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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-diethylpyrrolidine-1-sulfonamide —— C20H30N6O2S
(2R)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-diethylpyrrolidine-1-sulfonamide
—— (2S)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-diethylpyrrolidine-1-sulfonamide —— C20H30N6O2S
(2S)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-diethylpyrrolidine-1-sulfonamide
—— (2R)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C18H26N6O2S
(2R)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-ethyl-N-[(3-fluorophenyl)methyl]acetamide —— C19H19FN4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-ethyl-N-[(3-fluorophenyl)methyl]acetamide
—— N-[(2S)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C18H24N4O5S
N-[(2S)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(R)-phenyl(thiophen-2-yl)methyl]acetamide —— C21H18N4O3S
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(R)-phenyl(thiophen-2-yl)methyl]acetamide
—— (3S)-1-benzyl-3-methyl-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]azepan-2-one —— C24H30N4O2
(3S)-1-benzyl-3-methyl-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]azepan-2-one
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[2-(2-methylphenyl)ethyl]acetamide —— C19H20N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[2-(2-methylphenyl)ethyl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(S)-phenyl(thiophen-2-yl)methyl]acetamide —— C21H18N4O3S
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(S)-phenyl(thiophen-2-yl)methyl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2-methylphenyl)methyl]acetamide —— C18H18N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2-methylphenyl)methyl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2S)-heptan-2-yl]acetamide —— C17H24N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2S)-heptan-2-yl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2-fluorophenyl)methyl]acetamide —— C17H15FN4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2-fluorophenyl)methyl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(1S)-1-cyclopropylethyl]acetamide —— C15H18N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(1S)-1-cyclopropylethyl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-hexylacetamide —— C16H22N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-hexylacetamide
—— N-butyl-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-ethylacetamide —— C16H22N4O3
N-butyl-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-ethylacetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2R)-heptan-2-yl]acetamide —— C17H24N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2R)-heptan-2-yl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-(3-propan-2-yloxypropyl)acetamide —— C16H22N4O4
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-(3-propan-2-yloxypropyl)acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[4-(2-methylbutan-2-yl)cyclohexyl]acetamide —— C21H30N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[4-(2-methylbutan-2-yl)cyclohexyl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2S)-octan-2-yl]acetamide —— C18H26N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2S)-octan-2-yl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-cyclohexyl-N-[(4-fluorophenyl)methyl]acetamide —— C23H25FN4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-cyclohexyl-N-[(4-fluorophenyl)methyl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2S)-2-ethylhexyl]acetamide —— C18H26N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2S)-2-ethylhexyl]acetamide
—— N-benzyl-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-(furan-2-ylmethyl)acetamide —— C22H20N4O4
N-benzyl-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-(furan-2-ylmethyl)acetamide
—— (3R)-1-benzyl-3-methyl-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]azepan-2-one —— C24H30N4O2
(3R)-1-benzyl-3-methyl-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]azepan-2-one
—— (2,4-dimethylpyrimidin-5-yl)-[(3S)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C22H24FN5O2
(2,4-dimethylpyrimidin-5-yl)-[(3S)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— N-[(5-chlorothiophen-2-yl)methyl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-ethylacetamide —— C17H17ClN4O3S
N-[(5-chlorothiophen-2-yl)methyl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-ethylacetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[2-(2-fluorophenyl)ethyl]acetamide —— C18H17FN4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[2-(2-fluorophenyl)ethyl]acetamide
—— N,N-bis[(2S)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)acetamide —— C18H26N4O3
N,N-bis[(2S)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)acetamide
—— [(3S)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone —— C21H22F2N6O2
[(3S)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone
—— N-[(2R)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide —— C18H24N4O5S
N-[(2R)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2-fluorophenyl)methyl]-N-methylacetamide —— C18H17FN4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(2-fluorophenyl)methyl]-N-methylacetamide
—— N-[(2R)-butan-2-yl]-N-[(2S)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)acetamide —— C18H26N4O3
N-[(2R)-butan-2-yl]-N-[(2S)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N,N-dipropylacetamide —— C16H22N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N,N-dipropylacetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-cyclohexyl-N-propan-2-ylacetamide —— C19H26N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-cyclohexyl-N-propan-2-ylacetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-methyl-N-(thiophen-3-ylmethyl)acetamide —— C16H16N4O3S
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-methyl-N-(thiophen-3-ylmethyl)acetamide
—— N-[(2R)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C18H24N4O5S
N-[(2R)-butan-2-yl]-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide —— C18H24N4O5S
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(4-methylphenyl)methyl]-N-propylacetamide —— C21H24N4O3
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(4-methylphenyl)methyl]-N-propylacetamide
—— 2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide —— C18H24N4O5S
2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide
—— (2,4-dimethylpyrimidin-5-yl)-[(3R)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C22H24FN5O2
(2,4-dimethylpyrimidin-5-yl)-[(3R)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— [(3R)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone —— C21H22F2N6O2
[(3R)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone
—— [2-(dimethylamino)pyrimidin-5-yl]-[(3S)-3-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C22H25FN6O2
[2-(dimethylamino)pyrimidin-5-yl]-[(3S)-3-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— (2-amino-4-methylpyrimidin-5-yl)-[(3S)-3-[5-[2-(4-propan-2-ylphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C24H30N6O2
(2-amino-4-methylpyrimidin-5-yl)-[(3S)-3-[5-[2-(4-propan-2-ylphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— [2-(dimethylamino)pyrimidin-5-yl]-[(3R)-3-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C22H25FN6O2
[2-(dimethylamino)pyrimidin-5-yl]-[(3R)-3-[5-[2-(3-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— [(3S)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C22H25N5O3
[(3S)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3R)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C22H25N5O3
[(3R)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3R)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C21H22ClN5O2
[(3R)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3S)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C21H22ClN5O2
[(3S)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-[(2-chlorophenyl)methylsulfanyl]acetate —— C16H13ClN2O3S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-[(2-chlorophenyl)methylsulfanyl]acetate
—— [(3S)-3-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C21H22FN5O2
[(3S)-3-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3R)-3-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C21H22FN5O2
[(3R)-3-[5-[2-(2-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]-(5-methylpyrazin-2-yl)methanone