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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)acetamide —— C19H19FN6OS
2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)acetamide
—— [(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-phenylmethanone —— C22H22N4O2
[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-phenylmethanone
—— 5-(4-chlorophenyl)-4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H20ClN5
5-(4-chlorophenyl)-4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone —— C22H21ClN4O2
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone
—— 3-[4-[(2S)-1-acetylpyrrolidin-2-yl]-2-aminopyrimidin-5-yl]benzamide —— C17H19N5O2
3-[4-[(2S)-1-acetylpyrrolidin-2-yl]-2-aminopyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone —— C18H22N4O3
1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone
—— 4-[(2R)-1-benzylsulfonylpyrrolidin-2-yl]-5-(4-chlorophenyl)pyrimidin-2-amine —— C21H21ClN4O2S
4-[(2R)-1-benzylsulfonylpyrrolidin-2-yl]-5-(4-chlorophenyl)pyrimidin-2-amine
—— 2-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-1-pyrrolidin-1-ylethanone —— C20H24FN5O
2-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-1-pyrrolidin-1-ylethanone
—— [(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone —— C21H18F2N4O
[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone
—— 1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone —— C23H24N4O3
1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone
—— 5-(4-chlorophenyl)-4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine —— C20H18ClFN4O2S
5-(4-chlorophenyl)-4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone —— C22H21FN4O
1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C24H25FN4O2
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone —— C18H21FN4O2
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone
—— 5-(4-methoxyphenyl)-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C21H23N5O
5-(4-methoxyphenyl)-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-dimethylacetamide —— C18H22FN5O
2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-dimethylacetamide
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one —— C23H23FN4O
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one
—— 5-(3-methoxyphenyl)-4-[(2S)-1-pyrazin-2-ylpyrrolidin-2-yl]pyrimidin-2-amine —— C19H20N6O
5-(3-methoxyphenyl)-4-[(2S)-1-pyrazin-2-ylpyrrolidin-2-yl]pyrimidin-2-amine
—— 3-[2-amino-4-[(2R)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C24H25N5O2
3-[2-amino-4-[(2R)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— 5-(4-methoxyphenyl)-4-[(2S)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine —— C22H24N4O4S
5-(4-methoxyphenyl)-4-[(2S)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine
—— 2-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]ethanol —— C17H22N4O
2-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]ethanol
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone —— C21H20FN5O
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone —— C18H21FN4O2
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone
—— 1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone —— C23H24N4O2
1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone
—— (2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C16H20FN5O2S
(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— 5-(4-methoxyphenyl)-4-[(2R)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine —— C22H24N4O4S
5-(4-methoxyphenyl)-4-[(2R)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine
—— 2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-methoxyphenyl)acetamide —— C23H24FN5O2
2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-methoxyphenyl)acetamide
—— 2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-dimethylacetamide —— C18H22FN5O
2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-dimethylacetamide
—— 1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone —— C17H19FN4O2
1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone
—— 2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide —— C20H26ClN5O
2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide
—— [(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-2-ylmethanone —— C21H18F3N5O
[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-2-ylmethanone
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone —— C22H21FN4O
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone
—— [(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C20H18FN5O
[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— [(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-phenylmethanone —— C21H19FN4O
[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-phenylmethanone
—— [(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone —— C22H21FN4O2
[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone
—— 5-(3-fluorophenyl)-4-[(2R)-1-(2-phenylethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C22H23FN4
5-(3-fluorophenyl)-4-[(2R)-1-(2-phenylethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 5-(4-methoxyphenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C21H23N5O
5-(4-methoxyphenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]-5-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine —— C21H20F3N5
4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]-5-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine
—— 5-(3-fluorophenyl)-4-[(2S)-1-methylsulfonylpyrrolidin-2-yl]pyrimidin-2-amine —— C15H17FN4O2S
5-(3-fluorophenyl)-4-[(2S)-1-methylsulfonylpyrrolidin-2-yl]pyrimidin-2-amine
—— 3-[2-amino-4-[(2S)-1-benzoylpyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C22H21N5O2
3-[2-amino-4-[(2S)-1-benzoylpyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— 5-(4-methoxyphenyl)-4-[(2R)-1-methylpyrrolidin-2-yl]pyrimidin-2-amine —— C16H20N4O
5-(4-methoxyphenyl)-4-[(2R)-1-methylpyrrolidin-2-yl]pyrimidin-2-amine
—— 5-(4-fluorophenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H20FN5
5-(4-fluorophenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 3-[2-amino-4-[(2R)-1-benzoylpyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C22H21N5O2
3-[2-amino-4-[(2R)-1-benzoylpyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone —— C22H21ClN4O2
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanone —— C16H17ClN4O
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanone
—— [(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone —— C21H18ClFN4O
[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone
—— 2-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide —— C20H26ClN5O
2-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone —— C21H20ClN5O
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone
—— 2-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide —— C20H26FN5O
2-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide
—— 5-(3-fluorophenyl)-4-[(2R)-1-methylsulfonylpyrrolidin-2-yl]pyrimidin-2-amine —— C15H17FN4O2S
5-(3-fluorophenyl)-4-[(2R)-1-methylsulfonylpyrrolidin-2-yl]pyrimidin-2-amine