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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (4S)-6-methyl-5-(morpholine-4-carbonyl)-4-phenyl-3,4-dihydro-1H-pyrimidin-2-one —— C16H19N3O3
(4S)-6-methyl-5-(morpholine-4-carbonyl)-4-phenyl-3,4-dihydro-1H-pyrimidin-2-one
—— (2R)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-2-(trifluoromethyl)morpholine —— C16H17F3N4O
(2R)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-2-(trifluoromethyl)morpholine
—— (3S)-4-(cyclopropylmethyl)-1-(6-oxo-1H-pyrazine-3-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C17H24N4O3
(3S)-4-(cyclopropylmethyl)-1-(6-oxo-1H-pyrazine-3-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— N-[(3R)-1-(7-acetyl-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-yl]acetamide —— C20H24N6O2
N-[(3R)-1-(7-acetyl-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-yl]acetamide
—— (3S)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide —— C18H22N6O
(3S)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide
—— 4-cyclobutyl-N-[[(2R)-1,4-dioxan-2-yl]methyl]-6-methylpyrimidin-2-amine —— C14H21N3O2
4-cyclobutyl-N-[[(2R)-1,4-dioxan-2-yl]methyl]-6-methylpyrimidin-2-amine
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]pyrimidin-2-amine —— C20H21N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]pyrimidin-2-amine
—— N-methyl-N-[[(2R)-oxan-2-yl]methyl]-2-propan-2-ylpyrimidine-4-carboxamide —— C15H23N3O2
N-methyl-N-[[(2R)-oxan-2-yl]methyl]-2-propan-2-ylpyrimidine-4-carboxamide
—— N-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C14H18F3N5O
N-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— (4R)-6-methyl-5-(morpholine-4-carbonyl)-4-phenyl-3,4-dihydro-1H-pyrimidin-2-one —— C16H19N3O3
(4R)-6-methyl-5-(morpholine-4-carbonyl)-4-phenyl-3,4-dihydro-1H-pyrimidin-2-one
—— [4-[(2S)-2-(2-phenylethyl)morpholin-4-yl]piperidin-1-yl]-pyrazin-2-ylmethanone —— C22H28N4O2
[4-[(2S)-2-(2-phenylethyl)morpholin-4-yl]piperidin-1-yl]-pyrazin-2-ylmethanone
—— 6-methyl-2-[2-[2-[(3S)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one —— C14H19N5O2
6-methyl-2-[2-[2-[(3S)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one
—— 1-[4-[[(2S)-1-hydroxyhexan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H27N5O2
1-[4-[[(2S)-1-hydroxyhexan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— ethyl (3S)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]butanoate —— C17H22N4O2
ethyl (3S)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]butanoate
—— 5-[[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H28F2N4
5-[[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— (3R)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide —— C18H22N6O
(3R)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide
—— (3R)-4-(cyclopropylmethyl)-1-(6-oxo-1H-pyrazine-3-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C17H24N4O3
(3R)-4-(cyclopropylmethyl)-1-(6-oxo-1H-pyrazine-3-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— 6-methyl-2-[2-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one —— C14H19N5O2
6-methyl-2-[2-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one
—— 4-cyclopentyl-N-[(1S)-1-(3-methylpyridin-2-yl)propyl]pyrimidin-2-amine —— C18H24N4
4-cyclopentyl-N-[(1S)-1-(3-methylpyridin-2-yl)propyl]pyrimidin-2-amine
—— [4-[(2R)-2-(2-phenylethyl)morpholin-4-yl]piperidin-1-yl]-pyrazin-2-ylmethanone —— C22H28N4O2
[4-[(2R)-2-(2-phenylethyl)morpholin-4-yl]piperidin-1-yl]-pyrazin-2-ylmethanone
—— N-[(1R)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C14H18F3N5O
N-[(1R)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 1-[4-[[(2R)-2-hydroxybutyl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H23N5O2
1-[4-[[(2R)-2-hydroxybutyl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— (4S)-1-tert-butyl-4-[[[6-(2-methoxyphenyl)pyridazin-3-yl]-methylamino]methyl]pyrrolidin-2-one —— C21H28N4O2
(4S)-1-tert-butyl-4-[[[6-(2-methoxyphenyl)pyridazin-3-yl]-methylamino]methyl]pyrrolidin-2-one
—— 4-cyclopentyl-N-[(1R)-1-(3-methylpyridin-2-yl)propyl]pyrimidin-2-amine —— C18H24N4
4-cyclopentyl-N-[(1R)-1-(3-methylpyridin-2-yl)propyl]pyrimidin-2-amine
—— [(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone —— C20H33N5O
[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone
—— 5-[4-[(3R)-3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H29N5O4
5-[4-[(3R)-3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 2-methoxyethyl (4S)-6-methyl-2-oxo-4-(2,4,6-trimethylphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24N2O4
2-methoxyethyl (4S)-6-methyl-2-oxo-4-(2,4,6-trimethylphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine —— C16H19N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine —— C16H19N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
—— [(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone —— C20H33N5O
[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone
—— 5-[4-[(3S)-3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H29N5O4
5-[4-[(3S)-3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 7-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (3S)-N-cyclopropyl-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide —— C20H29N5O2
(3S)-N-cyclopropyl-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
—— (3S)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-ethyl-3-methylpiperazin-2-one —— C18H23N5O
(3S)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-ethyl-3-methylpiperazin-2-one
—— 7-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— ethyl (4R)-6-(butanoyloxymethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H22N2O5
ethyl (4R)-6-(butanoyloxymethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 4-cyclopentyl-N-[[(2R)-oxan-2-yl]methyl]pyrimidin-2-amine —— C15H23N3O
4-cyclopentyl-N-[[(2R)-oxan-2-yl]methyl]pyrimidin-2-amine
—— 2-ethyl-5-[1-[(2R)-2-methoxy-2-thiophen-2-ylethyl]imidazol-2-yl]pyrimidine —— C16H18N4OS
2-ethyl-5-[1-[(2R)-2-methoxy-2-thiophen-2-ylethyl]imidazol-2-yl]pyrimidine
—— [(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone —— C21H25F2N3O
[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone
—— [(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone —— C16H23N3O
[(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone
—— 2-ethyl-5-[1-[(2S)-2-methoxy-2-thiophen-2-ylethyl]imidazol-2-yl]pyrimidine —— C16H18N4OS
2-ethyl-5-[1-[(2S)-2-methoxy-2-thiophen-2-ylethyl]imidazol-2-yl]pyrimidine
—— [(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone —— C21H25F2N3O
[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone
—— [(2S)-2-butyl-2,5-dihydropyrrol-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone —— C16H23N3O
[(2S)-2-butyl-2,5-dihydropyrrol-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone
—— 5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidin-6-one —— C20H25FN4O2
5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidin-6-one
—— 5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidin-6-one —— C20H25FN4O2
5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidin-6-one
—— 1-[4-[[(2R)-2-phenylpropyl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C23H25N5O
1-[4-[[(2R)-2-phenylpropyl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— (1R)-1-[1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-4-yl]propan-1-ol —— C19H25N3O2
(1R)-1-[1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-4-yl]propan-1-ol
—— (3R)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-ethyl-3-methylpiperazin-2-one —— C18H23N5O
(3R)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-ethyl-3-methylpiperazin-2-one
—— (3R)-N-cyclopropyl-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide —— C20H29N5O2
(3R)-N-cyclopropyl-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
—— 6-[[(2R)-2-(trifluoromethyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C10H12F3N3O3
6-[[(2R)-2-(trifluoromethyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione