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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone —— C20H18FN5O
[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]ethanone —— C17H19FN4O
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]ethanone
—— 5-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one —— C21H20FN5O2
5-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone —— C23H23FN4O2
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone
—— 4-[(2R)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(3-fluorophenyl)pyrimidin-2-amine —— C22H22F2N4O
4-[(2R)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(3-fluorophenyl)pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone —— C17H19FN4O2
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone
—— 2-[4-[2-(Pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol —— C15H20N6O
2-[4-[2-(Pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyrrolidin-1-ylethanone —— C20H24FN5O
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyrrolidin-1-ylethanone
—— 1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C25H28N4O3
1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— [(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone —— C20H18ClN5O
[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone
—— 2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide —— C20H26FN5O
2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide
—— 3-[2-amino-4-[(2S)-1-[2-(4-chlorophenyl)ethyl]pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C23H24ClN5O
3-[2-amino-4-[(2S)-1-[2-(4-chlorophenyl)ethyl]pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone —— C23H23ClN4O2
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-morpholin-4-ylethanone —— C20H24FN5O2
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-morpholin-4-ylethanone
—— [(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C21H21N5O2
[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— 2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide —— C20H26FN5O
2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-diethylacetamide
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C22H20F2N4O2
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 1-[4-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidine-1-carbonyl]piperidin-1-yl]ethanone —— C22H26FN5O2
1-[4-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidine-1-carbonyl]piperidin-1-yl]ethanone
—— 4-[(2R)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine —— C22H22F2N4O
4-[(2R)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-fluorophenyl)ethanone —— C22H20F2N4O
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-fluorophenyl)ethanone
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone —— C22H21ClN4O
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone
—— 3-[2-amino-4-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C23H23N5O2
3-[2-amino-4-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— (2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C17H23N5O3S
(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— [(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C19H19FN6O
[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 1-[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-morpholin-4-ylethanone —— C21H24F3N5O2
1-[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-morpholin-4-ylethanone
—— (2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C16H20FN5O2S
(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— 1-[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone —— C21H20F3N5OS
1-[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone
—— N-pyrimidin-5-yl-4-(1-pyrimidin-2-ylpiperidin-4-yl)pyrimidin-2-amine —— C17H18N8
N-pyrimidin-5-yl-4-(1-pyrimidin-2-ylpiperidin-4-yl)pyrimidin-2-amine
—— 5-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one —— C22H23N5O3
5-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2S)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-hydroxy-2-methylpropan-1-one —— C19H21F3N4O2
1-[(2S)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-hydroxy-2-methylpropan-1-one
—— 4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C19H21N7
4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenoxypropan-1-one —— C23H23FN4O2
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenoxypropan-1-one
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenoxypropan-1-one —— C23H23ClN4O2
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenoxypropan-1-one
—— 4-[(2S)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine —— C22H22F2N4O
4-[(2S)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one —— C23H23ClN4O
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one
—— 5-(3-fluorophenyl)-4-[(2S)-1-(pyridin-2-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H20FN5
5-(3-fluorophenyl)-4-[(2S)-1-(pyridin-2-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C20H18ClN5O
[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— 1-[(2S)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]ethanone —— C17H17F3N4O
1-[(2S)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]ethanone
—— 5-(3-fluorophenyl)-4-[(2R)-1-(pyridin-2-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H20FN5
5-(3-fluorophenyl)-4-[(2R)-1-(pyridin-2-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone —— C21H20FN5O
1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone
—— 4-[(2S)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(3-fluorophenyl)pyrimidin-2-amine —— C22H22F2N4O
4-[(2S)-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-2-yl]-5-(3-fluorophenyl)pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]ethanone —— C17H19FN4O
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]ethanone
—— 5-(3-fluorophenyl)-4-[(2S)-1-(2-methoxyethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C17H21FN4O
5-(3-fluorophenyl)-4-[(2S)-1-(2-methoxyethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone —— C17H19FN4O2
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone
—— 3-[2-amino-4-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C23H23N5O2
3-[2-amino-4-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone —— C18H21FN4O2
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone
—— 3-[2-amino-4-[(2S)-1-(4-fluorobenzoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C22H20FN5O2
3-[2-amino-4-[(2S)-1-(4-fluorobenzoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone —— C24H26N4O3
1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone
—— 1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one —— C24H26N4O2
1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one
—— 5-(4-fluorophenyl)-4-[(2R)-1-(2-phenylethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C22H23FN4
5-(4-fluorophenyl)-4-[(2R)-1-(2-phenylethyl)pyrrolidin-2-yl]pyrimidin-2-amine