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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)morpholine-2-carboxamide —— C21H29N5O2
(2R)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)morpholine-2-carboxamide
—— (5-methylpyrazin-2-yl)-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C19H27N7O
(5-methylpyrazin-2-yl)-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (3S)-1-(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)piperidine-3-carboxamide —— C20H23N5O
(3S)-1-(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)piperidine-3-carboxamide
—— (3R)-1-[2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrimidin-4-yl]piperidin-3-ol —— C21H26N6O
(3R)-1-[2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrimidin-4-yl]piperidin-3-ol
—— (2R)-2-[[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]hexanamide —— C18H20FN5O
(2R)-2-[[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]hexanamide
—— (2S)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)morpholine-2-carboxamide —— C21H29N5O2
(2S)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)morpholine-2-carboxamide
—— N-[(3R)-1-(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)pyrrolidin-3-yl]acetamide —— C17H19N7O
N-[(3R)-1-(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)pyrrolidin-3-yl]acetamide
—— (3R)-1-(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)piperidine-3-carboxamide —— C20H23N5O
(3R)-1-(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)piperidine-3-carboxamide
—— N-(2-imidazol-1-ylethyl)-5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine —— C15H22N6O2S
N-(2-imidazol-1-ylethyl)-5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine
—— (3R)-1-[3-[(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]propyl]piperidin-3-ol —— C20H25N5O
(3R)-1-[3-[(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]propyl]piperidin-3-ol
—— N-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-2-(5-methyl-2,4-dioxopyrimidin-1-yl)acetamide —— C19H30N4O3
N-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-2-(5-methyl-2,4-dioxopyrimidin-1-yl)acetamide
—— (5-methylpyrazin-2-yl)-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C19H27N7O
(5-methylpyrazin-2-yl)-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (2-anilinopyrimidin-5-yl)-[(3S)-3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methanone —— C18H23N5O2
(2-anilinopyrimidin-5-yl)-[(3S)-3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methanone
—— 1,3-dimethyl-N-[(1S)-2-methyl-1-pyridin-2-ylpropyl]-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C21H23N7
1,3-dimethyl-N-[(1S)-2-methyl-1-pyridin-2-ylpropyl]-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— (3S)-1-[3-[(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]propyl]piperidin-3-ol —— C20H25N5O
(3S)-1-[3-[(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]propyl]piperidin-3-ol
—— N-(2-imidazol-1-ylethyl)-5-methylsulfonyl-4-[(3R)-piperidin-3-yl]pyrimidin-2-amine —— C15H22N6O2S
N-(2-imidazol-1-ylethyl)-5-methylsulfonyl-4-[(3R)-piperidin-3-yl]pyrimidin-2-amine
—— [(2S)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)morpholin-2-yl]methanamine —— C17H21N7O
[(2S)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)morpholin-2-yl]methanamine
—— 1,3-dimethyl-N-[(2S)-1-(6-methylpyridin-2-yl)propan-2-yl]-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C21H23N7
1,3-dimethyl-N-[(2S)-1-(6-methylpyridin-2-yl)propan-2-yl]-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— N-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-2-(5-methyl-2,4-dioxopyrimidin-1-yl)acetamide —— C19H30N4O3
N-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-2-(5-methyl-2,4-dioxopyrimidin-1-yl)acetamide
—— N-[[(1R)-3,4-dihydro-1H-isochromen-1-yl]methyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C21H20N6O
N-[[(1R)-3,4-dihydro-1H-isochromen-1-yl]methyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— [(2R)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)morpholin-2-yl]methanamine —— C17H21N7O
[(2R)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)morpholin-2-yl]methanamine
—— 1-methyl-6-pyridin-4-yl-N-[(3S)-thiolan-3-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C15H16N6S
1-methyl-6-pyridin-4-yl-N-[(3S)-thiolan-3-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 1,3-dimethyl-N-[(1R)-2-methyl-1-pyridin-2-ylpropyl]-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C21H23N7
1,3-dimethyl-N-[(1R)-2-methyl-1-pyridin-2-ylpropyl]-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— (3S)-3-[[methyl-[[2-(methylamino)pyrimidin-5-yl]methyl]amino]methyl]piperidin-3-ol —— C13H23N5O
(3S)-3-[[methyl-[[2-(methylamino)pyrimidin-5-yl]methyl]amino]methyl]piperidin-3-ol
—— (3R)-3-[[methyl-[[2-(methylamino)pyrimidin-5-yl]methyl]amino]methyl]piperidin-3-ol —— C13H23N5O
(3R)-3-[[methyl-[[2-(methylamino)pyrimidin-5-yl]methyl]amino]methyl]piperidin-3-ol
—— N-[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H19FN6O
N-[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— 5-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C17H18FN3O3
5-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— 4-[[(3S)-1-[2-(ethylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methyl]benzoic acid —— C19H22N4O3
4-[[(3S)-1-[2-(ethylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methyl]benzoic acid
—— 4-[[(3R)-1-[2-(ethylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methyl]benzoic acid —— C19H22N4O3
4-[[(3R)-1-[2-(ethylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methyl]benzoic acid
—— 5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C17H18FN3O3
5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— [6-[(3S)-3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl]pyrazin-2-yl]-piperidin-1-ylmethanone —— C23H29FN4O
[6-[(3S)-3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl]pyrazin-2-yl]-piperidin-1-ylmethanone
—— 1-methyl-6-pyridin-4-yl-N-[(3R)-thiolan-3-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C15H16N6S
1-methyl-6-pyridin-4-yl-N-[(3R)-thiolan-3-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— N-[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H19FN6O
N-[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— N-[[(1S)-3,4-dihydro-1H-isochromen-1-yl]methyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C21H20N6O
N-[[(1S)-3,4-dihydro-1H-isochromen-1-yl]methyl]-1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— 2-[(2R)-4-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)morpholin-2-yl]ethanamine —— C18H21N5O
2-[(2R)-4-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)morpholin-2-yl]ethanamine
—— 1,3-dimethyl-4-[(3R)-3-(propoxymethyl)pyrrolidin-1-yl]-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidine —— C20H26N6O
1,3-dimethyl-4-[(3R)-3-(propoxymethyl)pyrrolidin-1-yl]-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidine
—— 1-[(2R)-2-[[(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]morpholin-4-yl]ethanone —— C19H23N7O2
1-[(2R)-2-[[(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]morpholin-4-yl]ethanone
—— (1S)-3-[methyl-(1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]-1-phenylpropan-1-ol —— C21H22N6O
(1S)-3-[methyl-(1-methyl-6-pyridin-4-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]-1-phenylpropan-1-ol
—— N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine —— C20H25N5O
N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
—— N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine —— C20H25N5O
N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
—— 1-[(2S)-2-[[(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]morpholin-4-yl]ethanone —— C19H23N7O2
1-[(2S)-2-[[(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]morpholin-4-yl]ethanone
—— (3S)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)-3-methylpiperazin-2-one —— C17H19N7O
(3S)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)-3-methylpiperazin-2-one
—— 2-[(2S)-4-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)morpholin-2-yl]ethanol —— C19H25N5O2
2-[(2S)-4-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)morpholin-2-yl]ethanol
—— (3R)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)-3-methylpiperazin-2-one —— C17H19N7O
(3R)-4-(1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)-3-methylpiperazin-2-one
—— [6-[(3R)-3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl]pyrazin-2-yl]-piperidin-1-ylmethanone —— C23H29FN4O
[6-[(3R)-3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl]pyrazin-2-yl]-piperidin-1-ylmethanone
—— N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-amine —— C16H16N6O2S
N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-1,3-dimethyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-amine
—— 2-pyridin-4-yl-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine —— C18H22N8
2-pyridin-4-yl-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine
—— [(2R)-2-[2-(dimethylamino)ethyl]piperidin-1-yl]-(2-methylpyrimidin-5-yl)methanone —— C15H24N4O
[(2R)-2-[2-(dimethylamino)ethyl]piperidin-1-yl]-(2-methylpyrimidin-5-yl)methanone
—— 2-pyridin-4-yl-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine —— C18H22N8
2-pyridin-4-yl-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine
—— (2S)-N-phenyl-4-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]morpholine-2-carboxamide —— C21H21N5O2
(2S)-N-phenyl-4-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]morpholine-2-carboxamide