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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— pyrazin-2-yl-[(2R)-2-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C18H18N8O
pyrazin-2-yl-[(2R)-2-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— (3R)-N,N-dimethyl-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide —— C15H21N7O2S
(3R)-N,N-dimethyl-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide
—— (3S)-N,N-dimethyl-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide —— C15H21N7O2S
(3S)-N,N-dimethyl-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide
—— (3R)-N,N-dimethyl-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidine-1-sulfonamide —— C17H24N6O2S
(3R)-N,N-dimethyl-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidine-1-sulfonamide
—— N-(5-methylpyridin-2-yl)-4-[(2R)-1-(oxan-4-yl)pyrrolidin-2-yl]pyrimidin-2-amine —— C19H25N5O
N-(5-methylpyridin-2-yl)-4-[(2R)-1-(oxan-4-yl)pyrrolidin-2-yl]pyrimidin-2-amine
—— (3S)-N,N-dimethyl-3-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide —— C15H21N7O2S
(3S)-N,N-dimethyl-3-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide
—— 6-N-methyl-4-N-[4-[(3S)-1-(quinolin-6-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C24H26N8
6-N-methyl-4-N-[4-[(3S)-1-(quinolin-6-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 4-N-[4-[(3S)-1-benzylsulfonylpiperidin-3-yl]pyrimidin-2-yl]-6-N-methylpyrimidine-4,6-diamine —— C21H25N7O2S
4-N-[4-[(3S)-1-benzylsulfonylpiperidin-3-yl]pyrimidin-2-yl]-6-N-methylpyrimidine-4,6-diamine
—— (3R)-N,N-dimethyl-3-[2-[[3-(trifluoromethyl)pyridin-2-yl]amino]pyrimidin-4-yl]piperidine-1-sulfonamide —— C17H21F3N6O2S
(3R)-N,N-dimethyl-3-[2-[[3-(trifluoromethyl)pyridin-2-yl]amino]pyrimidin-4-yl]piperidine-1-sulfonamide
—— (2S)-N,N-dimethyl-2-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]pyrrolidine-1-sulfonamide —— C16H22N6O2S
(2S)-N,N-dimethyl-2-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]pyrrolidine-1-sulfonamide
—— 4-[(2S)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C19H26N6
4-[(2S)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— N-[4-[(2S)-1-(cyclohexylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C18H25N5S
N-[4-[(2S)-1-(cyclohexylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— 4-[(2S)-1-benzylsulfonylpyrrolidin-2-yl]-N-(5-methylpyridin-2-yl)pyrimidin-2-amine —— C21H23N5O2S
4-[(2S)-1-benzylsulfonylpyrrolidin-2-yl]-N-(5-methylpyridin-2-yl)pyrimidin-2-amine
—— (3R)-N,N-dimethyl-3-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide —— C15H21N7O2S
(3R)-N,N-dimethyl-3-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidine-1-sulfonamide
—— 4-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]piperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C18H22N8
4-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]piperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— pyrazin-2-yl-[(3S)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C18H18N8O
pyrazin-2-yl-[(3S)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 4-[(2S)-1-(3-phenylpropyl)piperidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C22H26N6
4-[(2S)-1-(3-phenylpropyl)piperidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— cyclobutyl-[(2S)-2-[2-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C18H22N6O
cyclobutyl-[(2S)-2-[2-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— pyrazin-2-yl-[(2S)-2-[2-(pyridin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C19H19N7O
pyrazin-2-yl-[(2S)-2-[2-(pyridin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 6-N-methyl-4-N-[4-[(3S)-1-(quinoxalin-6-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C23H25N9
6-N-methyl-4-N-[4-[(3S)-1-(quinoxalin-6-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— cyclobutyl-[(3S)-3-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C18H22N6O
cyclobutyl-[(3S)-3-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 4-[(2S)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C20H22N6O3S
4-[(2S)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— pyrazin-2-yl-[(2S)-2-[2-(pyridin-2-ylamino)pyrimidin-4-yl]pyrrolidin-1-yl]methanone —— C18H17N7O
pyrazin-2-yl-[(2S)-2-[2-(pyridin-2-ylamino)pyrimidin-4-yl]pyrrolidin-1-yl]methanone
—— (2S)-N,N-dimethyl-2-[2-(1,3-thiazol-2-ylamino)pyrimidin-4-yl]pyrrolidine-1-sulfonamide —— C13H18N6O2S2
(2S)-N,N-dimethyl-2-[2-(1,3-thiazol-2-ylamino)pyrimidin-4-yl]pyrrolidine-1-sulfonamide
—— 4-[(2R)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C19H26N6
4-[(2R)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— (3S)-N,N-dimethyl-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidine-1-sulfonamide —— C17H24N6O2S
(3S)-N,N-dimethyl-3-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidine-1-sulfonamide
—— 4-[(2R)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C19H20N6O3S
4-[(2R)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— pyrazin-2-yl-[(2R)-2-[2-(pyridin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C19H19N7O
pyrazin-2-yl-[(2R)-2-[2-(pyridin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 4-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C20H22N6O3S
4-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— N-pyridin-2-yl-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C20H22N6
N-pyridin-2-yl-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 4-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C17H20N8
4-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— 4-[(2S)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C18H17FN6O2S
4-[(2S)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— N-(3-methylpyridin-2-yl)-4-[(3R)-1-methylsulfonylpiperidin-3-yl]pyrimidin-2-amine —— C16H21N5O2S
N-(3-methylpyridin-2-yl)-4-[(3R)-1-methylsulfonylpiperidin-3-yl]pyrimidin-2-amine
—— N-pyrazin-2-yl-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C18H19N7
N-pyrazin-2-yl-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 6-N-methyl-4-N-[4-[(2S)-1-propan-2-ylpyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C16H23N7
6-N-methyl-4-N-[4-[(2S)-1-propan-2-ylpyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 6-N-methyl-4-N-[4-[(3S)-1-(2-phenylethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C22H27N7
6-N-methyl-4-N-[4-[(3S)-1-(2-phenylethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— N-(5-methylpyridin-2-yl)-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H24N6
N-(5-methylpyridin-2-yl)-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 4-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine —— C14H17N5O2S
4-[(2S)-1-methylsulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine
—— N-(5-methylpyridin-2-yl)-4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H24N6
N-(5-methylpyridin-2-yl)-4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— cyclohexyl-[(2R)-2-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C20H26N6O
cyclohexyl-[(2R)-2-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 4-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine —— C14H17N5O2S
4-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine
—— 4-[(3S)-1-(2-methoxyethyl)piperidin-3-yl]-N-(5-methylpyridin-2-yl)pyrimidin-2-amine —— C18H25N5O
4-[(3S)-1-(2-methoxyethyl)piperidin-3-yl]-N-(5-methylpyridin-2-yl)pyrimidin-2-amine
—— N-pyrazin-2-yl-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C19H21N7
N-pyrazin-2-yl-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 4-[(2R)-1-(2-phenylethyl)piperidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C21H24N6
4-[(2R)-1-(2-phenylethyl)piperidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— N-pyridin-2-yl-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C19H20N6
N-pyridin-2-yl-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— N-pyridin-2-yl-4-[(2R)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C19H20N6
N-pyridin-2-yl-4-[(2R)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 6-N-methyl-4-N-[4-[(3R)-1-(2-phenylethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C22H27N7
6-N-methyl-4-N-[4-[(3R)-1-(2-phenylethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 4-[(2R)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C19H20N6O3S
4-[(2R)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— N-(3-methylpyridin-2-yl)-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H24N6
N-(3-methylpyridin-2-yl)-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 6-N-methyl-4-N-[4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C20H24N8
6-N-methyl-4-N-[4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine