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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(2R)-2-cyclopentylpyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H19N3O2S
6-[(2R)-2-cyclopentylpyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 3-amino-N-[(R)-(4-propylphenyl)-thiophen-2-ylmethyl]pyrazine-2-carboxamide —— C19H20N4OS
3-amino-N-[(R)-(4-propylphenyl)-thiophen-2-ylmethyl]pyrazine-2-carboxamide
—— 3-amino-N-[(S)-(4-propylphenyl)-thiophen-2-ylmethyl]pyrazine-2-carboxamide —— C19H20N4OS
3-amino-N-[(S)-(4-propylphenyl)-thiophen-2-ylmethyl]pyrazine-2-carboxamide
—— N-[(1S)-1-(1-adamantyl)ethyl]-3-aminopyrazine-2-carboxamide —— C17H24N4O
N-[(1S)-1-(1-adamantyl)ethyl]-3-aminopyrazine-2-carboxamide
—— 2-methylpropyl (4R)-4-(3,4-dichlorophenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H18Cl2N2O2S
2-methylpropyl (4R)-4-(3,4-dichlorophenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-ethyl-6-[(3-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H20N2O5S
ethyl (4R)-4-ethyl-6-[(3-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(1S)-1-(furan-2-yl)ethyl]-2-(4-methyl-6-oxo-2-pyridin-3-yl-1H-pyrimidin-5-yl)acetamide —— C18H18N4O3
N-[(1S)-1-(furan-2-yl)ethyl]-2-(4-methyl-6-oxo-2-pyridin-3-yl-1H-pyrimidin-5-yl)acetamide
—— [2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] 6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxylate —— C18H21N3O6S
[2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] 6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxylate
—— N-[(1R)-1-(furan-2-yl)ethyl]-2-(4-methyl-6-oxo-2-pyridin-3-yl-1H-pyrimidin-5-yl)acetamide —— C18H18N4O3
N-[(1R)-1-(furan-2-yl)ethyl]-2-(4-methyl-6-oxo-2-pyridin-3-yl-1H-pyrimidin-5-yl)acetamide
—— ethyl (4S)-4-ethyl-6-[(3-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H20N2O5S
ethyl (4S)-4-ethyl-6-[(3-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (1R)-N'-(6-chloropyrazin-2-yl)-N,N-dimethyl-1-phenylethane-1,2-diamine —— C14H17ClN4
(1R)-N'-(6-chloropyrazin-2-yl)-N,N-dimethyl-1-phenylethane-1,2-diamine
—— (5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2S)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone —— C17H20ClN5O
(5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2S)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone
—— (5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2R)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone —— C17H20ClN5O
(5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2R)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone
—— (5R)-N'-(4,6-dimethylpyrimidin-2-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carbohydrazide —— C16H17N5O2
(5R)-N'-(4,6-dimethylpyrimidin-2-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carbohydrazide
—— (5S)-N'-(4,6-dimethylpyrimidin-2-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carbohydrazide —— C16H17N5O2
(5S)-N'-(4,6-dimethylpyrimidin-2-yl)-3-phenyl-4,5-dihydro-1,2-oxazole-5-carbohydrazide
—— ethyl (4R)-4-ethyl-2-oxo-6-[(4-phenyl-1,3-thiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H21N3O3S2
ethyl (4R)-4-ethyl-2-oxo-6-[(4-phenyl-1,3-thiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 6-[[(2S)-2-[(4-fluorophenyl)methyl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H22FN3O2
6-[[(2S)-2-[(4-fluorophenyl)methyl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-cyclopropyl-2-[(2R)-2-hydroxy-2-phenylethyl]-4-(trifluoromethyl)pyridazin-3-one —— C16H15F3N2O2
6-cyclopropyl-2-[(2R)-2-hydroxy-2-phenylethyl]-4-(trifluoromethyl)pyridazin-3-one
—— 6-cyclopropyl-2-[(2S)-2-hydroxy-2-phenylethyl]-4-(trifluoromethyl)pyridazin-3-one —— C16H15F3N2O2
6-cyclopropyl-2-[(2S)-2-hydroxy-2-phenylethyl]-4-(trifluoromethyl)pyridazin-3-one
—— 6-[[cyclopropyl-[(1S)-1-(2-fluorophenyl)ethyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H22FN3O2
6-[[cyclopropyl-[(1S)-1-(2-fluorophenyl)ethyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-cyclopropyl-2-[(2S)-2-hydroxy-3-morpholin-4-ylpropyl]-4-(trifluoromethyl)pyridazin-3-one —— C15H20F3N3O3
6-cyclopropyl-2-[(2S)-2-hydroxy-3-morpholin-4-ylpropyl]-4-(trifluoromethyl)pyridazin-3-one
—— 6-[[cyclopropyl-[(1R)-1-(2-fluorophenyl)ethyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H22FN3O2
6-[[cyclopropyl-[(1R)-1-(2-fluorophenyl)ethyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-cyclopropyl-2-[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]-4-(trifluoromethyl)pyridazin-3-one —— C15H20F3N3O3
6-cyclopropyl-2-[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]-4-(trifluoromethyl)pyridazin-3-one
—— 6-cyclopropyl-2-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-4-(trifluoromethyl)pyridazin-3-one —— C16H14F4N2O2
6-cyclopropyl-2-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-4-(trifluoromethyl)pyridazin-3-one
—— [(3S)-1-(2-methylpyrimidine-4-carbonyl)piperidin-3-yl]-morpholin-4-ylmethanone —— C16H22N4O3
[(3S)-1-(2-methylpyrimidine-4-carbonyl)piperidin-3-yl]-morpholin-4-ylmethanone
—— 6-[[[(1R)-1-(2-chlorophenyl)ethyl]-cyclopropylamino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H22ClN3O2
6-[[[(1R)-1-(2-chlorophenyl)ethyl]-cyclopropylamino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-cyclopropyl-2-[(2R)-2-(2-fluorophenyl)-2-hydroxyethyl]-4-(trifluoromethyl)pyridazin-3-one —— C16H14F4N2O2
6-cyclopropyl-2-[(2R)-2-(2-fluorophenyl)-2-hydroxyethyl]-4-(trifluoromethyl)pyridazin-3-one
—— 6-[[[(1R)-2,2-dimethyl-1-thiophen-2-ylpropyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C16H23N3O2S
6-[[[(1R)-2,2-dimethyl-1-thiophen-2-ylpropyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 1,3-dimethyl-6-[[(3R)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C15H21N5O3
1,3-dimethyl-6-[[(3R)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— 1,3-dimethyl-6-[[(3S)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C15H21N5O3
1,3-dimethyl-6-[[(3S)-3-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— 6-[[[(1S)-1-(2-chlorophenyl)ethyl]-cyclopropylamino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H22ClN3O2
6-[[[(1S)-1-(2-chlorophenyl)ethyl]-cyclopropylamino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-cyclopropyl-2-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-4-(trifluoromethyl)pyridazin-3-one —— C16H14F4N2O2
6-cyclopropyl-2-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-4-(trifluoromethyl)pyridazin-3-one
—— 6-[[[(1S)-2,2-dimethyl-1-thiophen-2-ylpropyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C16H23N3O2S
6-[[[(1S)-2,2-dimethyl-1-thiophen-2-ylpropyl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— [(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone —— C15H21N3O
[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone
—— [(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone —— C15H21N3O
[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone
—— [(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone —— C15H21N3O
[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone
—— N-[(1S)-1-(4-fluorophenyl)ethyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C19H16FN5
N-[(1S)-1-(4-fluorophenyl)ethyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— [(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone —— C15H21N3O
[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-(2-methylpyrimidin-4-yl)methanone
—— ethyl (4R)-4-ethyl-2-oxo-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyloxymethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O5S
ethyl (4R)-4-ethyl-2-oxo-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyloxymethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-ethyl-2-oxo-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyloxymethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O5S
ethyl (4S)-4-ethyl-2-oxo-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyloxymethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— propan-2-yl (4R)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17F3N2O3S
propan-2-yl (4R)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-6-propyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17F3N2O3S
methyl (4R)-6-propyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4S)-6-propyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17F3N2O3S
methyl (4S)-6-propyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— propan-2-yl (4S)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17F3N2O3S
propan-2-yl (4S)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(R)-cyclopropyl-(4-methoxyphenyl)methyl]pyrazine-2-carboxamide —— C16H17N3O2
N-[(R)-cyclopropyl-(4-methoxyphenyl)methyl]pyrazine-2-carboxamide
—— N-[(S)-cyclopropyl-(4-methoxyphenyl)methyl]pyrazine-2-carboxamide —— C16H17N3O2
N-[(S)-cyclopropyl-(4-methoxyphenyl)methyl]pyrazine-2-carboxamide
—— 2-methylpropyl (4S)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H19F3N2O3S
2-methylpropyl (4S)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H15F3N2O3S
ethyl (4S)-6-methyl-2-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[(4R)-4-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]-4,5,6,7-tetrahydroindazol-1-yl]ethanol —— C14H16F3N5O
2-[(4R)-4-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]-4,5,6,7-tetrahydroindazol-1-yl]ethanol
—— ethyl (4S)-4-methyl-2-oxo-6-[(2,4,5-trichlorophenoxy)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H15Cl3N2O4
ethyl (4S)-4-methyl-2-oxo-6-[(2,4,5-trichlorophenoxy)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate