetamide
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-phenylethanone —— C23H23FN4O
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-phenylethanone
—— 5-(2-fluorophenyl)-4-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C21H20F2N4O2S
5-(2-fluorophenyl)-4-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone —— C21H26ClN5O2
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone
—— [(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone —— C21H25FN4O
[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone
—— [(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone —— C22H28N4O2
[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone
—— [(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-3-ylmethanone —— C21H20ClN5O
[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-3-ylmethanone
—— (2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]-N,N-dimethylpiperidine-1-sulfonamide —— C18H22F3N5O2S
(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]-N,N-dimethylpiperidine-1-sulfonamide
—— 2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol —— C16H19ClN4O
2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol
—— [(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone —— C22H25F3N4O
[(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-phenoxyethanone —— C23H23ClN4O2
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-phenoxyethanone
—— 1-[(2S)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone —— C22H24FN5OS
1-[(2S)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone
—— [(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19ClN6O
[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— 2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N-pyridin-2-ylacetamide —— C22H23FN6O
2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N-pyridin-2-ylacetamide
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone —— C21H26FN5O2
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone
—— [(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-3-ylmethanone —— C21H20FN5O
[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-3-ylmethanone
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C25H27FN4O2
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— 5-(3-fluorophenyl)-4-[(2S)-1-(pyridin-2-ylmethyl)piperidin-2-yl]pyrimidin-2-amine —— C21H22FN5
5-(3-fluorophenyl)-4-[(2S)-1-(pyridin-2-ylmethyl)piperidin-2-yl]pyrimidin-2-amine
—— 5-(4-chlorophenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]pyrimidin-2-amine —— C21H22ClN5
5-(4-chlorophenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-fluorophenyl)ethanone —— C23H23FN4O
1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-phenylethanone —— C24H26N4O2
1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-phenylethanone
—— 2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N-pyridin-2-ylacetamide —— C22H23ClN6O
2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N-pyridin-2-ylacetamide
—— 1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone —— C24H25FN4O2
1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone —— C23H22F2N4O
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N-(1,3-thiazol-2-yl)acetamide —— C20H21FN6OS
2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N-(1,3-thiazol-2-yl)acetamide
—— 5-(4-fluorophenyl)-4-[(2S)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C22H23FN4O3S
5-(4-fluorophenyl)-4-[(2S)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone —— C18H21FN4O2
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone
—— 2-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-N,N-diethylacetamide —— C22H31N5O2
2-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-N,N-diethylacetamide
—— 5-(4-chlorophenyl)-4-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C21H20ClFN4O2S
5-(4-chlorophenyl)-4-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone —— C24H25FN4O2
1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenylpropan-1-one —— C24H25FN4O
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenylpropan-1-one
—— [(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-cyclopentylmethanone —— C21H26N4O
[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-cyclopentylmethanone
—— 2-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-N,N-diethylacetamide —— C21H29N5O
2-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-N,N-diethylacetamide
—— 2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N,N-diethylacetamide —— C21H28ClN5O
2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-N,N-diethylacetamide
—— [(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H21N5OS
[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-4-ylmethanone —— C22H23N5O2
[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-4-ylmethanone
—— 1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-methoxyphenyl)ethanone —— C24H26N4O2
1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-methoxyphenyl)ethanone
—— 2-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone —— C21H26ClN5O
2-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone
—— [(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19FN6O
[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— 5-(3-fluorophenyl)-4-[(2S)-1-pyrazin-2-ylpyrrolidin-2-yl]pyrimidin-2-amine —— C18H17FN6
5-(3-fluorophenyl)-4-[(2S)-1-pyrazin-2-ylpyrrolidin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-3-ylmethanone —— C21H20FN5O
[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-pyridin-3-ylmethanone
—— 1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenylpropan-1-one —— C24H25ClN4O
1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenylpropan-1-one
—— 1-[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-phenylethanone —— C24H23F3N4O
1-[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-phenylethanone
—— 2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone —— C21H26FN5O
2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone
—— 4-[2-amino-4-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)piperidin-2-yl]pyrimidin-5-yl]benzamide —— C22H28N6O2
4-[2-amino-4-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 4-[2-amino-4-[(2S)-1-(3-phenylpropanoyl)piperidin-2-yl]pyrimidin-5-yl]benzamide —— C25H27N5O2
4-[2-amino-4-[(2S)-1-(3-phenylpropanoyl)piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-pyridin-2-ylethanone —— C22H22FN5O
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-pyridin-2-ylethanone
—— 1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C26H30N4O3
1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— (2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylpiperidine-1-sulfonamide —— C17H22FN5O2S
(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylpiperidine-1-sulfonamide