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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2S)-1-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]propan-2-yl]cyclopropanecarboxamide —— C18H21N3O3
N-[(2S)-1-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]propan-2-yl]cyclopropanecarboxamide
—— 2-(benzotriazol-1-yl)-N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]acetamide —— C22H20F2N6O2
2-(benzotriazol-1-yl)-N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]acetamide
—— N-[(2S)-1-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]propan-2-yl]-5-methylpyrazine-2-carboxamide —— C20H21N5O3
N-[(2S)-1-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]propan-2-yl]-5-methylpyrazine-2-carboxamide
—— 2-[(2S)-2-amino-3-methylbutyl]-6-(3,4-difluorophenyl)pyridazin-3-one —— C15H17F2N3O
2-[(2S)-2-amino-3-methylbutyl]-6-(3,4-difluorophenyl)pyridazin-3-one
—— N-[(2S)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]-3-methylbutan-2-yl]-1-ethylpyrazole-4-carboxamide —— C21H23F2N5O2
N-[(2S)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]-3-methylbutan-2-yl]-1-ethylpyrazole-4-carboxamide
—— N-[(2S)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]-3-methylbutan-2-yl]-1,3-dimethylpyrazole-4-carboxamide —— C21H23F2N5O2
N-[(2S)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]-3-methylbutan-2-yl]-1,3-dimethylpyrazole-4-carboxamide
—— N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]-1,2-thiazole-4-carboxamide —— C18H16F2N4O2S
N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]-1,2-thiazole-4-carboxamide
—— N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H18F2N6O2
N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— ethyl (4R)-4-ethyl-6-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H23N5O3S
ethyl (4R)-4-ethyl-6-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-ethyl-6-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H23N5O3S
ethyl (4S)-4-ethyl-6-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (2R,6R)-2,6-dimethyl-4-[4-(4-methylphenyl)quinazolin-2-yl]morpholine —— C21H23N3O
(2R,6R)-2,6-dimethyl-4-[4-(4-methylphenyl)quinazolin-2-yl]morpholine
—— [4-(4-fluorophenyl)-2-[methyl(methylsulfonyl)amino]-6-propan-2-ylpyrimidin-5-yl] (3R,5S)-3,5-dihydroxyhept-6-enoate —— C22H28FN3O6S
[4-(4-fluorophenyl)-2-[methyl(methylsulfonyl)amino]-6-propan-2-ylpyrimidin-5-yl] (3R,5S)-3,5-dihydroxyhept-6-enoate
—— N-[(2-chloro-6-fluorophenyl)methyl]-N,1,3-trimethyl-2,4-dioxopyrimidine-5-sulfonamide —— C14H15ClFN3O4S
N-[(2-chloro-6-fluorophenyl)methyl]-N,1,3-trimethyl-2,4-dioxopyrimidine-5-sulfonamide
—— (2S,6S)-2,6-dimethyl-4-[4-(4-methylphenyl)quinazolin-2-yl]morpholine —— C21H23N3O
(2S,6S)-2,6-dimethyl-4-[4-(4-methylphenyl)quinazolin-2-yl]morpholine
—— (2R,6S)-2,6-dimethyl-4-[4-(4-methylphenyl)quinazolin-2-yl]morpholine —— C21H23N3O
(2R,6S)-2,6-dimethyl-4-[4-(4-methylphenyl)quinazolin-2-yl]morpholine
—— 1,3-dimethyl-2,4-dioxo-N-[(2S)-4-phenylbutan-2-yl]pyrimidine-5-sulfonamide —— C16H21N3O4S
1,3-dimethyl-2,4-dioxo-N-[(2S)-4-phenylbutan-2-yl]pyrimidine-5-sulfonamide
—— 1,3-dimethyl-2,4-dioxo-N-[(2R)-4-phenylbutan-2-yl]pyrimidine-5-sulfonamide —— C16H21N3O4S
1,3-dimethyl-2,4-dioxo-N-[(2R)-4-phenylbutan-2-yl]pyrimidine-5-sulfonamide
—— ethyl (4S)-6-[[(2-fluorophenyl)methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H22FN3O3
ethyl (4S)-6-[[(2-fluorophenyl)methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(2-fluorophenyl)methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H22FN3O3
ethyl (4R)-6-[[(2-fluorophenyl)methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (1R)-N-(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-N-(2-methoxyethyl)cyclohex-3-ene-1-carboxamide —— C21H26N4O4
(1R)-N-(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-N-(2-methoxyethyl)cyclohex-3-ene-1-carboxamide
—— [(2R)-1-(tert-butylamino)-1-oxopropan-2-yl] 3-amino-6-bromopyrazine-2-carboxylate —— C12H17BrN4O3
[(2R)-1-(tert-butylamino)-1-oxopropan-2-yl] 3-amino-6-bromopyrazine-2-carboxylate
—— (3S)-1-propan-2-yl-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]pyrrolidine-2,5-dione —— C17H16F3N5O2
(3S)-1-propan-2-yl-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]pyrrolidine-2,5-dione
—— 6-methoxy-5-[[2-[(2R)-oxolan-2-yl]ethylamino]methyl]pyrimidin-4-amine —— C12H20N4O2
6-methoxy-5-[[2-[(2R)-oxolan-2-yl]ethylamino]methyl]pyrimidin-4-amine
—— [(2S)-1-(tert-butylamino)-1-oxopropan-2-yl] 3-amino-6-bromopyrazine-2-carboxylate —— C12H17BrN4O3
[(2S)-1-(tert-butylamino)-1-oxopropan-2-yl] 3-amino-6-bromopyrazine-2-carboxylate
—— 6-methoxy-5-[[2-[(2S)-oxolan-2-yl]ethylamino]methyl]pyrimidin-4-amine —— C12H20N4O2
6-methoxy-5-[[2-[(2S)-oxolan-2-yl]ethylamino]methyl]pyrimidin-4-amine
—— N-[(1R,6S)-7-bicyclo[4.1.0]heptanyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C18H19N5
N-[(1R,6S)-7-bicyclo[4.1.0]heptanyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 6-amino-1-(2-methylpropyl)-5-[(R)-(5-methylthiophen-2-yl)-morpholin-4-ylmethyl]pyrimidine-2,4-dione —— C18H26N4O3S
6-amino-1-(2-methylpropyl)-5-[(R)-(5-methylthiophen-2-yl)-morpholin-4-ylmethyl]pyrimidine-2,4-dione
—— 6-amino-1-(2-methylpropyl)-5-[(S)-(5-methylthiophen-2-yl)-morpholin-4-ylmethyl]pyrimidine-2,4-dione —— C18H26N4O3S
6-amino-1-(2-methylpropyl)-5-[(S)-(5-methylthiophen-2-yl)-morpholin-4-ylmethyl]pyrimidine-2,4-dione
—— 6-amino-5-[(R)-(4-methylphenyl)-morpholin-4-ylmethyl]-1-(2-methylpropyl)pyrimidine-2,4-dione —— C20H28N4O3
6-amino-5-[(R)-(4-methylphenyl)-morpholin-4-ylmethyl]-1-(2-methylpropyl)pyrimidine-2,4-dione
—— 6-amino-5-[(S)-(4-methylphenyl)-morpholin-4-ium-4-ylmethyl]-1-(2-methylpropyl)pyrimidine-2,4-dione —— C20H29N4O3+
6-amino-5-[(S)-(4-methylphenyl)-morpholin-4-ium-4-ylmethyl]-1-(2-methylpropyl)pyrimidine-2,4-dione
—— N-benzyl-N-(furan-2-ylmethyl)-5-methylpyrazine-2-carboxamide —— C18H17N3O2
N-benzyl-N-(furan-2-ylmethyl)-5-methylpyrazine-2-carboxamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-prop-2-enyl-N-(thiophen-2-ylmethyl)acetamide —— C18H18N4O3S
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-prop-2-enyl-N-(thiophen-2-ylmethyl)acetamide
—— N-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-4-pyrazol-1-ylpyrimidin-2-amine —— C15H17N5O2
N-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-4-pyrazol-1-ylpyrimidin-2-amine
—— 5-[4-[[(2R)-oxolan-2-yl]methyl]piperazine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C14H20N4O4
5-[4-[[(2R)-oxolan-2-yl]methyl]piperazine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-bromo-N-[(1S)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]pyrimidin-2-amine —— C12H14BrN3O2
5-bromo-N-[(1S)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]pyrimidin-2-amine
—— (1R)-N,N-dimethyl-N'-(tetrazolo[1,5-a]pyrazin-8-yl)-1-thiophen-2-ylethane-1,2-diamine —— C12H15N7S
(1R)-N,N-dimethyl-N'-(tetrazolo[1,5-a]pyrazin-8-yl)-1-thiophen-2-ylethane-1,2-diamine
—— N-[(1S)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-4-pyrazol-1-ylpyrimidin-2-amine —— C15H17N5O2
N-[(1S)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-4-pyrazol-1-ylpyrimidin-2-amine
—— 6-chloro-N-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-2-methylpyrimidin-4-amine —— C13H16ClN3O2
6-chloro-N-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-2-methylpyrimidin-4-amine
—— morpholin-4-yl-[(2S)-1-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]piperidin-2-yl]methanone —— C20H22F3N5O2
morpholin-4-yl-[(2S)-1-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]piperidin-2-yl]methanone
—— 5-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-4-ium-1-carbonyl]-1H-pyrimidine-2,4-dione —— C14H21N4O4+
5-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-4-ium-1-carbonyl]-1H-pyrimidine-2,4-dione
—— [(2R)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)piperidin-2-yl]-morpholin-4-ylmethanone —— C20H25N5O2
[(2R)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)piperidin-2-yl]-morpholin-4-ylmethanone
—— 5-bromo-N-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]pyrimidin-2-amine —— C12H14BrN3O2
5-bromo-N-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]pyrimidin-2-amine
—— [(2S)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)piperidin-2-yl]-morpholin-4-ylmethanone —— C20H25N5O2
[(2S)-1-(6-methyl-2-pyridin-2-ylpyrimidin-4-yl)piperidin-2-yl]-morpholin-4-ylmethanone
—— 6-chloro-N-[(1S)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-2-methylpyrimidin-4-amine —— C13H16ClN3O2
6-chloro-N-[(1S)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-2-methylpyrimidin-4-amine
—— 5-chloro-N-[(2R,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2R,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— 5-chloro-N-[(2S,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2S,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— 5-chloro-N-[(2S,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2S,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— N-[[(2R)-1-(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-2-yl]methyl]benzamide —— C24H24N6O
N-[[(2R)-1-(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-2-yl]methyl]benzamide
—— 5-chloro-N-[(2R,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2R,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— N-[[(2S)-1-(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-2-yl]methyl]benzamide —— C24H24N6O
N-[[(2S)-1-(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-2-yl]methyl]benzamide