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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R,6R)-4-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)-2,6-dimethylmorpholine —— C25H29N5O
(2R,6R)-4-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)-2,6-dimethylmorpholine
—— N-cycloheptyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C22H26N4O3S
N-cycloheptyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-[(1R,2R)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C22H26N4O3S
N-[(1R,2R)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-cyclopentyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C20H22N4O3S
N-cyclopentyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N'-ethyl-N'-[7-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-N,N-dimethylethane-1,2-diamine —— C26H34N6O
N'-ethyl-N'-[7-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-N,N-dimethylethane-1,2-diamine
—— 4-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]-5-pyrazin-2-ylpyrimidin-2-amine —— C18H20N6O2
4-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]-5-pyrazin-2-ylpyrimidin-2-amine
—— N-(2-methoxyethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C18H20N4O4S
N-(2-methoxyethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-[(1S,2R)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C22H26N4O3S
N-[(1S,2R)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine —— C19H22N6O3S
N-[(3R)-1,1-dioxothiolan-3-yl]-5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine
—— (2R)-2-N-[7-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-1-N,1-N-dimethylpropane-1,2-diamine —— C24H29FN6
(2R)-2-N-[7-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-1-N,1-N-dimethylpropane-1,2-diamine
—— N'-[7-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-N,N,N'-trimethylethane-1,2-diamine —— C24H29FN6
N'-[7-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-N,N,N'-trimethylethane-1,2-diamine
—— N-(3-methoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(3-methylthiophen-2-yl)pyrimidin-2-amine —— C17H20N4O2S
N-(3-methoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-(3-methylthiophen-2-yl)pyrimidin-2-amine
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-morpholin-4-ylethyl)pyrimidin-2-amine —— C21H27N7O2
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-morpholin-4-ylethyl)pyrimidin-2-amine
—— 4-(3,5-dimethyl-1,2-oxazol-4-yl)-5-pyrazin-2-yl-N-[(1S)-1-pyridin-3-ylethyl]pyrimidin-2-amine —— C20H19N7O
4-(3,5-dimethyl-1,2-oxazol-4-yl)-5-pyrazin-2-yl-N-[(1S)-1-pyridin-3-ylethyl]pyrimidin-2-amine
—— N-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)-N',N'-dimethylethane-1,2-diamine —— C23H28N6
N-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)-N',N'-dimethylethane-1,2-diamine
—— 5-(3-methyl-1,2-oxazol-5-yl)-N-(3-morpholin-4-ylpropyl)-4-thiophen-2-ylpyrimidin-2-amine —— C19H23N5O2S
5-(3-methyl-1,2-oxazol-5-yl)-N-(3-morpholin-4-ylpropyl)-4-thiophen-2-ylpyrimidin-2-amine
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-(2-phenylethyl)acetamide —— C23H22N4O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-(2-phenylethyl)acetamide
—— (2S,6R)-4-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)-2,6-dimethylmorpholine —— C25H29N5O
(2S,6R)-4-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)-2,6-dimethylmorpholine
—— 1-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)piperidine-4-carboxamide —— C25H28N6O
1-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)piperidine-4-carboxamide
—— N-[(1R,2S)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C22H26N4O3S
N-[(1R,2S)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-tert-butyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C19H22N4O3S
N-tert-butyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-cyclopropyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C18H18N4O3S
N-cyclopropyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-[3-(2-methylimidazol-1-yl)propyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-thiophen-2-ylpyrimidin-2-amine —— C19H20N6OS
N-[3-(2-methylimidazol-1-yl)propyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-thiophen-2-ylpyrimidin-2-amine
—— N-[(1S,2S)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C22H26N4O3S
N-[(1S,2S)-2-methylcyclohexyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— 2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C20H18N4O3S
2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— 7-[(4-fluorophenyl)methyl]-N-(3-propan-2-yloxypropyl)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C25H30FN5O
7-[(4-fluorophenyl)methyl]-N-(3-propan-2-yloxypropyl)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— N-[4-(furan-3-yl)-5-pyridin-4-ylpyrimidin-2-yl]-N',N'-dimethylethane-1,2-diamine —— C17H19N5O
N-[4-(furan-3-yl)-5-pyridin-4-ylpyrimidin-2-yl]-N',N'-dimethylethane-1,2-diamine
—— N-(4-methylcyclohexyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide —— C22H26N4O3S
N-(4-methylcyclohexyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]acetamide
—— N-(3-ethenoxypropyl)-5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine —— C20H24N6O2
N-(3-ethenoxypropyl)-5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylthiophen-2-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine —— C19H17N5OS
5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylthiophen-2-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
—— 4-(furan-3-yl)-N-(2-pyrazin-2-ylethyl)-5-pyridin-4-ylpyrimidin-2-amine —— C19H16N6O
4-(furan-3-yl)-N-(2-pyrazin-2-ylethyl)-5-pyridin-4-ylpyrimidin-2-amine
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-propylacetamide —— C18H20N4O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-propylacetamide
—— N-[(2S)-1-methoxypropan-2-yl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine —— C21H26N6O3
N-[(2S)-1-methoxypropan-2-yl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-[(3R)-3-methylpiperidin-1-yl]ethyl]acetamide —— C22H27N5O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-[(3R)-3-methylpiperidin-1-yl]ethyl]acetamide
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]acetamide —— C22H27N5O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]acetamide
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[(1R)-1-thiophen-2-ylethyl]acetamide —— C20H18N4O3S2
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[(1R)-1-thiophen-2-ylethyl]acetamide
—— 5-[2-(Azepan-1-yl)-4-(2-methylpyridin-3-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole —— C20H23N5O
5-[2-(Azepan-1-yl)-4-(2-methylpyridin-3-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole
—— 2-[2-[4-(2-Methoxyethyl)piperazin-1-yl]-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C21H25N5O4S
2-[2-[4-(2-Methoxyethyl)piperazin-1-yl]-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— N-[(4-methoxyphenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-methylpyridin-3-yl)pyrimidin-2-amine —— C22H21N5O2
N-[(4-methoxyphenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-methylpyridin-3-yl)pyrimidin-2-amine
—— 2-[2-[(8aS)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C21H23N5O3S
2-[2-[(8aS)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— N-[(2R)-5-methylhexan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C21H26N4O3S
N-[(2R)-5-methylhexan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-(4-methylpiperidin-1-yl)ethyl]acetamide —— C22H27N5O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-(4-methylpiperidin-1-yl)ethyl]acetamide
—— N-[(3R)-3-(furan-2-yl)butyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C22H22N4O4S
N-[(3R)-3-(furan-2-yl)butyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 3-methyl-5-[2-[(3S)-3-methylpiperidin-1-yl]-4-(6-methylpyridin-3-yl)pyrimidin-5-yl]-1,2-oxazole —— C20H23N5O
3-methyl-5-[2-[(3S)-3-methylpiperidin-1-yl]-4-(6-methylpyridin-3-yl)pyrimidin-5-yl]-1,2-oxazole
—— N-[(2S)-5-methylhexan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C21H26N4O3S
N-[(2S)-5-methylhexan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 2-[2-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C21H23N5O3S
2-[2-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— N-[2-(furan-2-yl)ethyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C20H18N4O4S
N-[2-(furan-2-yl)ethyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— [4-(4-Ethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C21H28N6O2
[4-(4-Ethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-(5-methylpyrazol-1-yl)ethyl]acetamide —— C20H20N6O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[2-(5-methylpyrazol-1-yl)ethyl]acetamide
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-(2-pyrrolidin-1-ylethyl)acetamide —— C20H23N5O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-(2-pyrrolidin-1-ylethyl)acetamide