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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(3S)-3-(furan-2-yl)butyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C22H22N4O4S
N-[(3S)-3-(furan-2-yl)butyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(3-methylthiophen-2-yl)-N-(3-morpholin-4-ylpropyl)pyrimidin-2-amine —— C20H25N5O2S
5-(3-methyl-1,2-oxazol-5-yl)-4-(3-methylthiophen-2-yl)-N-(3-morpholin-4-ylpropyl)pyrimidin-2-amine
—— [4-(4,5-Dimethyl-6-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C21H28N6O
[4-(4,5-Dimethyl-6-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— N-[2-(dimethylamino)ethyl]-N-ethyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C20H25N5O3S
N-[2-(dimethylamino)ethyl]-N-ethyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N-(2,2-dimethoxyethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C18H20N4O5S
N-(2,2-dimethoxyethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C21H27N5O3S
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N-[(3-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine —— C21H18FN5O
N-[(3-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(2-methylpyridin-3-yl)pyrimidin-2-amine
—— [4-(4-Methyl-6-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-1-yl]-pyrazin-2-ylmethanone —— C19H24N6O
[4-(4-Methyl-6-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-1-yl]-pyrazin-2-ylmethanone
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-(2-thiophen-2-ylethyl)acetamide —— C20H18N4O3S2
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-(2-thiophen-2-ylethyl)acetamide
—— (2R)-N-(furan-2-ylmethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]propanamide —— C20H18N4O4S
(2R)-N-(furan-2-ylmethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]propanamide
—— [4-(4,5-Dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C21H28N6O2
[4-(4,5-Dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— N-[(2R)-1-methoxypropan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C18H20N4O4S
N-[(2R)-1-methoxypropan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 2-[4-(3-Methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C14H12N4O3S
2-[4-(3-Methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 1-[5-(3-Methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperidine-4-carboxamide —— C23H27N7O3
1-[5-(3-Methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperidine-4-carboxamide
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-morpholin-4-yl-2-oxoethyl)-6-thiophen-2-ylpyridazin-3-one —— C18H18N4O4S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-morpholin-4-yl-2-oxoethyl)-6-thiophen-2-ylpyridazin-3-one
—— N-[(2S)-1-methoxypropan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C18H20N4O4S
N-[(2S)-1-methoxypropan-2-yl]-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N,N-diethyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C18H20N4O3S
N,N-diethyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N-(furan-2-ylmethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C19H16N4O4S
N-(furan-2-ylmethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N-(2-methylbutan-2-yl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C19H22N4O3S
N-(2-methylbutan-2-yl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N-(2-methoxyethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C17H18N4O4S
N-(2-methoxyethyl)-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-piperidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one —— C19H22N4O2S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-piperidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine —— C23H23N7O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
—— 2-[(2-Chloro-6-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C19H13ClFN3O2S
2-[(2-Chloro-6-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N,N-di(propan-2-yl)acetamide —— C20H24N4O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N,N-di(propan-2-yl)acetamide
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-(thiophen-2-ylmethyl)acetamide —— C19H16N4O3S2
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-(thiophen-2-ylmethyl)acetamide
—— 2-[(4-Fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C19H14FN3O2S
2-[(4-Fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-propan-2-ylacetamide —— C17H18N4O3S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-propan-2-ylacetamide
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-[(2-methylphenyl)methyl]-6-thiophen-2-ylpyridazin-3-one —— C20H17N3O2S
5-(3-Methyl-1,2-oxazol-5-yl)-2-[(2-methylphenyl)methyl]-6-thiophen-2-ylpyridazin-3-one
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C19H20N4O4S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-cyclopropyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C17H16N4O3S
N-cyclopropyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-[(1S)-1-phenylethyl]pyrimidin-2-amine —— C25H26N6O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-[(1S)-1-phenylethyl]pyrimidin-2-amine
—— (3R)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol —— C22H26N6O3
(3R)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol
—— 2-(3,3-Dimethyl-2-oxobutyl)-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C18H19N3O3S
2-(3,3-Dimethyl-2-oxobutyl)-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— N-cyclohexyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C20H22N4O3S
N-cyclohexyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— (3S)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol —— C22H26N6O3
(3S)-1-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-ol
—— N,N-dimethyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C16H16N4O3S
N,N-dimethyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— 2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C19H20N4O4S
2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(2-Chloro-4-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C19H13ClFN3O2S
2-[(2-Chloro-4-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— N-cyclooctyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide —— C22H26N4O3S
N-cyclooctyl-2-[4-(3-methyl-1,2-oxazol-5-yl)-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
—— N',N'-dimethyl-N-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]propane-1,3-diamine —— C22H29N7O2
N',N'-dimethyl-N-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]propane-1,3-diamine
—— N-[(2-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine —— C24H23FN6O2
N-[(2-fluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine
—— N',N'-dimethyl-N-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]ethane-1,2-diamine —— C21H27N7O2
N',N'-dimethyl-N-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]ethane-1,2-diamine
—— 2-[(2,6-Difluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one —— C19H13F2N3O2S
2-[(2,6-Difluorophenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)-6-thiophen-2-ylpyridazin-3-one
—— N-benzyl-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine —— C24H24N6O2
N-benzyl-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine
—— N-cyclopentyl-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine —— C22H26N6O2
N-cyclopentyl-5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-amine
—— 4-[5-(3-Methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperazin-2-one —— C21H23N7O3
4-[5-(3-Methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]piperazin-2-one
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(pyridin-3-ylmethyl)-6-thiophen-2-ylpyridazin-3-one —— C18H14N4O2S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(pyridin-3-ylmethyl)-6-thiophen-2-ylpyridazin-3-one
—— 7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H26N6O
7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-(3-methoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-thiophen-2-ylpyrimidin-2-amine —— C16H18N4O2S
N-(3-methoxypropyl)-5-(3-methyl-1,2-oxazol-5-yl)-4-thiophen-2-ylpyrimidin-2-amine