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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(3S)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]-(4-propylpyrimidin-5-yl)methanone —— C22H29N3O
[(3S)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]-(4-propylpyrimidin-5-yl)methanone
—— (3R)-1-(7-acetyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide —— C20H24N6O2
(3R)-1-(7-acetyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide
—— 5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C20H25FN4O2
5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— (3S)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-amine —— C16H20N6
(3S)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-amine
—— [(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(4-methylpyrimidin-5-yl)methanone —— C21H27FN4O
[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(4-methylpyrimidin-5-yl)methanone
—— [(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methoxypyrimidin-5-yl)methanone —— C21H27FN4O2
[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methoxypyrimidin-5-yl)methanone
—— [(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methoxypyrimidin-5-yl)methanone —— C21H27FN4O2
[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methoxypyrimidin-5-yl)methanone
—— [(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(4-methylpyrimidin-5-yl)methanone —— C21H27FN4O
[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(4-methylpyrimidin-5-yl)methanone
—— (3R)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-amine —— C16H20N6
(3R)-1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-amine
—— 4-cyclobutyl-6-methyl-N-[(3S)-oxolan-3-yl]pyrimidin-2-amine —— C13H19N3O
4-cyclobutyl-6-methyl-N-[(3S)-oxolan-3-yl]pyrimidin-2-amine
—— (3R)-N,N-diethyl-1-[6-(2-methoxyphenyl)pyridazin-3-yl]pyrrolidin-3-amine —— C19H26N4O
(3R)-N,N-diethyl-1-[6-(2-methoxyphenyl)pyridazin-3-yl]pyrrolidin-3-amine
—— 4-cyclobutyl-6-methyl-N-[(3R)-oxolan-3-yl]pyrimidin-2-amine —— C13H19N3O
4-cyclobutyl-6-methyl-N-[(3R)-oxolan-3-yl]pyrimidin-2-amine
—— 5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C20H25FN4O2
5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— 4-[1-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]imidazol-2-yl]-2-propan-2-ylpyrimidine —— C18H24N6
4-[1-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]imidazol-2-yl]-2-propan-2-ylpyrimidine
—— 1-[4-[(3S)-3-methoxypiperidin-1-yl]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H25N5O2
1-[4-[(3S)-3-methoxypiperidin-1-yl]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 4-[1-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]imidazol-2-yl]-2-propan-2-ylpyrimidine —— C18H24N6
4-[1-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]imidazol-2-yl]-2-propan-2-ylpyrimidine
—— N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C14H21F3N4
N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 4-cyclopentyl-N-[(R)-cyclopropyl-(3-methylpyridin-2-yl)methyl]pyrimidin-2-amine —— C19H24N4
4-cyclopentyl-N-[(R)-cyclopropyl-(3-methylpyridin-2-yl)methyl]pyrimidin-2-amine
—— (3R)-4-[(4-fluorophenyl)methyl]-1-(5-methylpyrazine-2-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C21H25FN4O2
(3R)-4-[(4-fluorophenyl)methyl]-1-(5-methylpyrazine-2-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C14H21F3N4
N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— (3S)-4-[(4-fluorophenyl)methyl]-1-(2-methylpyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C21H25FN4O2
(3S)-4-[(4-fluorophenyl)methyl]-1-(2-methylpyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— 4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C17H22N4O
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— 1-[4-[(3R)-3-methoxypiperidin-1-yl]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H25N5O2
1-[4-[(3R)-3-methoxypiperidin-1-yl]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 4-cyclobutyl-N-[(R)-cyclopropyl-(3-methylpyridin-2-yl)methyl]-6-methylpyrimidin-2-amine —— C19H24N4
4-cyclobutyl-N-[(R)-cyclopropyl-(3-methylpyridin-2-yl)methyl]-6-methylpyrimidin-2-amine
—— 4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C17H22N4O
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (3R)-4-benzyl-1-(2,4-dimethylpyrimidine-5-carbonyl)-3-ethyl-1,4-diazepan-5-one —— C21H26N4O2
(3R)-4-benzyl-1-(2,4-dimethylpyrimidine-5-carbonyl)-3-ethyl-1,4-diazepan-5-one
—— 4-cyclobutyl-N-[(S)-cyclopropyl-(3-methylpyridin-2-yl)methyl]-6-methylpyrimidin-2-amine —— C19H24N4
4-cyclobutyl-N-[(S)-cyclopropyl-(3-methylpyridin-2-yl)methyl]-6-methylpyrimidin-2-amine
—— 4-[(1R)-2-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]-1-hydroxyethyl]phenol —— C19H20N4O2
4-[(1R)-2-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]-1-hydroxyethyl]phenol
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrimidin-2-amine —— C19H24N6
4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrimidin-2-amine
—— (3R)-4-[(4-fluorophenyl)methyl]-1-(2-methylpyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C21H25FN4O2
(3R)-4-[(4-fluorophenyl)methyl]-1-(2-methylpyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— 4-[(1S)-2-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]-1-hydroxyethyl]phenol —— C19H20N4O2
4-[(1S)-2-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]-1-hydroxyethyl]phenol
—— 4-cyclopentyl-N-[(S)-cyclopropyl-(3-methylpyridin-2-yl)methyl]pyrimidin-2-amine —— C19H24N4
4-cyclopentyl-N-[(S)-cyclopropyl-(3-methylpyridin-2-yl)methyl]pyrimidin-2-amine
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrimidin-2-amine —— C19H24N6
4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrimidin-2-amine
—— (3R)-4-benzyl-3-ethyl-1-[2-(methylamino)pyrimidine-5-carbonyl]-1,4-diazepan-5-one —— C20H25N5O2
(3R)-4-benzyl-3-ethyl-1-[2-(methylamino)pyrimidine-5-carbonyl]-1,4-diazepan-5-one
—— 1-[4-[[(2S)-1-methoxypropan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H23N5O2
1-[4-[[(2S)-1-methoxypropan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 5-[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— (3S)-4-benzyl-3-ethyl-1-[2-(methylamino)pyrimidine-5-carbonyl]-1,4-diazepan-5-one —— C20H25N5O2
(3S)-4-benzyl-3-ethyl-1-[2-(methylamino)pyrimidine-5-carbonyl]-1,4-diazepan-5-one
—— N-[[(3S)-1,1-dioxothiolan-3-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine —— C16H19N3O3S
N-[[(3S)-1,1-dioxothiolan-3-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine
—— 5-[[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine —— C20H26F2N4
5-[[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine
—— 1-[4-[[(2R)-1-methoxypropan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H23N5O2
1-[4-[[(2R)-1-methoxypropan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 5-[(2R)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C16H23N3O2
5-[(2R)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 3-[2-[(2S)-piperidin-2-yl]ethyl]-5-thieno[2,3-d]pyrimidin-4-ylphenol —— C19H21N3OS
3-[2-[(2S)-piperidin-2-yl]ethyl]-5-thieno[2,3-d]pyrimidin-4-ylphenol
—— 6-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione —— C20H25FN4O3
6-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione
—— N-[[(3R)-1,1-dioxothiolan-3-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine —— C16H19N3O3S
N-[[(3R)-1,1-dioxothiolan-3-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine
—— 5-[(2S)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C16H23N3O2
5-[(2S)-2-butyl-2,5-dihydropyrrole-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(3S)-3-imidazol-1-ylbutyl]pyrimidin-2-amine —— C18H22N6
4-(2,6-dimethylpyridin-3-yl)-N-[(3S)-3-imidazol-1-ylbutyl]pyrimidin-2-amine
—— 4-[(2S)-2-methylpyrrolidin-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine —— C17H21N5
4-[(2S)-2-methylpyrrolidin-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine
—— 5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C20H32N4O2
5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— [2-[2-(2-Methylanilino)-2-oxoethyl]-1,3-thiazol-4-yl]methyl 3-aminopyrazine-2-carboxylate —— C18H17N5O3S
[2-[2-(2-Methylanilino)-2-oxoethyl]-1,3-thiazol-4-yl]methyl 3-aminopyrazine-2-carboxylate