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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 6-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— [(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C21H21F3N6O
[(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 5-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone —— C21H22ClN5OS
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone
—— 1-[4-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]piperidin-1-yl]ethanone —— C23H28FN5O2
1-[4-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]piperidin-1-yl]ethanone
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenoxypropan-1-one —— C24H25FN4O2
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenoxypropan-1-one
—— 5-(3-fluorophenyl)-4-[(2S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine —— C22H25FN6
5-(3-fluorophenyl)-4-[(2S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19ClN6O
[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— [(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C21H20F3N5OS
[(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 6-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— 5-(4-fluorophenyl)-4-[(2R)-1-(1H-indol-5-ylmethyl)piperidin-2-yl]pyrimidin-2-amine —— C24H24FN5
5-(4-fluorophenyl)-4-[(2R)-1-(1H-indol-5-ylmethyl)piperidin-2-yl]pyrimidin-2-amine
—— 6-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— [(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C20H19F3N6O
[(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— 1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C25H27FN4O2
1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— [(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylimidazol-2-yl)methanone —— C21H21F3N6O
[(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylimidazol-2-yl)methanone
—— [(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone —— C21H25ClN4O
[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone —— C19H24ClN5O
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone —— C19H24FN5O
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone —— C21H22ClN5OS
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone
—— 1-[4-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidine-1-carbonyl]piperidin-1-yl]ethanone —— C23H29N5O2
1-[4-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidine-1-carbonyl]piperidin-1-yl]ethanone
—— 1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C25H27FN4O2
1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— [(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C20H22N6O2
[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— 1-[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone —— C20H24F3N5O
1-[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
—— [(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19FN6O
[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— 4-[2-amino-4-[(2S)-1-[2-(4-fluorophenoxy)ethyl]piperidin-2-yl]pyrimidin-5-yl]benzamide —— C24H26FN5O2
4-[2-amino-4-[(2S)-1-[2-(4-fluorophenoxy)ethyl]piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 4-[2-amino-4-[(2S)-1-[2-(azepan-1-yl)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide —— C24H32N6O2
4-[2-amino-4-[(2S)-1-[2-(azepan-1-yl)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-pyrrolidin-1-ylethanone —— C21H26ClN5O
1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-pyrrolidin-1-ylethanone
—— [(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20FN5OS
[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20FN5OS
[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone —— C19H24N4O3
1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone
—— 1-[4-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]piperidin-1-yl]ethanone —— C23H28ClN5O2
1-[4-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]piperidin-1-yl]ethanone
—— 6-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— [(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C21H23N5O2S
[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19ClN6O
[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— [(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20FN5OS
[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone —— C23H22F2N4O
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 3-[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidine-1-carbonyl]-1H-pyridazin-6-one —— C21H19F3N6O2
3-[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidine-1-carbonyl]-1H-pyridazin-6-one
—— [(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C20H21ClN6O
[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— [(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C20H22N6O
[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— [(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20FN5OS
[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20ClN5OS
[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(1H-indol-3-yl)ethanone —— C26H27N5O2
1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(1H-indol-3-yl)ethanone
—— 4-[2-amino-4-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide —— C24H24FN5O2
4-[2-amino-4-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(1H-indol-3-yl)ethanone —— C25H24ClN5O
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(1H-indol-3-yl)ethanone
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(1H-indol-3-yl)ethanone —— C25H24FN5O
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(1H-indol-3-yl)ethanone
—— 1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone —— C22H29N5O3
1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone —— C23H22ClFN4O
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 5-(3-chlorophenyl)-4-[(2R)-1-(quinoxalin-6-ylmethyl)piperidin-2-yl]pyrimidin-2-amine —— C24H23ClN6
5-(3-chlorophenyl)-4-[(2R)-1-(quinoxalin-6-ylmethyl)piperidin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19ClN6O
[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone