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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(3S)-3-[2-[(3-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]ethanol —— C17H23N5O
2-[(3S)-3-[2-[(3-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]ethanol
—— 4-[(2R)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C20H22N6O
4-[(2R)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— 1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H25FN4O
1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 4-[(2R)-1-methylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C13H16N6
4-[(2R)-1-methylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— 4-[(2S)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C20H22N6O
4-[(2S)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— 4-[(2R)-1-methylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C14H18N6
4-[(2R)-1-methylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— 6-N-methyl-4-N-[4-[(2S)-1-methylpyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C14H19N7
6-N-methyl-4-N-[4-[(2S)-1-methylpyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 5-(3-chlorophenyl)-4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine —— C22H25ClN6
5-(3-chlorophenyl)-4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine
—— 4-[(2R)-1-propan-2-ylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C16H22N6
4-[(2R)-1-propan-2-ylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— N-(5-methylpyridin-2-yl)-4-[(2R)-1-propan-2-ylpyrrolidin-2-yl]pyrimidin-2-amine —— C17H23N5
N-(5-methylpyridin-2-yl)-4-[(2R)-1-propan-2-ylpyrrolidin-2-yl]pyrimidin-2-amine
—— 4-[2-amino-4-[(2S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]pyrimidin-5-yl]benzamide —— C25H26FN5O2
4-[2-amino-4-[(2S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H25FN4O
1-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— N-[2-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]methanesulfonamide —— C18H22ClN5O3S
N-[2-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]methanesulfonamide
—— 5-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H22F2N4O2
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— [(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20FN5OS
[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone —— C22H28FN5O
[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone
—— [(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C20H21FN6O
[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— [(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylimidazol-2-yl)methanone —— C21H21F3N6O
[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylimidazol-2-yl)methanone
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H22ClFN4O2
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 5-(3-fluorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C19H21FN6O2S
5-(3-fluorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 5-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H22F2N4O2
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 5-(3-methoxyphenyl)-4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine —— C23H28N6O
5-(3-methoxyphenyl)-4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H22F2N4O2
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— [(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone —— C22H28ClN5O
[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone
—— 5-(4-chlorophenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C19H21ClN6O2S
5-(4-chlorophenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone —— C23H22ClFN4O
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24ClFN4O
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— [(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C21H24N6O2
[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 5-(3-methoxyphenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C20H24N6O3S
5-(3-methoxyphenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24F2N4O
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine —— C20H22FN5O3S
4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine
—— 4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]-5-phenylpyrimidin-2-amine —— C20H23N5O3S
4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]-5-phenylpyrimidin-2-amine
—— 5-(3-chlorophenyl)-4-[(2S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine —— C22H25ClN6
5-(3-chlorophenyl)-4-[(2S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone —— C22H28ClN5O
[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone
—— 1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenoxypropan-1-one —— C25H28N4O3
1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenoxypropan-1-one
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24F2N4O
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 5-(3-methoxyphenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C20H24N6O3S
5-(3-methoxyphenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone —— C22H28FN5O
[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone
—— 5-(3-chlorophenyl)-4-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine —— C20H22ClN5O3S
5-(3-chlorophenyl)-4-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine
—— 5-(3-chlorophenyl)-4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine —— C20H22ClN5O3S
5-(3-chlorophenyl)-4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24ClFN4O
1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— [(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone —— C21H25ClN4O
[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone
—— [(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C20H22N6O
[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 5-(3-fluorophenyl)-4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine —— C22H25FN6
5-(3-fluorophenyl)-4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24F2N4O
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 5-(4-chlorophenyl)-4-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine —— C20H22ClN5O3S
5-(4-chlorophenyl)-4-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone —— C20H24F3N5O
1-[(2S)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
—— 5-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C23H25N5O3
5-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one