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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(2S)-2-[2-methyl-6-[(4-methylthiadiazol-5-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C15H20N6O2S
1-[(2S)-2-[2-methyl-6-[(4-methylthiadiazol-5-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— [(6S)-6-[[5-(dimethylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-pyrazin-2-ylmethanone —— C17H22N6O2
[(6S)-6-[[5-(dimethylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-pyrazin-2-ylmethanone
—— [(6R)-6-[(5-methylpyrazin-2-yl)methyl]-1,4-oxazepan-4-yl]-pyrimidin-5-ylmethanone —— C16H19N5O2
[(6R)-6-[(5-methylpyrazin-2-yl)methyl]-1,4-oxazepan-4-yl]-pyrimidin-5-ylmethanone
—— 1-[(2S)-2-[2-methyl-6-[2-(5-methylpyrazol-1-yl)ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C17H24N6O2
1-[(2S)-2-[2-methyl-6-[2-(5-methylpyrazol-1-yl)ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C17H26N6O2
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-(5-methylpyrazol-1-yl)ethyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine —— C15H22N6O
2-methyl-N-[2-(5-methylpyrazol-1-yl)ethyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-6-[(2R)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C13H18N6O2
2-methyl-6-[(2R)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C17H26N6O2
N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C17H26N6O2
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2S)-4-[(4-methyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C15H21N5OS
N,2-dimethyl-6-[(2S)-4-[(4-methyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-[2-methyl-6-[2-[(S)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C14H22N4O3S
1-[(2R)-2-[2-methyl-6-[2-[(S)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— 1-[(2R)-2-[2-methyl-6-[(5-methyl-1,2,4-oxadiazol-3-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C15H20N6O3
1-[(2R)-2-[2-methyl-6-[(5-methyl-1,2,4-oxadiazol-3-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C16H24N6O3
N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2R)-4-methylmorpholin-2-yl]pyrimidin-4-amine —— C16H23N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2R)-4-methylmorpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine —— C12H20N4O2S
2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-[6-[(5-ethyl-1,2,4-oxadiazol-3-yl)methylamino]-2-methylpyrimidin-4-yl]morpholin-4-yl]ethanone —— C16H22N6O3
1-[(2R)-2-[6-[(5-ethyl-1,2,4-oxadiazol-3-yl)methylamino]-2-methylpyrimidin-4-yl]morpholin-4-yl]ethanone
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine —— C15H21N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C15H26N4O2S
2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2S)-4-methylmorpholin-2-yl]pyrimidin-4-amine —— C16H23N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2S)-4-methylmorpholin-2-yl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2S)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C15H21N5O2
N,2-dimethyl-6-[(2S)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine —— C14H20N6O2
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrimidin-4-amine —— C16H23N5OS
2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrimidin-4-amine
—— N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C17H25N5O3
N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-6-[(2S)-4-methylmorpholin-2-yl]-N-[2-(5-methylpyrazol-1-yl)ethyl]pyrimidin-4-amine —— C16H24N6O
2-methyl-6-[(2S)-4-methylmorpholin-2-yl]-N-[2-(5-methylpyrazol-1-yl)ethyl]pyrimidin-4-amine
—— N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(1-methylimidazol-2-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C17H26N6O2
N-(2-methoxyethyl)-2-methyl-6-[(2S)-4-[(1-methylimidazol-2-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2S)-4-(1H-pyrazol-4-ylsulfonyl)morpholin-2-yl]pyrimidin-4-amine —— C13H18N6O3S
N,2-dimethyl-6-[(2S)-4-(1H-pyrazol-4-ylsulfonyl)morpholin-2-yl]pyrimidin-4-amine
—— N-cyclopentyl-2-methyl-6-[(2S)-4-(oxan-4-yl)morpholin-2-yl]pyrimidin-4-amine —— C19H30N4O2
N-cyclopentyl-2-methyl-6-[(2S)-4-(oxan-4-yl)morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine —— C12H20N4O2S
2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2S)-2-(6-amino-2-methylpyrimidin-4-yl)morpholin-4-yl]-2-pyrazol-1-ylethanone —— C14H18N6O2
1-[(2S)-2-(6-amino-2-methylpyrimidin-4-yl)morpholin-4-yl]-2-pyrazol-1-ylethanone
—— 1-[(2S)-2-[2-methyl-6-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C15H20N6O3
1-[(2S)-2-[2-methyl-6-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— 2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine —— C12H20N4O2S
2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-6-[(2R)-4-(1-methylimidazol-4-yl)sulfonylmorpholin-2-yl]pyrimidin-4-amine —— C13H18N6O3S
2-methyl-6-[(2R)-4-(1-methylimidazol-4-yl)sulfonylmorpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C15H26N4O2S
2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-[2-methyl-6-[2-(5-methylpyrazol-1-yl)ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C17H24N6O2
1-[(2R)-2-[2-methyl-6-[2-(5-methylpyrazol-1-yl)ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— 2-methyl-6-[(2S)-4-methylmorpholin-2-yl]-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrimidin-4-amine —— C16H23N5OS
2-methyl-6-[(2S)-4-methylmorpholin-2-yl]-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrimidin-4-amine
—— 2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-(5-methylpyrazol-1-yl)ethyl]pyrimidin-4-amine —— C16H24N6O
2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-(5-methylpyrazol-1-yl)ethyl]pyrimidin-4-amine
—— 1-[(2R)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]morpholin-4-yl]-2-pyrazol-1-ylethanone —— C15H20N6O2
1-[(2R)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]morpholin-4-yl]-2-pyrazol-1-ylethanone
—— N-(2-methoxyethyl)-2-methyl-6-[(2R)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C17H26N6O2
N-(2-methoxyethyl)-2-methyl-6-[(2R)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-[2-methyl-6-[2-[(R)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C14H22N4O3S
1-[(2R)-2-[2-methyl-6-[2-[(R)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— 2-methyl-N-[(4-methylthiadiazol-5-yl)methyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine —— C13H18N6OS
2-methyl-N-[(4-methylthiadiazol-5-yl)methyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C18H27N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[(4-methylthiadiazol-5-yl)methyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine —— C13H18N6OS
2-methyl-N-[(4-methylthiadiazol-5-yl)methyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C15H26N4O2S
2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— 1-[(2S)-2-[6-[(5-ethyl-1,2,4-oxadiazol-3-yl)methylamino]-2-methylpyrimidin-4-yl]morpholin-4-yl]ethanone —— C16H22N6O3
1-[(2S)-2-[6-[(5-ethyl-1,2,4-oxadiazol-3-yl)methylamino]-2-methylpyrimidin-4-yl]morpholin-4-yl]ethanone
—— 2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C15H26N4O2S
2-methyl-N-[2-[(R)-methylsulfinyl]ethyl]-6-[(2R)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-6-[(2R)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C14H20N6O
2-methyl-6-[(2R)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2S)-2-[2-methyl-6-(2-pyrazin-2-ylethylamino)pyrimidin-4-yl]morpholin-4-yl]ethanone —— C17H22N6O2
1-[(2S)-2-[2-methyl-6-(2-pyrazin-2-ylethylamino)pyrimidin-4-yl]morpholin-4-yl]ethanone
—— N,2-dimethyl-6-[(2S)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C15H21N5OS
N,2-dimethyl-6-[(2S)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2S)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]morpholin-4-yl]-2-pyrazol-1-ylethanone —— C15H20N6O2
1-[(2S)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]morpholin-4-yl]-2-pyrazol-1-ylethanone
—— 2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-[(S)-methylsulfinyl]ethyl]pyrimidin-4-amine —— C13H22N4O2S
2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-[(S)-methylsulfinyl]ethyl]pyrimidin-4-amine