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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R)-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butanamide —— C14H14F3N5O
(3R)-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butanamide
—— ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H26N2O4S
ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— N-[(1R,3R)-3-ethoxyspiro[3.5]nonan-1-yl]tetrazolo[1,5-b]pyridazin-6-amine —— C15H22N6O
N-[(1R,3R)-3-ethoxyspiro[3.5]nonan-1-yl]tetrazolo[1,5-b]pyridazin-6-amine
—— N-[(1R,3S)-3-ethoxyspiro[3.5]nonan-1-yl]tetrazolo[1,5-b]pyridazin-6-amine —— C15H22N6O
N-[(1R,3S)-3-ethoxyspiro[3.5]nonan-1-yl]tetrazolo[1,5-b]pyridazin-6-amine
—— (3S)-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butanamide —— C14H14F3N5O
(3S)-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]butanamide
—— ethyl (6S)-4-[(3,4-dimethylphenoxy)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C22H26N2O4S
ethyl (6S)-4-[(3,4-dimethylphenoxy)methyl]-3-ethyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[(4-fluorophenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H23FN2O5
ethyl (6R)-4-[(4-fluorophenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[(2-fluorophenoxy)methyl]-6-(2-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H23FN2O5
ethyl (6S)-4-[(2-fluorophenoxy)methyl]-6-(2-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H28N2O5
ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (1R,2S)-2-(2,5-difluorophenyl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]cyclopropane-1-carboxamide —— C17H18F2N4O
(1R,2S)-2-(2,5-difluorophenyl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]cyclopropane-1-carboxamide
—— ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C21H24N2O4S
ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[(4-fluorophenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C19H19FN2O4S
ethyl (6R)-4-[(4-fluorophenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[(4-fluorophenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C19H19FN2O4S
ethyl (6S)-4-[(4-fluorophenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— propan-2-yl (6R)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate —— C23H33N3O4
propan-2-yl (6R)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2-fluorophenyl)-4-[(4-methoxyphenoxy)methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H23FN2O5
ethyl (6S)-6-(2-fluorophenyl)-4-[(4-methoxyphenoxy)methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[(2,3-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H28N2O5
ethyl (6S)-4-[(2,3-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— propan-2-yl (6S)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate —— C23H33N3O4
propan-2-yl (6S)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[(2,3-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H28N2O5
ethyl (6R)-4-[(2,3-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2-fluorophenyl)-4-[(4-methoxyphenoxy)methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H23FN2O5
ethyl (6R)-6-(2-fluorophenyl)-4-[(4-methoxyphenoxy)methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2-fluorophenyl)-3-methyl-2-oxo-4-[(2,3,5-trimethylphenoxy)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H27FN2O4
ethyl (6S)-6-(2-fluorophenyl)-3-methyl-2-oxo-4-[(2,3,5-trimethylphenoxy)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-4-[(4-fluorophenoxy)methyl]-6-(2-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H23FN2O5
ethyl (6R)-4-[(4-fluorophenoxy)methyl]-6-(2-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— methyl (6S)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate —— C21H29N3O4
methyl (6S)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2-fluorophenyl)-3-methyl-2-oxo-4-[(2,3,5-trimethylphenoxy)methyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H27FN2O4
ethyl (6R)-6-(2-fluorophenyl)-3-methyl-2-oxo-4-[(2,3,5-trimethylphenoxy)methyl]-1,6-dihydropyrimidine-5-carboxylate
—— methyl (6R)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate —— C21H29N3O4
methyl (6R)-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate
—— [(3S)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-imidazo[1,2-a]pyrazin-8-ylmethanone —— C16H18N6O2
[(3S)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-imidazo[1,2-a]pyrazin-8-ylmethanone
—— (6S)-3-cyclopropyl-6-(4-fluorophenyl)-N,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxamide —— C16H18FN3OS
(6S)-3-cyclopropyl-6-(4-fluorophenyl)-N,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxamide
—— [(3R)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-imidazo[1,2-a]pyrazin-8-ylmethanone —— C16H18N6O2
[(3R)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-imidazo[1,2-a]pyrazin-8-ylmethanone
—— 4-chloro-5-[[(1R,2S)-2-(3-chlorophenyl)cyclopropyl]amino]-2-[5-(trifluoromethyl)pyridin-2-yl]pyridazin-3-one —— C19H13Cl2F3N4O
4-chloro-5-[[(1R,2S)-2-(3-chlorophenyl)cyclopropyl]amino]-2-[5-(trifluoromethyl)pyridin-2-yl]pyridazin-3-one
—— 4-chloro-5-[[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]amino]-2-methylpyridazin-3-one —— C12H14ClN3O2S
4-chloro-5-[[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]amino]-2-methylpyridazin-3-one
—— 4-[[(1S,2R)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile —— C16H15ClN4O2
4-[[(1S,2R)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile
—— 4-[[(1R,2S)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile —— C16H15ClN4O2
4-[[(1R,2S)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile
—— (3R)-4-methylsulfanyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]butan-1-ol —— C17H22N4OS
(3R)-4-methylsulfanyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]butan-1-ol
—— N-[(3R,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]tetrazolo[1,5-b]pyridazin-6-amine —— C15H20N8S
N-[(3R,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]tetrazolo[1,5-b]pyridazin-6-amine
—— (3S)-4-methylsulfanyl-3-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]butan-1-ol —— C16H19N5OS
(3S)-4-methylsulfanyl-3-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]butan-1-ol
—— 4-chloro-5-[[(1R)-3-hydroxy-1-thiophen-2-ylpropyl]amino]-2-methylpyridazin-3-one —— C12H14ClN3O2S
4-chloro-5-[[(1R)-3-hydroxy-1-thiophen-2-ylpropyl]amino]-2-methylpyridazin-3-one
—— 3-[[(1S)-3-hydroxy-1-thiophen-2-ylpropyl]amino]pyrazine-2-carbonitrile —— C12H12N4OS
3-[[(1S)-3-hydroxy-1-thiophen-2-ylpropyl]amino]pyrazine-2-carbonitrile
—— 4-chloro-5-[[(1S)-3-hydroxy-1-thiophen-2-ylpropyl]amino]-2-methylpyridazin-3-one —— C12H14ClN3O2S
4-chloro-5-[[(1S)-3-hydroxy-1-thiophen-2-ylpropyl]amino]-2-methylpyridazin-3-one
—— 4-[[(1S,2S)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile —— C16H15ClN4O2
4-[[(1S,2S)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile
—— 3-amino-N-[(1S,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylpyrazine-2-carboxamide —— C16H24N4O2
3-amino-N-[(1S,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylpyrazine-2-carboxamide
—— 4-[[(1R,2R)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile —— C16H15ClN4O2
4-[[(1R,2R)-2-(3-chlorophenyl)cyclopropyl]amino]-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonitrile
—— N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-pyridin-3-ylquinazolin-4-amine —— C22H18N4O2
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-pyridin-3-ylquinazolin-4-amine
—— 3-[[(1R)-3-hydroxy-1-thiophen-2-ylpropyl]amino]pyrazine-2-carbonitrile —— C12H12N4OS
3-[[(1R)-3-hydroxy-1-thiophen-2-ylpropyl]amino]pyrazine-2-carbonitrile
—— (3R)-3-[(6-chloropyrazin-2-yl)amino]-3-thiophen-2-ylpropan-1-ol —— C11H12ClN3OS
(3R)-3-[(6-chloropyrazin-2-yl)amino]-3-thiophen-2-ylpropan-1-ol
—— (3S)-4-methylsulfanyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]butan-1-ol —— C17H22N4OS
(3S)-4-methylsulfanyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]butan-1-ol
—— (3S)-3-[(6-chloropyrazin-2-yl)amino]-3-thiophen-2-ylpropan-1-ol —— C11H12ClN3OS
(3S)-3-[(6-chloropyrazin-2-yl)amino]-3-thiophen-2-ylpropan-1-ol
—— N-[(1S,5S,6R)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amine —— C19H24N4O
N-[(1S,5S,6R)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amine
—— 4-chloro-5-[[(1S,2R)-2-(3-chlorophenyl)cyclopropyl]amino]-2-[5-(trifluoromethyl)pyridin-2-yl]pyridazin-3-one —— C19H13Cl2F3N4O
4-chloro-5-[[(1S,2R)-2-(3-chlorophenyl)cyclopropyl]amino]-2-[5-(trifluoromethyl)pyridin-2-yl]pyridazin-3-one
—— N-[(1S,5S,6S)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amine —— C19H24N4O
N-[(1S,5S,6S)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amine
—— 3-amino-N-[(1R,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylpyrazine-2-carboxamide —— C16H24N4O2
3-amino-N-[(1R,3R)-3-ethoxyspiro[3.4]octan-1-yl]-N-methylpyrazine-2-carboxamide
—— (3S)-3-[(6-chloropyrazin-2-yl)amino]-4-methylsulfanylbutan-1-ol —— C9H14ClN3OS
(3S)-3-[(6-chloropyrazin-2-yl)amino]-4-methylsulfanylbutan-1-ol