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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (4S)-4-methyl-2-oxo-6-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17N5O4S
ethyl (4S)-4-methyl-2-oxo-6-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-methyl-2-oxo-6-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17N5O4S
ethyl (4R)-4-methyl-2-oxo-6-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (2S)-N,N-dimethyl-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propanamide —— C15H16F3N5O
(2S)-N,N-dimethyl-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propanamide
—— 5,6-dimethyl-2-pyridin-3-yl-N-[(1S)-1-pyridin-2-ylethyl]pyrimidin-4-amine —— C18H19N5
5,6-dimethyl-2-pyridin-3-yl-N-[(1S)-1-pyridin-2-ylethyl]pyrimidin-4-amine
—— (2R)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butan-1-ol —— C14H15F3N4O
(2R)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butan-1-ol
—— (2S)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butan-1-ol —— C14H15F3N4O
(2S)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butan-1-ol
—— 2-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]-4-(4-methylphenyl)phthalazin-1-one —— C24H27N3O2
2-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]-4-(4-methylphenyl)phthalazin-1-one
—— (3R)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-3-(trifluoromethyl)piperidin-3-ol —— C16H17F3N4O
(3R)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-3-(trifluoromethyl)piperidin-3-ol
—— (3S)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-3-(trifluoromethyl)piperidin-3-ol —— C16H17F3N4O
(3S)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-3-(trifluoromethyl)piperidin-3-ol
—— 2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-4-(4-methylphenyl)phthalazin-1-one —— C24H27N3O2
2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-4-(4-methylphenyl)phthalazin-1-one
—— ethyl (4R)-6-[[2-(3,4-dimethylphenyl)acetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O5
ethyl (4R)-6-[[2-(3,4-dimethylphenyl)acetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[2-(3,4-dimethylphenyl)acetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O5
ethyl (4S)-6-[[2-(3,4-dimethylphenyl)acetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(2R)-2-cyclohexylazepan-1-yl]-pyrazin-2-ylmethanone —— C17H25N3O
[(2R)-2-cyclohexylazepan-1-yl]-pyrazin-2-ylmethanone
—— [(2S)-2-cyclohexylazepan-1-yl]-pyrazin-2-ylmethanone —— C17H25N3O
[(2S)-2-cyclohexylazepan-1-yl]-pyrazin-2-ylmethanone
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]prop-2-enoate —— C18H19ClN4O3S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]prop-2-enoate
—— (5aS,8aS)-5-(2-pyridin-4-ylquinazolin-4-yl)-2,3,4,5a,6,7,8,8a-octahydrocyclopenta[b][1,4]oxazepine —— C21H22N4O
(5aS,8aS)-5-(2-pyridin-4-ylquinazolin-4-yl)-2,3,4,5a,6,7,8,8a-octahydrocyclopenta[b][1,4]oxazepine
—— (2R)-2-ethyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine —— C16H17F3N4O
(2R)-2-ethyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine
—— (5aS,8aR)-5-(2-pyridin-3-ylquinazolin-4-yl)-2,3,4,5a,6,7,8,8a-octahydrocyclopenta[b][1,4]oxazepine —— C21H22N4O
(5aS,8aR)-5-(2-pyridin-3-ylquinazolin-4-yl)-2,3,4,5a,6,7,8,8a-octahydrocyclopenta[b][1,4]oxazepine
—— (2S)-2-ethyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine —— C16H17F3N4O
(2S)-2-ethyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine
—— (3S)-3-methyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine —— C15H15F3N4O
(3S)-3-methyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine
—— (2R)-2-[[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol —— C13H13F3N4O
(2R)-2-[[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol
—— (5aS,8aS)-5-(2-pyridin-3-ylquinazolin-4-yl)-2,3,4,5a,6,7,8,8a-octahydrocyclopenta[b][1,4]oxazepine —— C21H22N4O
(5aS,8aS)-5-(2-pyridin-3-ylquinazolin-4-yl)-2,3,4,5a,6,7,8,8a-octahydrocyclopenta[b][1,4]oxazepine
—— (3R)-3-methyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine —— C15H15F3N4O
(3R)-3-methyl-4-[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine
—— N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine —— C19H22N6
N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine
—— (2S)-2-[[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol —— C13H13F3N4O
(2S)-2-[[2-pyridin-3-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol
—— N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine —— C19H22N6
N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine
—— (2S)-2-(4-fluorophenyl)-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]ethanol —— C19H16FN5O
(2S)-2-(4-fluorophenyl)-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]ethanol
—— (2R)-2-(4-fluorophenyl)-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]ethanol —— C19H16FN5O
(2R)-2-(4-fluorophenyl)-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]ethanol
—— N-[(2R)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-4-ethylpyrimidine-5-carboxamide —— C17H20F2N4O
N-[(2R)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-4-ethylpyrimidine-5-carboxamide
—— N-[(2S)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-4-ethylpyrimidine-5-carboxamide —— C17H20F2N4O
N-[(2S)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-4-ethylpyrimidine-5-carboxamide
—— 4-ethyl-2-[6-[[(3S)-3-hydroxybutyl]amino]pyridin-3-yl]-1H-pyrimidin-6-one —— C15H20N4O2
4-ethyl-2-[6-[[(3S)-3-hydroxybutyl]amino]pyridin-3-yl]-1H-pyrimidin-6-one
—— 4-ethyl-2-[6-[[(3R)-3-hydroxybutyl]amino]pyridin-3-yl]-1H-pyrimidin-6-one —— C15H20N4O2
4-ethyl-2-[6-[[(3R)-3-hydroxybutyl]amino]pyridin-3-yl]-1H-pyrimidin-6-one
—— [(3S)-3-phenoxypyrrolidin-1-yl]-(2-phenylpyrimidin-5-yl)methanone —— C21H19N3O2
[(3S)-3-phenoxypyrrolidin-1-yl]-(2-phenylpyrimidin-5-yl)methanone
—— [(3R)-3-phenoxypyrrolidin-1-yl]-(2-phenylpyrimidin-5-yl)methanone —— C21H19N3O2
[(3R)-3-phenoxypyrrolidin-1-yl]-(2-phenylpyrimidin-5-yl)methanone
—— methyl 3-[(2-methylpyrimidine-4-carbonyl)-[[(2R)-oxolan-2-yl]methyl]amino]propanoate —— C15H21N3O4
methyl 3-[(2-methylpyrimidine-4-carbonyl)-[[(2R)-oxolan-2-yl]methyl]amino]propanoate
—— methyl 3-[(2-methylpyrimidine-4-carbonyl)-[[(2S)-oxolan-2-yl]methyl]amino]propanoate —— C15H21N3O4
methyl 3-[(2-methylpyrimidine-4-carbonyl)-[[(2S)-oxolan-2-yl]methyl]amino]propanoate
—— 3-[[(2R)-2-(2,4-difluorophenyl)-2-hydroxypropyl]amino]pyrazine-2-carbonitrile —— C14H12F2N4O
3-[[(2R)-2-(2,4-difluorophenyl)-2-hydroxypropyl]amino]pyrazine-2-carbonitrile
—— (2R)-1-[(5-bromopyrimidin-2-yl)amino]-2-phenylpropan-2-ol —— C13H14BrN3O
(2R)-1-[(5-bromopyrimidin-2-yl)amino]-2-phenylpropan-2-ol
—— 3-[[(2S)-2-(2,4-difluorophenyl)-2-hydroxypropyl]amino]pyrazine-2-carbonitrile —— C14H12F2N4O
3-[[(2S)-2-(2,4-difluorophenyl)-2-hydroxypropyl]amino]pyrazine-2-carbonitrile
—— (2S)-1-[(5-bromopyrimidin-2-yl)amino]-2-phenylpropan-2-ol —— C13H14BrN3O
(2S)-1-[(5-bromopyrimidin-2-yl)amino]-2-phenylpropan-2-ol
—— ethyl (4R)-4-[4-(cyanomethoxy)phenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17N3O4
ethyl (4R)-4-[4-(cyanomethoxy)phenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-[4-(cyanomethoxy)phenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17N3O4
ethyl (4S)-4-[4-(cyanomethoxy)phenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-2-(2,4-dioxopyrimidin-1-yl)acetamide —— C19H22ClFN4O4
N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-2-(2,4-dioxopyrimidin-1-yl)acetamide
—— 4-(4-methylphenyl)-2-[[4-[(3R)-3-methylpiperidine-1-carbonyl]piperidin-1-yl]methyl]phthalazin-1-one —— C28H34N4O2
4-(4-methylphenyl)-2-[[4-[(3R)-3-methylpiperidine-1-carbonyl]piperidin-1-yl]methyl]phthalazin-1-one
—— tert-butyl N-[(2R)-2,3-dimethyl-2-(pyrazine-2-carbonylamino)butyl]carbamate —— C16H26N4O3
tert-butyl N-[(2R)-2,3-dimethyl-2-(pyrazine-2-carbonylamino)butyl]carbamate
—— (2R)-2-(4,6-dimethylpyrimidin-2-yl)-3-oxo-5-(1,3-thiazol-4-yl)pentanenitrile —— C14H14N4OS
(2R)-2-(4,6-dimethylpyrimidin-2-yl)-3-oxo-5-(1,3-thiazol-4-yl)pentanenitrile
—— 3-[2-[(2R)-2-ethylpiperidin-1-yl]ethylamino]pyrazine-2-carbonitrile —— C14H21N5
3-[2-[(2R)-2-ethylpiperidin-1-yl]ethylamino]pyrazine-2-carbonitrile
—— N-[(2R)-1-ethylsulfonylpropan-2-yl]-4-(trifluoromethyl)pyrimidin-2-amine —— C10H14F3N3O2S
N-[(2R)-1-ethylsulfonylpropan-2-yl]-4-(trifluoromethyl)pyrimidin-2-amine
—— 3-[[(2S)-1-ethylsulfonylpropan-2-yl]amino]pyrazine-2-carbonitrile —— C10H14N4O2S
3-[[(2S)-1-ethylsulfonylpropan-2-yl]amino]pyrazine-2-carbonitrile
—— N-[(2S)-1-ethylsulfonylpropan-2-yl]-4-(trifluoromethyl)pyrimidin-2-amine —— C10H14F3N3O2S
N-[(2S)-1-ethylsulfonylpropan-2-yl]-4-(trifluoromethyl)pyrimidin-2-amine